IL163683A0 - Substituted 3-phenyl-5-alkoxy-1,3,4,-oxadiazol-2-ones, their preparation and use in medicaments - Google Patents

Substituted 3-phenyl-5-alkoxy-1,3,4,-oxadiazol-2-ones, their preparation and use in medicaments

Info

Publication number
IL163683A0
IL163683A0 IL16368303A IL16368303A IL163683A0 IL 163683 A0 IL163683 A0 IL 163683A0 IL 16368303 A IL16368303 A IL 16368303A IL 16368303 A IL16368303 A IL 16368303A IL 163683 A0 IL163683 A0 IL 163683A0
Authority
IL
Israel
Prior art keywords
oxadiazol
medicaments
alkoxy
ones
phenyl
Prior art date
Application number
IL16368303A
Other languages
English (en)
Original Assignee
Aventis Pharma Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Gmbh filed Critical Aventis Pharma Gmbh
Publication of IL163683A0 publication Critical patent/IL163683A0/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D271/00Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/101,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles
    • C07D271/1131,3,4-Oxadiazoles; Hydrogenated 1,3,4-oxadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4245Oxadiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Steroid Compounds (AREA)
IL16368303A 2002-02-28 2003-02-14 Substituted 3-phenyl-5-alkoxy-1,3,4,-oxadiazol-2-ones, their preparation and use in medicaments IL163683A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10208987A DE10208987A1 (de) 2002-02-28 2002-02-28 Substituierte 3-Phenyl-5-alkoxi-1,3,4-oxidiazol-2-one, ihre Herstellung und Verwendung in Arzneistoffen
PCT/EP2003/001484 WO2003072555A1 (de) 2002-02-28 2003-02-14 Substituierte 3-phenyl-5-alkoxy-1,3,4-oxadiazol-2-one sowie ihre herstellung und verwendung in arzneistoffen

Publications (1)

Publication Number Publication Date
IL163683A0 true IL163683A0 (en) 2005-12-18

Family

ID=27740558

Family Applications (1)

Application Number Title Priority Date Filing Date
IL16368303A IL163683A0 (en) 2002-02-28 2003-02-14 Substituted 3-phenyl-5-alkoxy-1,3,4,-oxadiazol-2-ones, their preparation and use in medicaments

Country Status (22)

Country Link
EP (1) EP1480960B1 (xx)
JP (1) JP4486363B2 (xx)
KR (1) KR20040095240A (xx)
CN (1) CN1639137A (xx)
AR (1) AR038701A1 (xx)
AT (1) ATE557012T1 (xx)
AU (1) AU2003226977A1 (xx)
BR (1) BR0307921A (xx)
CA (1) CA2477031A1 (xx)
CO (1) CO5611146A2 (xx)
DE (1) DE10208987A1 (xx)
HR (1) HRP20040782A2 (xx)
HU (1) HUP0402671A3 (xx)
IL (1) IL163683A0 (xx)
MA (1) MA27172A1 (xx)
MX (1) MXPA04007960A (xx)
NO (1) NO20044090L (xx)
PE (1) PE20030928A1 (xx)
PL (1) PL370423A1 (xx)
RU (1) RU2004128933A (xx)
TW (1) TW200400951A (xx)
WO (1) WO2003072555A1 (xx)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7074822B2 (en) 2004-02-23 2006-07-11 Solvay Pharmaceuticals Gmbh Alkyl carbamate-substituted β-lactones, process for their preparation, and pharmaceutical compositions containing them
RU2007119315A (ru) 2004-10-25 2008-11-27 Зольвай Фармасьютиклз Гмбх (De) Фармацевтические композиции, содержащие антагонисты каннабиноидного рецептора св1 и открыватели калиевых каналов, предназначенные для лечения сахарного диабета типа i, ожирения и связанных с ними состояний
AU2008344032A1 (en) * 2007-12-27 2009-07-09 Bial-Portela & Ca., S.A. 5-O-substituted 3-N-phenyl-1,3,4-oxadiazolones for medical use
WO2010074587A2 (en) 2008-12-23 2010-07-01 Bial - Portela & Ca., S.A. 5-o-substituted 3-n-aryl-1,3,4-oxadiazolones for medical use

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19942354A1 (de) * 1999-09-04 2001-03-08 Aventis Pharma Gmbh Substituierte 3-Phenyl-5-alkoxi-1,3,4-oxdiazol-2-one, ihre Herstellung und Verwendung in Arzneimitteln
EE04877B1 (et) * 2000-03-07 2007-08-15 Aventis Pharma Deutschland Gmbh Asendatud 3-fenl-5-alkoks-1,3,4-oksadiasol-2-oon, selle valmistamine ja kasutamine hormoontundlikku lipaasi p„rssivas ravimis ning seda sisaldav suhkurt?ve ravim

Also Published As

Publication number Publication date
RU2004128933A (ru) 2005-04-20
HRP20040782A2 (en) 2005-02-28
HUP0402671A3 (en) 2006-07-28
WO2003072555A1 (de) 2003-09-04
NO20044090L (no) 2004-11-04
CN1639137A (zh) 2005-07-13
KR20040095240A (ko) 2004-11-12
MA27172A1 (fr) 2005-01-03
AR038701A1 (es) 2005-01-26
AU2003226977A1 (en) 2003-09-09
HUP0402671A2 (hu) 2005-04-28
BR0307921A (pt) 2004-12-21
CO5611146A2 (es) 2006-02-28
PL370423A1 (en) 2005-05-30
MXPA04007960A (es) 2004-11-26
DE10208987A1 (de) 2003-09-11
JP4486363B2 (ja) 2010-06-23
ATE557012T1 (de) 2012-05-15
EP1480960A1 (de) 2004-12-01
CA2477031A1 (en) 2003-09-04
TW200400951A (en) 2004-01-16
PE20030928A1 (es) 2003-12-17
JP2005519085A (ja) 2005-06-30
EP1480960B1 (de) 2012-05-09

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