IL62101A - 2-(3-(4-(3-chloro-4-fluorophenyl)-1-piperazinyl)propyl)-1,2,4-triazolo(4,3-a)pyridin-3(2h)-one,its salts,their preparation and pharmaceutical compositions containing them - Google Patents
2-(3-(4-(3-chloro-4-fluorophenyl)-1-piperazinyl)propyl)-1,2,4-triazolo(4,3-a)pyridin-3(2h)-one,its salts,their preparation and pharmaceutical compositions containing themInfo
- Publication number
- IL62101A IL62101A IL62101A IL6210181A IL62101A IL 62101 A IL62101 A IL 62101A IL 62101 A IL62101 A IL 62101A IL 6210181 A IL6210181 A IL 6210181A IL 62101 A IL62101 A IL 62101A
- Authority
- IL
- Israel
- Prior art keywords
- triazolo
- piperazinyl
- pyridin
- fluorophenyl
- chloro
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Biomedical Technology (AREA)
- Public Health (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT21246/80A IT1147349B (it) | 1980-04-09 | 1980-04-09 | 2-parentesi quadra aperta 3-parentesi quadra aperta 4-(3-cloro-4-fluorofenil)-1-piperfrazinil parentesi quadra propil parentesi quadra chiusa-1,2,4-triazolo parentesi quadra aperta 4,3 parentesi quadra chiusa piridin-3(2h)-one |
Publications (2)
Publication Number | Publication Date |
---|---|
IL62101A0 IL62101A0 (en) | 1981-03-31 |
IL62101A true IL62101A (en) | 1984-01-31 |
Family
ID=11178966
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL62101A IL62101A (en) | 1980-04-09 | 1981-02-10 | 2-(3-(4-(3-chloro-4-fluorophenyl)-1-piperazinyl)propyl)-1,2,4-triazolo(4,3-a)pyridin-3(2h)-one,its salts,their preparation and pharmaceutical compositions containing them |
Country Status (21)
Country | Link |
---|---|
US (1) | US4402956A (el) |
JP (1) | JPS56158784A (el) |
KR (1) | KR840002292B1 (el) |
AR (1) | AR225076A1 (el) |
AT (1) | AT377262B (el) |
AU (1) | AU529605B2 (el) |
BE (1) | BE887547A (el) |
CA (1) | CA1176253A (el) |
CH (1) | CH652397A5 (el) |
DE (1) | DE3112984A1 (el) |
ES (1) | ES501188A0 (el) |
FI (1) | FI69306C (el) |
FR (1) | FR2480285A1 (el) |
GB (1) | GB2073747B (el) |
GR (1) | GR73620B (el) |
IL (1) | IL62101A (el) |
IT (1) | IT1147349B (el) |
NL (1) | NL8100998A (el) |
PT (1) | PT72813B (el) |
SE (1) | SE442201B (el) |
YU (1) | YU83181A (el) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2001504121A (ja) * | 1996-11-12 | 2001-03-27 | セプラコール,インク. | 2r,4s,r,s―および2s,4r,r,s―ヒドロキシイトラコナゾール―およびヒドロキシサパーコナゾール誘導体 |
JP2001504465A (ja) | 1996-11-12 | 2001-04-03 | セプラコール,インク. | 2r,4s,s,s―および2s,4r,s,s―ヒドロキシイトラコナゾール |
US6147077A (en) * | 1999-04-29 | 2000-11-14 | Sepracor Inc. | 2R,4S-hydroxyitraconazole isomers |
US8686158B2 (en) * | 2008-06-05 | 2014-04-01 | President And Fellows Of Harvard College | High-valent palladium fluoride complexes and uses thereof |
WO2010059943A2 (en) | 2008-11-20 | 2010-05-27 | President And Fellows Of Harvard College | Fluorination of organic compounds |
JP2012514655A (ja) * | 2009-01-09 | 2012-06-28 | プレジデント アンド フェローズ オブ ハーバード カレッジ | フッ素含有化合物およびその使用法 |
CN103596931B (zh) | 2011-04-12 | 2016-10-12 | 哈佛大学校长及研究员协会 | 有机化合物的氟化 |
WO2014052622A1 (en) | 2012-09-26 | 2014-04-03 | President And Fellows Of Harvard College | Nickel fluorinating complexes and uses thereof |
US10759764B2 (en) | 2013-10-18 | 2020-09-01 | President And Fellows Of Harvard College | Fluorination of organic compounds |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IT1066857B (it) * | 1965-12-15 | 1985-03-12 | Acraf | Derivati della s ipiazolo 4.3 a piridina e processi per la loro preparazione |
