IL63206A - 7beta-((2-lower alkoxy)imino)-2-((2-amino-4-thiazolyl)acet-amido-3-((2-sulfamino(lower alkyl))tetrazol-5-yl thiomethyl)-3-cephem-4-carboxylic acids,their preparation and pharmaceutical compositions comprising them - Google Patents

7beta-((2-lower alkoxy)imino)-2-((2-amino-4-thiazolyl)acet-amido-3-((2-sulfamino(lower alkyl))tetrazol-5-yl thiomethyl)-3-cephem-4-carboxylic acids,their preparation and pharmaceutical compositions comprising them

Info

Publication number
IL63206A
IL63206A IL63206A IL6320681A IL63206A IL 63206 A IL63206 A IL 63206A IL 63206 A IL63206 A IL 63206A IL 6320681 A IL6320681 A IL 6320681A IL 63206 A IL63206 A IL 63206A
Authority
IL
Israel
Prior art keywords
7beta
sulfamino
acet
cephem
thiomethyl
Prior art date
Application number
IL63206A
Other languages
English (en)
Other versions
IL63206A0 (en
Original Assignee
Smithkline Beckman Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beckman Corp filed Critical Smithkline Beckman Corp
Publication of IL63206A0 publication Critical patent/IL63206A0/xx
Publication of IL63206A publication Critical patent/IL63206A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/36—Methylene radicals, substituted by sulfur atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IL63206A 1980-07-03 1981-06-29 7beta-((2-lower alkoxy)imino)-2-((2-amino-4-thiazolyl)acet-amido-3-((2-sulfamino(lower alkyl))tetrazol-5-yl thiomethyl)-3-cephem-4-carboxylic acids,their preparation and pharmaceutical compositions comprising them IL63206A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/165,822 US4308267A (en) 1980-07-03 1980-07-03 7-[2-Alkoxyimino-2-(amino-thiazole)acetamido]-3-[1-(sulfaminoalkly)tetrazolthiomethyl]cephalosporins

Publications (2)

Publication Number Publication Date
IL63206A0 IL63206A0 (en) 1981-09-13
IL63206A true IL63206A (en) 1986-09-30

Family

ID=22600626

Family Applications (1)

Application Number Title Priority Date Filing Date
IL63206A IL63206A (en) 1980-07-03 1981-06-29 7beta-((2-lower alkoxy)imino)-2-((2-amino-4-thiazolyl)acet-amido-3-((2-sulfamino(lower alkyl))tetrazol-5-yl thiomethyl)-3-cephem-4-carboxylic acids,their preparation and pharmaceutical compositions comprising them

Country Status (23)

Country Link
US (1) US4308267A (xx)
EP (1) EP0043713B1 (xx)
JP (1) JPS5745189A (xx)
KR (1) KR840002046B1 (xx)
AR (1) AR228606A1 (xx)
AT (1) ATE9585T1 (xx)
AU (1) AU547942B2 (xx)
CA (1) CA1151150A (xx)
DE (1) DE3166321D1 (xx)
DK (1) DK286981A (xx)
ES (1) ES8203908A1 (xx)
FI (1) FI66876C (xx)
GR (1) GR74363B (xx)
HU (1) HU185934B (xx)
IE (1) IE51365B1 (xx)
IL (1) IL63206A (xx)
NO (1) NO812268L (xx)
NZ (1) NZ197573A (xx)
PH (1) PH17670A (xx)
PT (1) PT73292B (xx)
YU (1) YU162481A (xx)
ZA (1) ZA814484B (xx)
ZW (1) ZW15181A1 (xx)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4526977A (en) * 1981-10-07 1985-07-02 American Home Products Corporation 2-(3-Amino-5-isoxazolyl)-2-oxyimino-acetic acids

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4171362A (en) * 1975-10-30 1979-10-16 Smithkline Corporation 7-Acylamino-3-(sulfaminoalkyl substituted tetrazolylthiomethyl)cephalosporins antibacterial compositions containing them and methods of treating bacterial infections with them
DE2760123C2 (de) * 1976-01-23 1986-04-30 Roussel-Uclaf, Paris 7-Aminothiazolyl-syn-oxyiminoacetamidocephalosporansäuren, ihre Herstellung und sie enthaltende pharmazeutische Zusammensetzungen
JPS52125188A (en) 1976-04-14 1977-10-20 Takeda Chem Ind Ltd Cephalosporin derivatives and their preparation
US4066762A (en) * 1976-07-12 1978-01-03 Smithkline Corporation Derivatives of 7-(2-substituted-2-hydroxyiminoacetamido)-3-(1-substituted tetrazol-5-ylthiomethyl-3-cephem-4-carboxylic acid
DE2714880A1 (de) 1977-04-02 1978-10-26 Hoechst Ag Cephemderivate und verfahren zu ihrer herstellung
MC1259A1 (fr) 1978-05-30 1980-01-14 Hoffmann La Roche Derives acyles
US4220761A (en) * 1978-09-12 1980-09-02 Fujisawa Pharmaceutical Co., Ltd. 7-[Substituted oximinoacetamido]-3-[hydroxy alkyltetrazolo]cephalosporin derivatives

Also Published As

Publication number Publication date
AR228606A1 (es) 1983-03-30
EP0043713A1 (en) 1982-01-13
FI66876C (fi) 1984-12-10
GR74363B (xx) 1984-06-28
HU185934B (en) 1985-04-28
ZA814484B (en) 1982-07-28
YU162481A (en) 1983-06-30
AU547942B2 (en) 1985-11-14
EP0043713B1 (en) 1984-09-26
KR830006310A (ko) 1983-09-20
ATE9585T1 (de) 1984-10-15
AU7234381A (en) 1982-01-07
ES503622A0 (es) 1982-04-01
DE3166321D1 (en) 1984-10-31
ZW15181A1 (en) 1981-09-29
IE811481L (en) 1982-01-03
CA1151150A (en) 1983-08-02
JPS5745189A (en) 1982-03-13
PT73292B (en) 1982-07-22
PT73292A (en) 1981-07-01
US4308267A (en) 1981-12-29
IE51365B1 (en) 1986-12-10
DK286981A (da) 1982-01-04
ES8203908A1 (es) 1982-04-01
KR840002046B1 (ko) 1984-11-06
FI66876B (fi) 1984-08-31
IL63206A0 (en) 1981-09-13
FI812046L (fi) 1982-01-04
PH17670A (en) 1984-11-02
NO812268L (no) 1982-01-04
NZ197573A (en) 1984-09-28

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