IN2014DN09053A - - Google Patents

Download PDF

Info

Publication number
IN2014DN09053A
IN2014DN09053A IN9053DEN2014A IN2014DN09053A IN 2014DN09053 A IN2014DN09053 A IN 2014DN09053A IN 9053DEN2014 A IN9053DEN2014 A IN 9053DEN2014A IN 2014DN09053 A IN2014DN09053 A IN 2014DN09053A
Authority
IN
India
Prior art keywords
tetrahydrolactoylpterin
lactoylpterin
sepiapterin
reaction formula
good yield
Prior art date
Application number
Other languages
English (en)
Inventor
Hiroshi Yoshino
Taichi Komoda
Yuichi Shiro
Shunichi Murata
Shizuaki Murata
Yasuhiro Kuroda
Original Assignee
Shiratori Pharm
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shiratori Pharm filed Critical Shiratori Pharm
Publication of IN2014DN09053A publication Critical patent/IN2014DN09053A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D475/00Heterocyclic compounds containing pteridine ring systems
    • C07D475/02Heterocyclic compounds containing pteridine ring systems with an oxygen atom directly attached in position 4
    • C07D475/04Heterocyclic compounds containing pteridine ring systems with an oxygen atom directly attached in position 4 with a nitrogen atom directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
IN9053DEN2014 2012-05-07 2013-05-07 IN2014DN09053A (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2012105758 2012-05-07
JP2012247255 2012-11-09
PCT/JP2013/062817 WO2013168693A1 (fr) 2012-05-07 2013-05-07 Procédé de production de sépiaptérine et de tétrahydrolactoylptérine

Publications (1)

Publication Number Publication Date
IN2014DN09053A true IN2014DN09053A (fr) 2015-05-22

Family

ID=49550728

Family Applications (1)

Application Number Title Priority Date Filing Date
IN9053DEN2014 IN2014DN09053A (fr) 2012-05-07 2013-05-07

Country Status (7)

Country Link
US (1) US9181254B2 (fr)
EP (1) EP2848619B1 (fr)
JP (1) JP6084967B2 (fr)
CN (1) CN104736539B (fr)
ES (1) ES2681345T3 (fr)
IN (1) IN2014DN09053A (fr)
WO (1) WO2013168693A1 (fr)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20130197000A1 (en) 2010-04-22 2013-08-01 Nihon University Drug and food/drink for preventing or improving cerebral dysfunction
JP6809781B2 (ja) * 2015-11-18 2021-01-06 白鳥製薬株式会社 プテリン誘導体又はその塩
WO2018102314A1 (fr) 2016-11-29 2018-06-07 Censa Pharmaceuticals Inc. Forme polymorphe de sépiaptérine
BR112019010222A8 (pt) * 2016-11-29 2022-11-22 Censa Pharmaceuticals Inc Polimorfos de sepiapterina e sais dos mesmos
CA3073957A1 (fr) 2017-09-01 2019-03-07 Censa Pharmaceuticals Inc. Composition pharmaceutique comprenant de la sepiapterine et ses utilisations
WO2019232120A1 (fr) * 2018-05-30 2019-12-05 Censa Pharmaceuticals Inc. Sels pharmaceutiquement acceptables de sépiaptérine
WO2019232130A1 (fr) 2018-05-30 2019-12-05 Censa Pharmaceuticals Inc. Procédés pour augmenter l'exposition au plasma de sépiaptérine

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4713454A (en) 1985-01-28 1987-12-15 Shiratori Pharmaceutical Co., Ltd. Preparation process of (6R)-tetrahydro-L-biopterin
JPS61172877A (ja) 1985-01-28 1986-08-04 Shiratori Seiyaku Kk (6r)−テトラヒドロ−l−バイオプテリンの製造方法
EP1776364A2 (fr) 2003-11-17 2007-04-25 BioMarin Pharmaceutical Inc. Procedes de preparation de tetrahydrobiopterine et d'analogues de la tetrahydrobiopterine
JP2011011976A (ja) 2007-10-10 2011-01-20 Shiratori Pharmaceutical Co Ltd プテリジン化合物及びl−ビオプテリンの製造方法
US20130197000A1 (en) 2010-04-22 2013-08-01 Nihon University Drug and food/drink for preventing or improving cerebral dysfunction

Also Published As

Publication number Publication date
WO2013168693A1 (fr) 2013-11-14
US9181254B2 (en) 2015-11-10
EP2848619A4 (fr) 2015-11-04
JPWO2013168693A1 (ja) 2016-01-07
EP2848619A1 (fr) 2015-03-18
ES2681345T3 (es) 2018-09-12
JP6084967B2 (ja) 2017-02-22
CN104736539B (zh) 2017-09-01
EP2848619B1 (fr) 2018-07-11
CN104736539A (zh) 2015-06-24
US20150119574A1 (en) 2015-04-30

Similar Documents

Publication Publication Date Title
MX2015002616A (es) Sintesis de bis(fluorosulfonil)imida.
MX353553B (es) Metodo para producir derivados de 4,4-difluoro-3,4-dihidroisoquino lina.
IN2014DN09053A (fr)
AP3450A (en) Process for the synthesis of methanol
MX2015002487A (es) Proceso para la preparacion de teneligliptina.
WO2015008218A3 (fr) Procédé pour la préparation de suvorexant et intermédiaires utiles pour la synthèse de suvorexant
MY192466A (en) Processes for the preparation of an apoptosis-inducing agent
IN2015DN01061A (fr)
PH12015501807A1 (en) Vortioxetine manufacturing process
MX2015007645A (es) Cyanobacterium sp. para produccion de compuestos.
MX344858B (es) Nuevo procedimiento para la síntesis de rifaximina y una nueva forma pseudocristalina de rifaximina obtenida con el mismo.
MX362689B (es) Procedimiento de preparacion de derivados de acido 3,5-bis(fluoroalquil)pirazol-4-carboxilico y 3,5-bis(fluoroalquil) pirazoles.
MX2016005496A (es) Sintesis de fluorotrifluorometilsulfonil-imida.
UA119435C2 (uk) Об'єднаний спосіб одержання метанолу і метилацетату
IN2014DN06192A (fr)
NZ720106A (en) A process for the preparation of regadenoson
MX2015013589A (es) Proceso e intermediario para la preparacion de pregabalina.
PH12015502121A1 (en) Novel processes for producing sovaprevir
MX343856B (es) Procedimiento para la preparación de derivados 1-h-pirrolidin-2,4-diona.
MX2014003936A (es) Procedimiento para preparar ditiina-tetracarboximidas.
EP2714766A4 (fr) Procédé de production de polymères faisant appel à des réactions de couplage
MX2013002395A (es) Procedimiento de preparacion de ditiin-tetracarboximidas.
MY156773A (en) Preparing ether carboxylates
MX2015017747A (es) Proceso para producir 2-fenil-1, 3-benzoxazoles.
PH12014501760A1 (en) Method for stereoselective synthesis of 1,4-protected 9-hydroxy-5-oxo-1,4-diaza-spiro[5.5]undecanes