IL59046A - Process for the preparation of 7-sulfonimidoyl xanthone-2-carboxylic acid derivatives - Google Patents

Process for the preparation of 7-sulfonimidoyl xanthone-2-carboxylic acid derivatives

Info

Publication number
IL59046A
IL59046A IL59046A IL5904679A IL59046A IL 59046 A IL59046 A IL 59046A IL 59046 A IL59046 A IL 59046A IL 5904679 A IL5904679 A IL 5904679A IL 59046 A IL59046 A IL 59046A
Authority
IL
Israel
Prior art keywords
preparation
sulfonimidoyl
xanthone
carboxylic acid
acid derivatives
Prior art date
Application number
IL59046A
Other versions
IL59046A0 (en
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of IL59046A0 publication Critical patent/IL59046A0/en
Publication of IL59046A publication Critical patent/IL59046A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/78—Ring systems having three or more relevant rings
    • C07D311/80—Dibenzopyrans; Hydrogenated dibenzopyrans
    • C07D311/82—Xanthenes
    • C07D311/84—Xanthenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 9
    • C07D311/86—Oxygen atoms, e.g. xanthones

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pyrane Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Diaphragms For Electromechanical Transducers (AREA)
  • Peptides Or Proteins (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

A process for the preparation of compounds of general formula I, <IMAGE> (wherein R represents a hydrogen atom or an alkyl radical containing from 1 to 9 carbon atoms and R1 represents an alkyl radical containing from 1 to 5 carbon atoms) which comprises cyclising a compound of formula II, <IMAGE> (wherein R and R1 are as defined above, Ar represents an aryl group and R2 and R3, which may be the same or different, each represents an esterifying group) followed if required, by hydrolysis to the free acid of formula I. The compounds of general formula I possess interesting anti-allergic activity.
IL59046A 1979-02-09 1979-12-27 Process for the preparation of 7-sulfonimidoyl xanthone-2-carboxylic acid derivatives IL59046A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB7904649 1979-02-09

Publications (2)

Publication Number Publication Date
IL59046A0 IL59046A0 (en) 1980-03-31
IL59046A true IL59046A (en) 1985-03-31

Family

ID=10503083

Family Applications (1)

Application Number Title Priority Date Filing Date
IL59046A IL59046A (en) 1979-02-09 1979-12-27 Process for the preparation of 7-sulfonimidoyl xanthone-2-carboxylic acid derivatives

Country Status (15)

Country Link
EP (1) EP0016665B1 (en)
JP (1) JPS55108867A (en)
AT (1) ATE967T1 (en)
AU (1) AU531013B2 (en)
CA (1) CA1146571A (en)
DE (1) DE3060348D1 (en)
DK (1) DK145948C (en)
ES (1) ES488385A0 (en)
FI (1) FI800392A (en)
GB (1) GB2042540B (en)
HU (1) HU180552B (en)
IE (1) IE49389B1 (en)
IL (1) IL59046A (en)
PT (1) PT70795B (en)
ZA (1) ZA80141B (en)

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL47519A (en) * 1974-07-09 1979-03-12 Roussel Uclaf 7-sulphinimidoyl(sulphimidoyl)-xanthone-2-carboxylic acid derivatives, their preparation and pharmaceutical compositions containing them
JPS5850225B2 (en) * 1976-01-01 1983-11-09 ルセル・ユクラフ Novel xanthones, their salts and esters, and pharmaceuticals comprising these compounds
SE445346B (en) * 1978-03-03 1986-06-16 Roussel Uclaf SET TO PREPARE 7-SULPHONIMIDOYL-XANTON-2-CARBOXYLIC ACID DERIVATIVE

Also Published As

Publication number Publication date
ES8102115A1 (en) 1980-12-16
JPS55108867A (en) 1980-08-21
GB2042540B (en) 1982-11-24
CA1146571A (en) 1983-05-17
HU180552B (en) 1983-03-28
JPH0144710B2 (en) 1989-09-29
IL59046A0 (en) 1980-03-31
GB2042540A (en) 1980-09-24
EP0016665A1 (en) 1980-10-01
PT70795A (en) 1980-03-01
ZA80141B (en) 1981-02-25
AU531013B2 (en) 1983-08-04
PT70795B (en) 1981-06-11
FI800392A (en) 1980-08-10
AU5535080A (en) 1980-08-14
IE49389B1 (en) 1985-10-02
DK54180A (en) 1980-08-10
ES488385A0 (en) 1980-12-16
IE800250L (en) 1980-08-09
EP0016665B1 (en) 1982-05-05
DE3060348D1 (en) 1982-06-24
DK145948C (en) 1983-09-26
ATE967T1 (en) 1982-05-15
DK145948B (en) 1983-04-25

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