IL62101A - 2-(3-(4-(3-chloro-4-fluorophenyl)-1-piperazinyl)propyl)-1,2,4-triazolo(4,3-a)pyridin-3(2h)-one,its salts,their preparation and pharmaceutical compositions containing them - Google Patents

2-(3-(4-(3-chloro-4-fluorophenyl)-1-piperazinyl)propyl)-1,2,4-triazolo(4,3-a)pyridin-3(2h)-one,its salts,their preparation and pharmaceutical compositions containing them

Info

Publication number
IL62101A
IL62101A IL62101A IL6210181A IL62101A IL 62101 A IL62101 A IL 62101A IL 62101 A IL62101 A IL 62101A IL 6210181 A IL6210181 A IL 6210181A IL 62101 A IL62101 A IL 62101A
Authority
IL
Israel
Prior art keywords
triazolo
piperazinyl
pyridin
fluorophenyl
chloro
Prior art date
Application number
IL62101A
Other languages
English (en)
Other versions
IL62101A0 (en
Original Assignee
Acraf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Acraf filed Critical Acraf
Publication of IL62101A0 publication Critical patent/IL62101A0/xx
Publication of IL62101A publication Critical patent/IL62101A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IL62101A 1980-04-09 1981-02-10 2-(3-(4-(3-chloro-4-fluorophenyl)-1-piperazinyl)propyl)-1,2,4-triazolo(4,3-a)pyridin-3(2h)-one,its salts,their preparation and pharmaceutical compositions containing them IL62101A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT21246/80A IT1147349B (it) 1980-04-09 1980-04-09 2-parentesi quadra aperta 3-parentesi quadra aperta 4-(3-cloro-4-fluorofenil)-1-piperfrazinil parentesi quadra propil parentesi quadra chiusa-1,2,4-triazolo parentesi quadra aperta 4,3 parentesi quadra chiusa piridin-3(2h)-one

Publications (2)

Publication Number Publication Date
IL62101A0 IL62101A0 (en) 1981-03-31
IL62101A true IL62101A (en) 1984-01-31

Family

ID=11178966

Family Applications (1)

Application Number Title Priority Date Filing Date
IL62101A IL62101A (en) 1980-04-09 1981-02-10 2-(3-(4-(3-chloro-4-fluorophenyl)-1-piperazinyl)propyl)-1,2,4-triazolo(4,3-a)pyridin-3(2h)-one,its salts,their preparation and pharmaceutical compositions containing them

Country Status (21)

Country Link
US (1) US4402956A (OSRAM)
JP (1) JPS56158784A (OSRAM)
KR (1) KR840002292B1 (OSRAM)
AR (1) AR225076A1 (OSRAM)
AT (1) AT377262B (OSRAM)
AU (1) AU529605B2 (OSRAM)
BE (1) BE887547A (OSRAM)
CA (1) CA1176253A (OSRAM)
CH (1) CH652397A5 (OSRAM)
DE (1) DE3112984A1 (OSRAM)
ES (1) ES501188A0 (OSRAM)
FI (1) FI69306C (OSRAM)
FR (1) FR2480285A1 (OSRAM)
GB (1) GB2073747B (OSRAM)
GR (1) GR73620B (OSRAM)
IL (1) IL62101A (OSRAM)
IT (1) IT1147349B (OSRAM)
NL (1) NL8100998A (OSRAM)
PT (1) PT72813B (OSRAM)
SE (1) SE442201B (OSRAM)
YU (1) YU83181A (OSRAM)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2001504121A (ja) * 1996-11-12 2001-03-27 セプラコール，インク． ２ｒ，４ｓ，ｒ，ｓ―および２ｓ，４ｒ，ｒ，ｓ―ヒドロキシイトラコナゾール―およびヒドロキシサパーコナゾール誘導体
CA2269608A1 (en) 1996-11-12 1998-05-22 Sepracor Inc. 2r,4s,s,s- and 2s,4r,s,s-hydroxyitraconazole
US6147077A (en) * 1999-04-29 2000-11-14 Sepracor Inc. 2R,4S-hydroxyitraconazole isomers
US8686158B2 (en) * 2008-06-05 2014-04-01 President And Fellows Of Harvard College High-valent palladium fluoride complexes and uses thereof
JP2012509351A (ja) 2008-11-20 2012-04-19 プレジデント アンド フェローズ オブ ハーバード カレッジ 有機化合物のフッ素化
KR20110110297A (ko) * 2009-01-09 2011-10-06 프레지던트 앤드 펠로우즈 오브 하바드 칼리지 불소 함유 화합물 및 이의 사용방법
WO2012142162A2 (en) 2011-04-12 2012-10-18 President And Fellows Of Harvard College Fluorination of organic compounds
US9273083B2 (en) 2012-09-26 2016-03-01 President And Fellows Of Harvard College Nickel fluorinating complexes and uses thereof
WO2015058047A2 (en) 2013-10-18 2015-04-23 President And Fellows Of Harvard College Fluorination of organic compounds

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1066857B (it) * 1965-12-15 1985-03-12 Acraf Derivati della s ipiazolo 4.3 a piridina e processi per la loro preparazione
FR8135M (OSRAM) * 1968-12-31 1970-08-10
US4267179A (en) * 1978-06-23 1981-05-12 Janssen Pharmaceutica, N.V. Heterocyclic derivatives of (4-phenylpiperazin-1-yl-aryloxymethyl-1,3-dioxolan-2-yl)methyl-1H-imidazoles and 1H-1,2,4-triazoles
UST100505I4 (en) 1980-03-17 1981-04-07 Triazolo[4,3-a]pyridin-3(2H)-ones

Also Published As

Publication number Publication date
NL8100998A (nl) 1981-11-02
AT377262B (de) 1985-02-25
FR2480285B1 (OSRAM) 1984-02-24
ES8202817A1 (es) 1982-02-01
AU6904381A (en) 1981-10-15
BE887547A (fr) 1981-06-15
IL62101A0 (en) 1981-03-31
IT1147349B (it) 1986-11-19
IT8021246A0 (it) 1980-04-09
PT72813B (en) 1982-04-02
AU529605B2 (en) 1983-06-16
DE3112984A1 (de) 1981-12-24
FI69306B (fi) 1985-09-30
SE442201B (sv) 1985-12-09
PT72813A (en) 1981-05-01
GB2073747A (en) 1981-10-21
FI811000L (fi) 1981-10-10
KR830005218A (ko) 1983-08-03
US4402956A (en) 1983-09-06
FI69306C (fi) 1986-01-10
GR73620B (OSRAM) 1984-03-26
JPS56158784A (en) 1981-12-07
KR840002292B1 (ko) 1984-12-15
ATA165081A (de) 1984-07-15
CH652397A5 (it) 1985-11-15
YU83181A (en) 1983-12-31
FR2480285A1 (fr) 1981-10-16
SE8102093L (sv) 1981-10-10
AR225076A1 (es) 1982-02-15
CA1176253A (en) 1984-10-16
GB2073747B (en) 1983-09-07
ES501188A0 (es) 1982-02-01

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