IL68205A - 5-(2-pyridylethenyl)-1h,7h-pyrazolo(1,5-a)pyrimidin-7-ones,their preparation and pharmaceutical compositions containing them - Google Patents

5-(2-pyridylethenyl)-1h,7h-pyrazolo(1,5-a)pyrimidin-7-ones,their preparation and pharmaceutical compositions containing them

Info

Publication number
IL68205A
IL68205A IL68205A IL6820583A IL68205A IL 68205 A IL68205 A IL 68205A IL 68205 A IL68205 A IL 68205A IL 6820583 A IL6820583 A IL 6820583A IL 68205 A IL68205 A IL 68205A
Authority
IL
Israel
Prior art keywords
pyridylethenyl
pyrazolo
pyrimidin
ones
preparation
Prior art date
Application number
IL68205A
Other languages
English (en)
Other versions
IL68205A0 (en
Inventor
Doria Gianfenderico
Passarotti Carlo
Arcari Guiliana
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of IL68205A0 publication Critical patent/IL68205A0/xx
Publication of IL68205A publication Critical patent/IL68205A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IL68205A 1982-03-25 1983-03-23 5-(2-pyridylethenyl)-1h,7h-pyrazolo(1,5-a)pyrimidin-7-ones,their preparation and pharmaceutical compositions containing them IL68205A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB8208763 1982-03-25

Publications (2)

Publication Number Publication Date
IL68205A0 IL68205A0 (en) 1983-06-15
IL68205A true IL68205A (en) 1986-01-31

Family

ID=10529266

Family Applications (1)

Application Number Title Priority Date Filing Date
IL68205A IL68205A (en) 1982-03-25 1983-03-23 5-(2-pyridylethenyl)-1h,7h-pyrazolo(1,5-a)pyrimidin-7-ones,their preparation and pharmaceutical compositions containing them

Country Status (16)

Country Link
US (1) US4490376A (sv)
JP (1) JPS58172391A (sv)
AU (1) AU557360B2 (sv)
BE (1) BE896255A (sv)
CA (1) CA1192547A (sv)
CH (1) CH655115A5 (sv)
DE (1) DE3310796A1 (sv)
DK (1) DK133883A (sv)
FI (1) FI74470C (sv)
FR (1) FR2523972B1 (sv)
IL (1) IL68205A (sv)
IT (1) IT1164159B (sv)
NL (1) NL8300837A (sv)
SE (1) SE447478B (sv)
SU (1) SU1301315A3 (sv)
ZA (1) ZA831407B (sv)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK170219B1 (da) * 1993-06-25 1995-07-03 Sanovo Eng As Apparat til rensning af æg
EP1921079A1 (en) * 2006-11-08 2008-05-14 Ferrer Internacional, S.A. Amorphous form of N-{2-Fluoro-5-[3-(thiophene-2-carbonyl)-pyrazolo[1,5-a] pyrimidin-7-yl]-phenyl}-N-methyl-acetamide
DK2387557T3 (da) * 2009-01-13 2013-09-08 Interquim Sa Fremgangsmåde til fremstilling af n-[5-(3-dimethylamino-acryloyl)-2-fluorphenyl]-n-methyl-acetamid

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE786611A (fr) * 1971-08-16 1973-01-22 Int Chem & Nuclear Corp Nouveaux inhibiteurs de xanthine-oxydase et leur procede de preparatio
US3907799A (en) * 1971-08-16 1975-09-23 Icn Pharmaceuticals Xanthine oxidase inhibitors
BE792533A (fr) * 1971-12-09 1973-06-08 Int Chem & Nuclear Corp Nouvelles pyrazolo (1,5a) pyrimidines et leur procede de preparation
US3925385A (en) * 1972-04-20 1975-12-09 Icn Pharmaceuticals 6-Carbethoxy-3,7-disubstitutedpyrazolo{8 1,5a{9 pyrimidines
US4093617A (en) * 1974-11-12 1978-06-06 Icn Pharmaceuticals, Inc. 3,5,7-Trisubstituted pyrazolo[1,5-a]pyrimidines
US4048184A (en) * 1976-11-15 1977-09-13 E. R. Squibb & Sons, Inc. 6-Phenyl-2H-pyrazolo[3,4-b]pyridines
US4281000A (en) * 1979-07-09 1981-07-28 American Cyanamid Company Substituted pyrazolo (1,5-a)pyrimidines and their use as anxiolytic agents

