IL164044A0 - New crystalline forms of (2S)-N-5-Äamino(inino)methylÜ-2-thienylmethyl-1-(2R)-2-Ä(carboxsymethyl)aminoÜ-3,3-diphenylpropanoyl-2-pyrrolidinecarboxamide-nh2o - Google Patents
New crystalline forms of (2S)-N-5-Äamino(inino)methylÜ-2-thienylmethyl-1-(2R)-2-Ä(carboxsymethyl)aminoÜ-3,3-diphenylpropanoyl-2-pyrrolidinecarboxamide-nh2oInfo
- Publication number
- IL164044A0 IL164044A0 IL16404403A IL16404403A IL164044A0 IL 164044 A0 IL164044 A0 IL 164044A0 IL 16404403 A IL16404403 A IL 16404403A IL 16404403 A IL16404403 A IL 16404403A IL 164044 A0 IL164044 A0 IL 164044A0
- Authority
- IL
- Israel
- Prior art keywords
- äamino
- methylü
- carboxsymethyl
- aminoü
- diphenylpropanoyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06008—Dipeptides with the first amino acid being neutral
- C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K2299/00—Coordinates from 3D structures of peptides, e.g. proteins or enzymes
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| KR20020015627 | 2002-03-22 | ||
| PCT/KR2003/000558 WO2003080601A1 (fr) | 2002-03-22 | 2003-03-21 | Nouvelles formes cristallines de (2s)-n-5-[amino(imino)methyl]-2-thienylmethyl-1-(2r)-2-[(carboxymethyl)amino]-3,3-diphenylpropanoyl-2-pyrrolidinecarboxamide . nh2o |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL164044A0 true IL164044A0 (en) | 2005-12-18 |
Family
ID=36649957
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL16404403A IL164044A0 (en) | 2002-03-22 | 2003-03-21 | New crystalline forms of (2S)-N-5-Äamino(inino)methylÜ-2-thienylmethyl-1-(2R)-2-Ä(carboxsymethyl)aminoÜ-3,3-diphenylpropanoyl-2-pyrrolidinecarboxamide-nh2o |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US20050113309A1 (fr) |
| EP (1) | EP1487826A4 (fr) |
| JP (1) | JP2005526800A (fr) |
| KR (1) | KR20030076445A (fr) |
| CN (1) | CN1642947A (fr) |
| AU (1) | AU2003210055A1 (fr) |
| BR (1) | BR0308525A (fr) |
| CA (1) | CA2479888A1 (fr) |
| IL (1) | IL164044A0 (fr) |
| MX (1) | MXPA04009100A (fr) |
| PL (1) | PL372597A1 (fr) |
| RU (1) | RU2004131204A (fr) |
| WO (1) | WO2003080601A1 (fr) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PT2195293E (pt) | 2007-08-22 | 2014-01-21 | Astrazeneca Ab | Derivados da ciclopropilamida |
| TW201039825A (en) | 2009-02-20 | 2010-11-16 | Astrazeneca Ab | Cyclopropyl amide derivatives 983 |
| AU2011218490B9 (en) * | 2010-02-18 | 2014-12-18 | Astrazeneca Ab | Solid forms comprising a cyclopropyl amide derivative |
| RU2012136148A (ru) | 2010-02-18 | 2014-03-27 | Астразенека Аб | Новая кристаллическая форма производного циклопропилбензамида |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ZA951617B (en) * | 1994-03-04 | 1997-02-27 | Lilly Co Eli | Antithrombotic agents. |
| US5856480A (en) * | 1994-11-11 | 1999-01-05 | Nippon Soda Co., Ltd. | Optically active compound |
| WO1999037611A1 (fr) * | 1998-01-26 | 1999-07-29 | Basf Aktiengesellschaft | Amidines heterocycliques utilisees comme inhibiteurs de la kallicreine |
| KR20000047461A (ko) * | 1998-12-29 | 2000-07-25 | 성재갑 | 트롬빈 억제제 |
-
2003
- 2003-03-21 CN CNA038066947A patent/CN1642947A/zh active Pending
- 2003-03-21 MX MXPA04009100A patent/MXPA04009100A/es unknown
- 2003-03-21 BR BR0308525-2A patent/BR0308525A/pt not_active IP Right Cessation
- 2003-03-21 EP EP03744723A patent/EP1487826A4/fr not_active Withdrawn
- 2003-03-21 JP JP2003578355A patent/JP2005526800A/ja not_active Withdrawn
- 2003-03-21 CA CA002479888A patent/CA2479888A1/fr not_active Abandoned
- 2003-03-21 IL IL16404403A patent/IL164044A0/xx unknown
- 2003-03-21 AU AU2003210055A patent/AU2003210055A1/en not_active Abandoned
- 2003-03-21 PL PL03372597A patent/PL372597A1/xx unknown
- 2003-03-21 KR KR1020030017851A patent/KR20030076445A/ko not_active Application Discontinuation
- 2003-03-21 RU RU2004131204/04A patent/RU2004131204A/ru not_active Application Discontinuation
- 2003-03-21 WO PCT/KR2003/000558 patent/WO2003080601A1/fr not_active Application Discontinuation
- 2003-03-21 US US10/508,524 patent/US20050113309A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| CN1642947A (zh) | 2005-07-20 |
| WO2003080601A1 (fr) | 2003-10-02 |
| US20050113309A1 (en) | 2005-05-26 |
| EP1487826A1 (fr) | 2004-12-22 |
| PL372597A1 (en) | 2005-07-25 |
| AU2003210055A1 (en) | 2003-10-08 |
| MXPA04009100A (es) | 2004-12-06 |
| EP1487826A4 (fr) | 2005-06-29 |
| CA2479888A1 (fr) | 2003-10-02 |
| JP2005526800A (ja) | 2005-09-08 |
| KR20030076445A (ko) | 2003-09-26 |
| RU2004131204A (ru) | 2005-04-10 |
| BR0308525A (pt) | 2005-02-01 |
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