FR8135M (el) * | 1968-12-31 | 1970-08-10 | ||
US4267179A (en) * | 1978-06-23 | 1981-05-12 | Janssen Pharmaceutica, N.V. | Heterocyclic derivatives of (4-phenylpiperazin-1-yl-aryloxymethyl-1,3-dioxolan-2-yl)methyl-1H-imidazoles and 1H-1,2,4-triazoles |
UST100505I4 (en) | 1980-03-17 | 1981-04-07 | Triazolo[4,3-a]pyridin-3(2H)-ones |
-
1980
- 1980-04-09 IT IT21246/80A patent/IT1147349B/it active
-
1981
- 1981-02-10 IL IL62101A patent/IL62101A/xx unknown
- 1981-02-12 US US06/234,065 patent/US4402956A/en not_active Expired - Fee Related
- 1981-02-17 BE BE0/203815A patent/BE887547A/fr not_active IP Right Cessation
- 1981-02-25 CH CH1240/81A patent/CH652397A5/it not_active IP Right Cessation
- 1981-03-02 NL NL8100998A patent/NL8100998A/nl not_active Application Discontinuation
- 1981-03-16 GB GB8108158A patent/GB2073747B/en not_active Expired
- 1981-03-30 YU YU00831/81A patent/YU83181A/xx unknown
- 1981-03-30 CA CA000374133A patent/CA1176253A/en not_active Expired
- 1981-04-01 FI FI811000A patent/FI69306C/fi not_active IP Right Cessation
- 1981-04-01 DE DE19813112984 patent/DE3112984A1/de not_active Withdrawn
- 1981-04-01 SE SE8102093A patent/SE442201B/sv not_active IP Right Cessation
- 1981-04-02 AU AU69043/81A patent/AU529605B2/en not_active Ceased
- 1981-04-07 PT PT72813A patent/PT72813B/pt unknown
- 1981-04-07 AR AR284885A patent/AR225076A1/es active
- 1981-04-07 FR FR8106952A patent/FR2480285A1/fr active Granted
- 1981-04-07 KR KR1019810001166A patent/KR840002292B1/ko active IP Right Grant
- 1981-04-07 GR GR64614A patent/GR73620B/el unknown
- 1981-04-08 ES ES501188A patent/ES501188A0/es active Granted
- 1981-04-09 JP JP5420581A patent/JPS56158784A/ja active Pending
- 1981-04-09 AT AT0165081A patent/AT377262B/de not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
US4402956A (en) | 1983-09-06 |
GB2073747A (en) | 1981-10-21 |
AU6904381A (en) | 1981-10-15 |
CA1176253A (en) | 1984-10-16 |
IT1147349B (it) | 1986-11-19 |
SE442201B (sv) | 1985-12-09 |
KR830005218A (ko) | 1983-08-03 |
JPS56158784A (en) | 1981-12-07 |
FR2480285A1 (fr) | 1981-10-16 |
FI811000L (fi) | 1981-10-10 |
YU83181A (en) | 1983-12-31 |
DE3112984A1 (de) | 1981-12-24 |
GB2073747B (en) | 1983-09-07 |
CH652397A5 (it) | 1985-11-15 |
GR73620B (el) | 1984-03-26 |
BE887547A (fr) | 1981-06-15 |
NL8100998A (nl) | 1981-11-02 |
SE8102093L (sv) | 1981-10-10 |
AU529605B2 (en) | 1983-06-16 |
FI69306B (fi) | 1985-09-30 |
ES8202817A1 (es) | 1982-02-01 |
KR840002292B1 (ko) | 1984-12-15 |
IL62101A0 (en) | 1981-03-31 |
PT72813A (en) | 1981-05-01 |
FR2480285B1 (el) | 1984-02-24 |
ES501188A0 (es) | 1982-02-01 |
ATA165081A (de) | 1984-07-15 |
PT72813B (en) | 1982-04-02 |
IT8021246A0 (it) | 1980-04-09 |
AT377262B (de) | 1985-02-25 |
AR225076A1 (es) | 1982-02-15 |
FI69306C (fi) | 1986-01-10 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
IL62494A0 (en) | 3-(1-piperidinylalkyl)-4h-pyrido(1,2-a)pyrimidin-4-one derivatives,their preparation and pharmaceutical compositions containing them | |
IL70093A (en) | Leukotriene antagonist and antiinflammatory pharmaceutical compositions containing 4-acyl-3-hydroxy phenoxyalkane derivatives,some such new derivatives and their preparation | |
