IN2014MN00875A - - Google Patents

Info

Publication number
IN2014MN00875A
IN2014MN00875A IN875MUN2014A IN2014MN00875A IN 2014MN00875 A IN2014MN00875 A IN 2014MN00875A IN 875MUN2014 A IN875MUN2014 A IN 875MUN2014A IN 2014MN00875 A IN2014MN00875 A IN 2014MN00875A
Authority
IN
India
Prior art keywords
fluoropegylated
aryl
relates
provide access
improved methods
Prior art date
Application number
Inventor
Franz Meier
Keith Graham
Original Assignee
Piramal Imaging Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Piramal Imaging Sa filed Critical Piramal Imaging Sa
Publication of IN2014MN00875A publication Critical patent/IN2014MN00875A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/63—One oxygen atom
    • C07D213/64—One oxygen atom attached in position 2 or 6
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B59/00—Introduction of isotopes of elements into organic compounds ; Labelled organic compounds per se
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C213/00—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton
    • C07C213/08—Preparation of compounds containing amino and hydroxy, amino and etherified hydroxy or amino and esterified hydroxy groups bound to the same carbon skeleton by reactions not involving the formation of amino groups, hydroxy groups or etherified or esterified hydroxy groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/06—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom containing only hydrogen and carbon atoms in addition to the ring nitrogen atom
    • C07D213/16—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom containing only hydrogen and carbon atoms in addition to the ring nitrogen atom containing only one pyridine ring
    • C07D213/18—Salts thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/05—Isotopically modified compounds, e.g. labelled

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Pyridine Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

This invention relates to improved methods which provide access [F 18]fluoropegylated (aryl/heteroaryl vinyl) phenyl methyl amine derivatives.
IN875MUN2014 2011-10-19 2012-10-18 IN2014MN00875A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP11075236 2011-10-19
PCT/EP2012/070669 WO2013057199A1 (en) 2011-10-19 2012-10-18 IMPROVED METHOD FOR PRODUCTION OF F-18 LABELED Aß LIGANDS

Publications (1)

Publication Number Publication Date
IN2014MN00875A true IN2014MN00875A (en) 2015-04-17

Family

ID=47022716

Family Applications (1)

Application Number Title Priority Date Filing Date
IN875MUN2014 IN2014MN00875A (en) 2011-10-19 2012-10-18

Country Status (11)

Country Link
US (1) US20140243533A1 (en)
EP (1) EP2768790A1 (en)
JP (1) JP2015501305A (en)
AU (1) AU2012324940A1 (en)
BR (1) BR112014009013A2 (en)
CA (1) CA2852840A1 (en)
IL (1) IL231964A0 (en)
IN (1) IN2014MN00875A (en)
MX (1) MX2014004274A (en)
SG (1) SG11201401640QA (en)
WO (1) WO2013057199A1 (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN116794184B (en) * 2023-06-26 2024-02-09 天津键凯科技有限公司 Method for detecting polyethylene glycol with single polymerization degree and homologous impurities

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100789847B1 (en) 2004-12-15 2007-12-28 (주)퓨쳐켐 A Preparation Method of Organo Fluoro Compounds in Alcohol Solvents
SG194363A1 (en) 2004-12-17 2013-11-29 Univ Pennsylvania Stilbene derivatives and their use for binding and imaging amyloid plaques
SI1999109T1 (en) 2006-03-30 2012-04-30 Univ Pennsylvania Styrylpyridine derivatives and their use for binding and imaging amyloid plaques
JP5717650B2 (en) 2008-12-31 2015-05-13 アビド・ラジオファーマシューティカルス・インコーポレイテッドＡｖｉｄ Ｒａｄｉｏｐｈａｒｍａｃｅｕｔｉｃａｌｓ， Ｉｎｃ． Synthesis of 18F-radiolabeled styrylpyridine and its stable pharmaceutical composition from tosylate precursor
CN103328011A (en) * 2010-06-04 2013-09-25 皮拉马影像股份公司 Method for production of F-18 labeled amyloid beta ligand
TWI504414B (en) * 2010-06-04 2015-10-21 Bayer Schering Pharma Ag Method for production of f-18 labeled aβ ligands
KR101761451B1 (en) * 2010-06-04 2017-07-25 피라말 이미징 에스에이 Method for production of f-18 labeled amyloid beta ligands
CA2801525A1 (en) * 2010-06-04 2011-12-08 Piramal Imaging Sa Method for production of f-18 labeled amyloid beta ligands
SG188444A1 (en) * 2010-09-09 2013-04-30 Piramal Imaging Sa Method for rapid preparation of suitable [18f]fluoride for nucleophilic [18f]fluorination.
CN108218650A (en) * 2010-12-29 2018-06-29 通用电气健康护理有限公司 Elute solution

Also Published As

Publication number Publication date
US20140243533A1 (en) 2014-08-28
SG11201401640QA (en) 2014-07-30
BR112014009013A2 (en) 2017-05-02
CA2852840A1 (en) 2013-04-25
MX2014004274A (en) 2014-07-09
EP2768790A1 (en) 2014-08-27
IL231964A0 (en) 2014-05-28
JP2015501305A (en) 2015-01-15
AU2012324940A1 (en) 2014-04-17
WO2013057199A1 (en) 2013-04-25

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