IL308211A - Gastric residence systems comprising methadone - Google Patents
Gastric residence systems comprising methadoneInfo
- Publication number
- IL308211A IL308211A IL308211A IL30821123A IL308211A IL 308211 A IL308211 A IL 308211A IL 308211 A IL308211 A IL 308211A IL 30821123 A IL30821123 A IL 30821123A IL 308211 A IL308211 A IL 308211A
- Authority
- IL
- Israel
- Prior art keywords
- segment
- gastric residence
- drug
- residence system
- arms
- Prior art date
Links
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/12—Carboxylic acids; Salts or anhydrides thereof
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/32—Macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. carbomers, poly(meth)acrylates, or polyvinyl pyrrolidone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/34—Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
- A61K47/38—Cellulose; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/0065—Forms with gastric retention, e.g. floating on gastric juice, adhering to gastric mucosa, expanding to prevent passage through the pylorus
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Inorganic Chemistry (AREA)
- Nutrition Science (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Physiology (AREA)
- Emergency Medicine (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
- Medicines Containing Plant Substances (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202163184760P | 2021-05-05 | 2021-05-05 | |
| PCT/US2022/072115 WO2022236289A1 (en) | 2021-05-05 | 2022-05-04 | Gastric residence systems comprising methadone |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL308211A true IL308211A (en) | 2024-01-01 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL308211A IL308211A (en) | 2021-05-05 | 2022-05-04 | Gastric residence systems comprising methadone |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20240335400A1 (enExample) |
| EP (1) | EP4333824A4 (enExample) |
| JP (1) | JP2024517829A (enExample) |
| CN (1) | CN117615755A (enExample) |
| AU (1) | AU2022270208A1 (enExample) |
| CA (1) | CA3216743A1 (enExample) |
| IL (1) | IL308211A (enExample) |
| WO (1) | WO2022236289A1 (enExample) |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2020117855A1 (en) | 2018-12-03 | 2020-06-11 | Lyndra, Inc. | Stomach simulating device |
| BR112021018496A2 (pt) | 2019-03-20 | 2021-11-30 | Lyndra Therapeutics Inc | Cápsulas e revestimento de cápsula para formas de dosagem de residência gástrica |
| AU2020242062B2 (en) | 2019-03-20 | 2025-12-11 | Nortiva Bio, Inc. | Coatings for gastric residence dosage forms |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2011276170B2 (en) * | 2010-07-06 | 2016-03-10 | Grunenthal Gmbh | Novel gastro- retentive dosage forms comprising a GABA Analog and an opioid |
| AU2013369379B2 (en) * | 2012-12-27 | 2018-03-15 | Hennig Arzneimittel Gmbh & Co. Kg | Monolithic dosage form for the modified release of an active ingredient combination |
| US11576859B2 (en) * | 2015-10-23 | 2023-02-14 | Lyndra Therapeutics, Inc. | Gastric residence systems for sustained release of therapeutic agents and methods of use thereof |
| WO2017100367A1 (en) * | 2015-12-08 | 2017-06-15 | Lyndra, Inc. | Geometric configurations for gastric residence systems |
| SG11201901294QA (en) * | 2016-09-13 | 2019-03-28 | Alar Pharmaceuticals Inc | Sustained-release buprenorphine formulations background of invention |
| JP2019532947A (ja) * | 2016-09-30 | 2019-11-14 | リンドラ，インコーポレイティド | アダマンタン系薬物の持続的送達のための胃内滞留システム |
| CA3066658A1 (en) * | 2017-06-09 | 2018-12-13 | Lyndra, Inc. | Gastric residence systems with release rate-modulating films |
-
2022
- 2022-05-04 JP JP2023568006A patent/JP2024517829A/ja active Pending
- 2022-05-04 EP EP22799801.0A patent/EP4333824A4/en active Pending
- 2022-05-04 CN CN202280046388.1A patent/CN117615755A/zh active Pending
- 2022-05-04 CA CA3216743A patent/CA3216743A1/en active Pending
- 2022-05-04 AU AU2022270208A patent/AU2022270208A1/en not_active Abandoned
- 2022-05-04 IL IL308211A patent/IL308211A/en unknown
- 2022-05-04 WO PCT/US2022/072115 patent/WO2022236289A1/en not_active Ceased
- 2022-05-04 US US18/289,326 patent/US20240335400A1/en active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| AU2022270208A1 (en) | 2023-12-07 |
| EP4333824A1 (en) | 2024-03-13 |
| JP2024517829A (ja) | 2024-04-23 |
| CA3216743A1 (en) | 2022-11-10 |
| EP4333824A4 (en) | 2025-04-09 |
| WO2022236289A1 (en) | 2022-11-10 |
| CN117615755A (zh) | 2024-02-27 |
| US20240335400A1 (en) | 2024-10-10 |
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