IL63784A0 (en) | Phenyl piperazine derivatives,their preparation and pharmaceutical compositions containing them | |
ZA815243B (en) | Piperidyl derivatives of triazine copolymers,processes for their preparation and stabilised composition containing these derivatives | |
IL62101A (en) | 2-(3-(4-(3-chloro-4-fluorophenyl)-1-piperazinyl)propyl)-1,2,4-triazolo(4,3-a)pyridin-3(2h)-one,its salts,their preparation and pharmaceutical compositions containing them | |
AU7452587A (en) | Sustained release formulations containing 4-(1-methyl-4- piperidylidene)-4H-benzo(4,5)-cyclohepta(1,2-b)thiophen- 10(9H)-one | |
IL72601A (en) | 1-h-imidazo(1',2':1,2)pyrrolo(3,4-b)pyridine-2,5-(3h,11bh)-dione derivatives,their preparation and herbicidal compositions containing them | |
IL58592A (en) | 9-(3-(3,5-cis-dimethylpiperazino)propyl)carbazole and salts thereof,their preparation and pharmaceutical composition containing them | |
IL62229A0 (en) | Heterocyclic derivatives,their preparation and pharmaceutical compositions containing them | |
PH15900A (en) | Derivatives of 5-(pyridyl-2'-oxy)-2-nitrobenzoic acid and herbicidal compositions containing them | |
DE2963350D1 (en) | Heterocyclic carboxamidine compounds, their preparation and pharmaceutical compositions containing them | |
IL60308A (en) | 4-(substituted)thio-1-beta-d-ribofuranosylpyrazolo-(3,4-d)pyrimidine derivatives,their preparation and pharmaceutical compositions containing them | |
IL60557A0 (en) | 1-benzoxepin-5(2h)-one derivatives,their preparation and phrmaceutical compositions containing them | |
IL65470A (en) | 2-(4-phenyl-polyhhydro-piperidinyl-or pyrrolidinyl alkyl)-1,2,4-triazolo(4,3-a)pyridin-3(2h)-ones,their preparation and pharmaceutical compositions containing them | |
NZ190698A (en) | 2-(1h-imidazol-l-yl) ethoxy derivatives of pyrazolo (3,4-b) pyridine-5-methanols | |
IL58229A (en) | Substituted benzylidene-benzofuran-3-(2h)-one compounds,their preparation and pharmaceutical compositions containing them | |
IL58155A0 (en) | 2h-(1)benzothiono(2,3-e)-1,2-thiazine-3-carbox-amide-1,1-dioxide derivatves their preparation and pharmaceutical compositions containing them | |
DE2860750D1 (en) | Antithrombotic 2-(gamma-(1-piperidinyl)propyl)1,2-benzisothiazol 3-one, its pharmaceutically acceptable acid addition salts, their preparation and their compositions | |
IL56558A (en) | 1alpha-alkyl-1-(3-(substituted amino)propyl)-1,2,3,4,6,7,12b beta-octahydro-indolo(2,3-a)quinolizines,their preparation and pharmaceutical compositions containing them | |
ZA803964B (en) | 2-(perhydro-1,4-diazine)-pyrimido(5,4-d)pyrimidines,and salts thereof,their preparation,pharmaceutical compositions,and use thereof | |
IL63783A0 (en) | Phenyl piperazine derivatives,their preparation and pharmaceutical compositions containing them | |
PT73123B (en) | 4-(1-piperazinyl)-furo<3,2-c>pyridine derivatives processes for their preparation and pharmaceutical compositions containing same | |
IL65555A (en) | 5-pyridyl-1h-pyrazolo(3,4-b)pyridin-3-amine derivatives,their preparation and pharmaceutical compositions containing them | |
IL64672A0 (en) | Substituted tetrahydro-1,2,4-oxadiazin-5-one derivatives,their preparation and pharmaceutical compositions containing them | |
IL64673A0 (en) | N4-substituted tetrahydro-1,2,4-oxadiazin-5-one derivatives,their preparation and pharmaceutical compositions containing them |