IN2012DE00082A - - Google Patents

Info

Publication number
IN2012DE00082A
IN2012DE00082A IN82DE2012A IN2012DE00082A IN 2012DE00082 A IN2012DE00082 A IN 2012DE00082A IN 82DE2012 A IN82DE2012 A IN 82DE2012A IN 2012DE00082 A IN2012DE00082 A IN 2012DE00082A
Authority
IN
India
Prior art keywords
synthesis
relates
hiv protease
synazido
sequinavirvia
Prior art date
Application number
Other languages
English (en)
Inventor
Khanderao Gadakh Sunita
Santhosh Rekula Reddy
Sudalai Arumugam
Original Assignee
Council Scient Ind Res
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Council Scient Ind Res filed Critical Council Scient Ind Res
Priority to PCT/IN2013/000021 priority Critical patent/WO2013105118A1/en
Priority to IN82DE2012 priority patent/IN2012DE00082A/en
Priority to US14/371,466 priority patent/US9233943B2/en
Publication of IN2012DE00082A publication Critical patent/IN2012DE00082A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D301/00Preparation of oxiranes
    • C07D301/02Synthesis of the oxirane ring
    • C07D301/03Synthesis of the oxirane ring by oxidation of unsaturated compounds, or of mixtures of unsaturated and saturated compounds
    • C07D301/14Synthesis of the oxirane ring by oxidation of unsaturated compounds, or of mixtures of unsaturated and saturated compounds with organic peracids, or salts, anhydrides or esters thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C247/00Compounds containing azido groups
    • C07C247/02Compounds containing azido groups with azido groups bound to acyclic carbon atoms of a carbon skeleton
    • C07C247/04Compounds containing azido groups with azido groups bound to acyclic carbon atoms of a carbon skeleton being saturated
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D301/00Preparation of oxiranes
    • C07D301/02Synthesis of the oxirane ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/04Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D307/18Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D307/20Oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D493/00Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/02Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
    • C07D493/04Ortho-condensed systems
IN82DE2012 2012-01-10 2013-01-10 IN2012DE00082A (US06559137-20030506-C00166.png)

Priority Applications (3)

Application Number Priority Date Filing Date Title
PCT/IN2013/000021 WO2013105118A1 (en) 2012-01-10 2013-01-10 A process for synthesis of syn azido epoxide and its use as intermediate the synthesis of amprenavir & saquinavir
IN82DE2012 IN2012DE00082A (US06559137-20030506-C00166.png) 2012-01-10 2013-01-10
US14/371,466 US9233943B2 (en) 2012-01-10 2013-01-10 Process for synthesis of syn azido epdxide and its use as intermediate for the synthesis of amprenavir and saquinavir

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IN82DE2012 IN2012DE00082A (US06559137-20030506-C00166.png) 2012-01-10 2013-01-10

Publications (1)

Publication Number Publication Date
IN2012DE00082A true IN2012DE00082A (US06559137-20030506-C00166.png) 2015-05-01

Family

ID=47750776

Family Applications (1)

Application Number Title Priority Date Filing Date
IN82DE2012 IN2012DE00082A (US06559137-20030506-C00166.png) 2012-01-10 2013-01-10

Country Status (3)

Country Link
US (1) US9233943B2 (US06559137-20030506-C00166.png)
IN (1) IN2012DE00082A (US06559137-20030506-C00166.png)
WO (1) WO2013105118A1 (US06559137-20030506-C00166.png)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2017173308A1 (en) 2016-03-31 2017-10-05 Goergetown University Radiation mitigator and method of use thereof
CN108486647A (zh) * 2018-05-24 2018-09-04 蔡凡 提拉法CeAlO3晶体生长装置及其控制方法
CN111233794A (zh) * 2020-03-27 2020-06-05 江巨东 一种安普那韦的精制方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8927913D0 (en) 1989-12-11 1990-02-14 Hoffmann La Roche Amino acid derivatives
US6436989B1 (en) 1997-12-24 2002-08-20 Vertex Pharmaceuticals, Incorporated Prodrugs of aspartyl protease inhibitors
ATE500823T1 (de) 1998-06-23 2011-03-15 Us Of America Represented By The Secretary Dept Of Health And Human Services Arzneimittel zur behandlung von hiv-infizierten säugetieren
WO1999067254A2 (en) 1998-06-23 1999-12-29 The United States Of America Represented By The Secretary, Department Of Health And Human Services Multi-drug resistant retroviral protease inhibitors and use thereof
GB9815567D0 (en) 1998-07-18 1998-09-16 Glaxo Group Ltd Antiviral compound
WO2000018384A2 (en) 1998-09-28 2000-04-06 Glaxo Group Limited Antiviral combinations comprising (s)-2-ethyl-7-fluoro-3-oxo-3,4-dihydro-2h-quinoxaline-1-carboxylic acid isopropyl ester and amprenavir

Also Published As

Publication number Publication date
WO2013105118A1 (en) 2013-07-18
US9233943B2 (en) 2016-01-12
US20150011782A1 (en) 2015-01-08
WO2013105118A8 (en) 2013-10-10

Similar Documents

Publication Publication Date Title
MX2017014351A (es) Un proceso para la preparacion de epoxido de terpinoleno.
BR112012028395A2 (pt) processo para preparar ditiina-tetracarboxi-diimidas
IN2014CN02584A (US06559137-20030506-C00166.png)
WO2013121436A3 (en) A process for preparation of rivaroxaban and intermediates thereof
PH12015500040B1 (en) Supercritical hydrolysis of biomass
MX2015006915A (es) Preparacion de una bebida estable.
GB201103836D0 (en) Conjugation process
IN2015KN00323A (US06559137-20030506-C00166.png)
IN2012MU03723A (US06559137-20030506-C00166.png)
IN2012DE00849A (US06559137-20030506-C00166.png)
MX2013007567A (es) Procedimiento para preparar poliestereteroles.
AU2010280497A8 (en) Anhydrate of tiotropium bromide
WO2014086732A8 (en) Reassortant influenza a viren
IN2012DE00082A (US06559137-20030506-C00166.png)
BR112012026157A2 (pt) processo para preparar ditiina-tetracarboximidas.
WO2014174483A3 (fr) Nouvelle algue radioresistante du genre coccomyxa
MX2015003034A (es) Jeringa que contiene una composicion, en particular farmaceutica, que comprende inmunoglobulinas, su metodo de fabricacion y uso.
MX2013004872A (es) Procesos para preparar un fenilciclohexano.
MX2012010443A (es) Proceso para la preparacion de 1-alquiltetrazoles 5-sustituidos.
WO2014064712A3 (en) An improved process for the preparation of fulvestrant
IN2014DN09451A (US06559137-20030506-C00166.png)
WO2012035303A8 (en) A novel process for synthesis of ramelteon, and key intermediates for the synthesis of ramelteon
IN2015DN00725A (US06559137-20030506-C00166.png)
BR112014018492A8 (pt) Processo aperfeiçoado para a produção de etileno 1,1-disubstituído
WO2014030173A3 (en) Improved process for preparation of atazanavir bisulfate