IN2013MU00646A - - Google Patents

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Publication number
IN2013MU00646A
IN2013MU00646A IN646MU2013A IN2013MU00646A IN 2013MU00646 A IN2013MU00646 A IN 2013MU00646A IN 646MU2013 A IN646MU2013 A IN 646MU2013A IN 2013MU00646 A IN2013MU00646 A IN 2013MU00646A
Authority
IN
India
Prior art keywords
preparation
present
crystalline form
provides novel
endoxifen
Prior art date
Application number
Other languages
English (en)
Inventor
Jagdish Desai Sanjay
Dinkarrai Desai Brijesh
Viththal Guna Jayesh
Chandulal Patel Sunil
Original Assignee
Intas Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Intas Pharmaceuticals Ltd filed Critical Intas Pharmaceuticals Ltd
Priority to IN646MU2013 priority Critical patent/IN2013MU00646A/en
Priority to PCT/IN2014/000136 priority patent/WO2014141292A2/en
Publication of IN2013MU00646A publication Critical patent/IN2013MU00646A/en

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C217/00Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton
    • C07C217/02Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C217/04Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
    • C07C217/06Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one etherified hydroxy group and one amino group bound to the carbon skeleton, which is not further substituted
    • C07C217/14Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one etherified hydroxy group and one amino group bound to the carbon skeleton, which is not further substituted the oxygen atom of the etherified hydroxy group being further bound to a carbon atom of a six-membered aromatic ring
    • C07C217/18Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one etherified hydroxy group and one amino group bound to the carbon skeleton, which is not further substituted the oxygen atom of the etherified hydroxy group being further bound to a carbon atom of a six-membered aromatic ring the six-membered aromatic ring or condensed ring system containing that ring being further substituted
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
IN646MU2013 2013-03-04 2014-03-03 IN2013MU00646A (ru)

Priority Applications (2)

Application Number Priority Date Filing Date Title
IN646MU2013 IN2013MU00646A (ru) 2013-03-04 2014-03-03
PCT/IN2014/000136 WO2014141292A2 (en) 2013-03-04 2014-03-03 Endoxifen citrate polymorph and process for preparing the same

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IN646MU2013 IN2013MU00646A (ru) 2013-03-04 2014-03-03

Publications (1)

Publication Number Publication Date
IN2013MU00646A true IN2013MU00646A (ru) 2015-06-26

Family

ID=51538243

Family Applications (1)

Application Number Title Priority Date Filing Date
IN646MU2013 IN2013MU00646A (ru) 2013-03-04 2014-03-03

Country Status (2)

Country Link
IN (1) IN2013MU00646A (ru)
WO (1) WO2014141292A2 (ru)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10087191B2 (en) 2015-06-16 2018-10-02 Jiangsu Hengrui Medicine Co., Ltd. Piperidine derivative and preparation method and pharmaceutical use thereof
US10398689B2 (en) 2015-12-22 2019-09-03 Jiangsu Hengrui Medicine Co., Ltd. Benzopiperidine derivative, preparation method thereof and medical use thereof
CA3073836A1 (en) 2017-09-11 2019-03-14 Atossa Therapeutics, Inc. Methods for making and using endoxifen
AU2018369091B2 (en) 2017-11-14 2021-02-18 Kind Pharmaceutical Heterocyclic compound and application thereof in medicine
CN114746424B (zh) 2020-01-10 2023-06-16 江苏恒瑞医药股份有限公司 三环四氢异喹啉类衍生物、其制备方法及其在医药上的应用
CN115484941A (zh) * 2020-04-10 2022-12-16 金纳药业公司 因多昔芬用于治疗双相i型障碍
CA3177266A1 (en) * 2020-04-10 2021-10-14 Jina Pharmaceuticals, Inc. Endoxifen for the treatment of bipolar i disorder
AU2022307207A1 (en) 2021-07-09 2024-02-15 Jiangsu Hengrui Pharmaceuticals Co., Ltd. Salt types of tricyclic tetrahydro isoquinoline derivative
WO2023137044A2 (en) 2022-01-12 2023-07-20 Atossa Therapeutics, Inc. Compositions of (z)-endoxifen and methods of enrichment thereof

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW593256B (en) * 1999-11-16 2004-06-21 Hormos Medical Oy Ltd Triphenylalkene derivatives and their use as selective estrogen receptor modulators
US20090291134A1 (en) * 2006-11-21 2009-11-26 Jina Pharmaceuticals, Inc. Endoxifen methods and compositions in the treatment of psychiatric and neurodegenerative diseases
WO2009120999A2 (en) * 2008-03-28 2009-10-01 Olema Pharmaceuticals, Inc. Use of an endoxifen prodrug for treatment of breast cancer
KR101308258B1 (ko) * 2010-10-15 2013-09-13 씨제이제일제당 (주) 엔독시펜의 신규한 제조 방법

Also Published As

Publication number Publication date
WO2014141292A3 (en) 2014-12-24
WO2014141292A2 (en) 2014-09-18

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