IT1118186B - Procedimento per la produzione di derivati dell'ossadiazolo quali agenti contro protozoi - Google Patents

Procedimento per la produzione di derivati dell'ossadiazolo quali agenti contro protozoi

Info

Publication number
IT1118186B
IT1118186B IT49742/79A IT4974279A IT1118186B IT 1118186 B IT1118186 B IT 1118186B IT 49742/79 A IT49742/79 A IT 49742/79A IT 4974279 A IT4974279 A IT 4974279A IT 1118186 B IT1118186 B IT 1118186B
Authority
IT
Italy
Prior art keywords
protozoi
procedure
production
oxadiazole derivatives
agents against
Prior art date
Application number
IT49742/79A
Other languages
English (en)
Other versions
IT7949742A0 (it
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wellcome Found filed Critical Wellcome Found
Publication of IT7949742A0 publication Critical patent/IT7949742A0/it
Application granted granted Critical
Publication of IT1118186B publication Critical patent/IT1118186B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D271/00Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/061,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/50Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
    • C07C323/51Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/60Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton with the carbon atom of at least one of the carboxyl groups bound to nitrogen atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IT49742/79A 1978-07-13 1979-07-12 Procedimento per la produzione di derivati dell'ossadiazolo quali agenti contro protozoi IT1118186B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB7829818 1978-07-13

Publications (2)

Publication Number Publication Date
IT7949742A0 IT7949742A0 (it) 1979-07-12
IT1118186B true IT1118186B (it) 1986-02-24

Family

ID=10498430

Family Applications (1)

Application Number Title Priority Date Filing Date
IT49742/79A IT1118186B (it) 1978-07-13 1979-07-12 Procedimento per la produzione di derivati dell'ossadiazolo quali agenti contro protozoi

Country Status (6)

Country Link
US (1) US4294842A (it)
EP (1) EP0007529B1 (it)
JP (1) JPS5515479A (it)
DE (1) DE2965905D1 (it)
DK (1) DK294579A (it)
IT (1) IT1118186B (it)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1118186B (it) * 1978-07-13 1986-02-24 Wellcome Found Procedimento per la produzione di derivati dell'ossadiazolo quali agenti contro protozoi
DE4232418A1 (de) * 1992-09-28 1994-03-31 Bayer Ag Verwendung von substituierten 1,2,4-Oxadiazolderivaten zur Bekämpfung von Endoparasiten, neue substituierte 1,2,4-Oxadiazolderivate und Verfahren zu ihrer Herstellung
DE4401108A1 (de) * 1994-01-17 1995-07-20 Bayer Ag 1,2,4-Oxadiazol-Derivate
MX2018014032A (es) 2017-03-20 2019-08-21 Forma Therapeutics Inc Composiciones de pirrolopirrol como activadores de piruvato cinasa (pkr).
CN113226356A (zh) 2018-09-19 2021-08-06 福马治疗股份有限公司 活化丙酮酸激酶r
EP3853206B1 (en) 2018-09-19 2024-04-10 Novo Nordisk Health Care AG Treating sickle cell disease with a pyruvate kinase r activating compound

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2219841A1 (de) * 1972-04-22 1973-10-25 Basf Ag Verfahren zur herstellung von 2-(oalkylthiophenyl)-1,3-diazacycloalkenhydrohalogeniden
US3897447A (en) * 1973-04-30 1975-07-29 Merck & Co Inc Anthelmintic 1,2,4-oxadiazolines
FR2307531A1 (fr) * 1975-04-16 1976-11-12 Cassenne Lab Sa Nouveaux derives de l'oxadiazole et leurs sels, procede de preparation et application a titre de medicaments
FR2347926A2 (fr) * 1976-04-15 1977-11-10 Cassenne Lab Sa Nouveaux derives de l'oxadiazole et leurs sels, procede de preparation et application a titre de medicaments
IT1118186B (it) * 1978-07-13 1986-02-24 Wellcome Found Procedimento per la produzione di derivati dell'ossadiazolo quali agenti contro protozoi

Also Published As

Publication number Publication date
DE2965905D1 (en) 1983-08-25
EP0007529A1 (en) 1980-02-06
EP0007529B1 (en) 1983-07-20
DK294579A (da) 1980-01-14
IT7949742A0 (it) 1979-07-12
US4294842A (en) 1981-10-13
JPS5515479A (en) 1980-02-02

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