Also Published As

Publication number Publication date
DK133883A (da) 1983-09-26
CH655115A5 (de) 1986-03-27
DE3310796A1 (de) 1983-09-29
DK133883D0 (da) 1983-03-24
SU1301315A3 (ru) 1987-03-30
ZA831407B (en) 1983-11-30
NL8300837A (nl) 1983-10-17
FR2523972B1 (fr) 1985-12-06
IT8320095A0 (it) 1983-03-16
CA1192547A (en) 1985-08-27
FI830949A0 (fi) 1983-03-22
FR2523972A1 (fr) 1983-09-30
JPS58172391A (ja) 1983-10-11
SE8301641L (sv) 1983-09-26
FI74470B (fi) 1987-10-30
SE8301641D0 (sv) 1983-03-24
FI830949L (fi) 1983-09-26
US4490376A (en) 1984-12-25
IT1164159B (it) 1987-04-08
FI74470C (sv) 1988-02-08
AU557360B2 (en) 1986-12-18
AU1201983A (en) 1983-09-29
BE896255A (fr) 1983-09-26
IL68205A0 (en) 1983-06-15
SE447478B (sv) 1986-11-17

Similar Documents

Publication Publication Date Title
IL69955A (en) 1-phenyl-2-piperidinoalkanol derivatives,their preparation and pharmaceutical compositions containing them
IL68913A (en) 3-aminoalkyl-1h-indole-5-alkan-sulphonamide derivatives,their preparation and pharmaceutical compositions containing them
IL69157A0 (en) Fluoromorphinan derivatives,their preparation and pharmaceutical compositions containing them
IL71126A0 (en) Azole compounds,their preparation and pharmaceutical compositions containing them
IL69111A0 (en) Imidazole derivatives,their preparation and pharmaceutical compositions containing them
IL67826A0 (en) Pyrazolooxazines,pyrazolothiazines and pyrazoloquinolines,their preparation and pharmaceutical compositions containing them
IL68133A (en) 1-substituted-7-oxo-1h,7h-pyrazolo(1,5-a)pyrimidine-6-carboxylic acid derivatives,their preparation and pharmaceutical compositions containing them
IL68360A (en) Imidazopyrazolopyrimidine derivatives,their preparation and pharmaceutical compositions containing them
IL68442A0 (en) Imidazo(1,2-a)pyridine derivatives,their preparation and pharmaceutical compositions containing them
IL68817A0 (en) Oxoazetidine derivatives,their preparation and pharmaceutical compositions containing them
IL63405A0 (en) Benzodiazepine derivatives,their preparation and pharmaceutical compositions containing them
IL68497A0 (en) Benzoazacycloalkyl-spiro-imidazolidines,their preparation and pharmaceutical compositions containing them
ZM9283A1 (en) Substituted phenylsulfonyloxybenzimidazolecarbamates,processes for their preparation and pharmaceutical compositions containing the same
IL63406A0 (en) Benzodiazepine derivatives,their preparation and pharmaceutical compositions containing them
IL68586A0 (en) 4-aryl-4-piperidinecarbinols,their preparation and pharmaceutical compositions containing them
IL70485A (en) Imidazo(1,5-a)pyridine derivatives,their preparation and pharmaceutical compositions containing them
IL68699A (en) 3-phenoxy-1-azetidine-carboxamides,their preparation and pharmaceutical compositions containing them
IL70034A0 (en) Heterocyclic amino compounds,their preparation and pharmaceutical compositions containing them
DE3173130D1 (en) Amino-1,2,4-triazole derivatives, processes for their preparation and pharmaceutical compositions containing them
IL62229A (en) 3-substituted-5-amino-1,2,4-triazole derivatives,their preparation and pharmaceutical compositions containing them
IL68496A (en) 8-heteroarylalkyl-ergoline derivatives,their preparation and pharmaceutical compositions containing them
IL66316A (en) Substituted thiazolo(3,2-a)-pyrimidin-5-ones,their preparation and pharmaceutical compositions containing them
IL64489A0 (en) Benzodiazepine compounds,their preparation and pharmaceutical compositions containing them
DE3380093D1 (en) 3-aminopropoxyphenyl derivatives, their preparation and pharmaceutical compositions containing them
IL69001A0 (en) Triazole derivatives,their preparation and pharmaceutical compositions containing them