IL188175A0 - 2-n-(5-[[4-(2-methyl-2-pyridinylamino)ethoxy] phenyl] methyl]-2,4-thiazolidinedione)butanedioic acid, methods of preparation and compositions with rosiglitazone maleate - Google Patents

2-n-(5-[[4-(2-methyl-2-pyridinylamino)ethoxy] phenyl] methyl]-2,4-thiazolidinedione)butanedioic acid, methods of preparation and compositions with rosiglitazone maleate

Info

Publication number
IL188175A0
IL188175A0 IL188175A IL18817507A IL188175A0 IL 188175 A0 IL188175 A0 IL 188175A0 IL 188175 A IL188175 A IL 188175A IL 18817507 A IL18817507 A IL 18817507A IL 188175 A0 IL188175 A0 IL 188175A0
Authority
IL
Israel
Prior art keywords
methyl
pyridinylamino
thiazolidinedione
ethoxy
phenyl
Prior art date
Application number
IL188175A
Other languages
English (en)
Original Assignee
Teva Pharma
Leibovici Minutza
Solomon Ben Sion
Avezov Yoseph
Dolitzky Yehudit
Spivak Dina
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Teva Pharma, Leibovici Minutza, Solomon Ben Sion, Avezov Yoseph, Dolitzky Yehudit, Spivak Dina filed Critical Teva Pharma
Publication of IL188175A0 publication Critical patent/IL188175A0/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IL188175A 2006-05-09 2007-12-17 2-n-(5-[[4-(2-methyl-2-pyridinylamino)ethoxy] phenyl] methyl]-2,4-thiazolidinedione)butanedioic acid, methods of preparation and compositions with rosiglitazone maleate IL188175A0 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/US2006/017994 WO2007130064A1 (fr) 2006-05-09 2006-05-09 Acide 2-n-(5-[[4-(2-methyl-2-pyridinylamino)ethoxy]phenyl]methyl]-2,4-thiazolidinedione)butanedioique, procedes de preparation et compositions a base de maleate de rosiglitazone

Publications (1)

Publication Number Publication Date
IL188175A0 true IL188175A0 (en) 2008-03-20

Family

ID=38668055

Family Applications (2)

Application Number Title Priority Date Filing Date
IL188175A IL188175A0 (en) 2006-05-09 2007-12-17 2-n-(5-[[4-(2-methyl-2-pyridinylamino)ethoxy] phenyl] methyl]-2,4-thiazolidinedione)butanedioic acid, methods of preparation and compositions with rosiglitazone maleate
IL199822A IL199822A0 (en) 2006-05-09 2009-07-13 Sealed package of pharmaceutical composition comprising 2-n-(5-[[4-(2-methyl-2-pyridinylamino)ethoxy] phenyl] methyl]-2,4-thiazolidinedione)butanedioic acid, methods of preparation and compositions with rosiglitazone maleate

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL199822A IL199822A0 (en) 2006-05-09 2009-07-13 Sealed package of pharmaceutical composition comprising 2-n-(5-[[4-(2-methyl-2-pyridinylamino)ethoxy] phenyl] methyl]-2,4-thiazolidinedione)butanedioic acid, methods of preparation and compositions with rosiglitazone maleate

Country Status (8)

Country Link
JP (1) JP2009536643A (fr)
CN (1) CN101426789A (fr)
BR (1) BRPI0621551A2 (fr)
CA (1) CA2647829A1 (fr)
IL (2) IL188175A0 (fr)
MX (1) MX2008014298A (fr)
NO (2) NO20085124L (fr)
WO (1) WO2007130064A1 (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2010013141A2 (fr) * 2008-08-01 2010-02-04 Actavis Group Ptc Ehf Hydrogénosulfate de rosiglitazone essentiellement pur
CN102863436B (zh) * 2012-06-19 2018-02-09 重庆医科大学 噻唑烷二酮类衍生物及其制备和用途

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5741803A (en) * 1992-09-05 1998-04-21 Smithkline Beecham Plc Substituted thiazolidinedionle derivatives

Also Published As

Publication number Publication date
NO20085124L (no) 2009-02-04
IL199822A0 (en) 2011-07-31
WO2007130064A1 (fr) 2007-11-15
NO20092362L (no) 2009-02-04
CA2647829A1 (fr) 2007-11-15
MX2008014298A (es) 2008-11-26
CN101426789A (zh) 2009-05-06
BRPI0621551A2 (pt) 2016-08-16
JP2009536643A (ja) 2009-10-15
WO2007130064A8 (fr) 2008-11-13

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