IL148084A0 - Substituted (aminoiminomethyl or aminomethyl) dihydrobenzofurans and benzopyrans - Google Patents
Substituted (aminoiminomethyl or aminomethyl) dihydrobenzofurans and benzopyransInfo
- Publication number
- IL148084A0 IL148084A0 IL14808400A IL14808400A IL148084A0 IL 148084 A0 IL148084 A0 IL 148084A0 IL 14808400 A IL14808400 A IL 14808400A IL 14808400 A IL14808400 A IL 14808400A IL 148084 A0 IL148084 A0 IL 148084A0
- Authority
- IL
- Israel
- Prior art keywords
- factor
- dihydrobenzofurans
- aminoiminomethyl
- benzopyrans
- aminomethyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
- C07D307/81—Radicals substituted by nitrogen atoms not forming part of a nitro radical
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
- C07D407/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
- C07D407/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Immunology (AREA)
- Rheumatology (AREA)
- Communicable Diseases (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Oncology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Virology (AREA)
- Physical Education & Sports Medicine (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pyrane Compounds (AREA)
- Saccharide Compounds (AREA)
- Fats And Perfumes (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US15076799P | 1999-08-26 | 1999-08-26 | |
GBGB9924155.6A GB9924155D0 (en) | 1999-10-12 | 1999-10-12 | Chemical compounds |
PCT/IB2000/001562 WO2001014358A2 (en) | 1999-08-26 | 2000-08-12 | Substituted (aminoiminomethyl or aminomethyl) dihydrobenzofurans and benozopyrans |
Publications (1)
Publication Number | Publication Date |
---|---|
IL148084A0 true IL148084A0 (en) | 2002-09-12 |
Family
ID=26316000
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL14808400A IL148084A0 (en) | 1999-08-26 | 2000-08-12 | Substituted (aminoiminomethyl or aminomethyl) dihydrobenzofurans and benzopyrans |
Country Status (10)
Country | Link |
---|---|
US (1) | US6599918B2 (es) |
EP (1) | EP1222182B1 (es) |
AT (1) | ATE309995T1 (es) |
AU (1) | AU7812900A (es) |
CA (1) | CA2383257C (es) |
DE (1) | DE60024120T2 (es) |
ES (1) | ES2250196T3 (es) |
IL (1) | IL148084A0 (es) |
MX (1) | MXPA02001735A (es) |
WO (1) | WO2001014358A2 (es) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR100957516B1 (ko) * | 2001-08-15 | 2010-05-14 | 이코스 코포레이션 | 2h-프탈라진-1-온 및 이것의 사용 방법 |
CA2461381A1 (en) * | 2001-10-04 | 2003-04-10 | Wyeth | Chroman derivatives as 5-hydroxytryptamine-6 ligands |
JP4561698B2 (ja) * | 2002-02-19 | 2010-10-13 | 小野薬品工業株式会社 | 縮合ピリダジン誘導体化合物およびその化合物を有効成分として含有する薬剤 |
DE60325956D1 (de) * | 2002-04-10 | 2009-03-12 | Dongbu Hitek Co Ltd | Benzopyranderivate, die mit sekundären aminen einschliesslich tetrazol substituiert sind, verfahren etzungen, die diese enthalten |
US7593482B2 (en) | 2004-09-30 | 2009-09-22 | St-Ericsson Sa | Wireless communication system with hardware-based frequency burst detection |
ES2402362T3 (es) * | 2004-09-30 | 2013-05-03 | Takeda Pharmaceutical Company Limited | Inhibidores de la bomba de protones |
CA2621182C (en) * | 2005-08-30 | 2014-03-18 | Takeda Pharmaceutical Company Limited | 1-heterocyclylsulfonyl, 2-aminomethyl, 5-(hetero-)aryl substituted 1-h-pyrrole derivatives as acid secretion inhibitors |
MY154798A (en) | 2006-06-27 | 2015-07-31 | Takeda Pharmaceutical | Fused cyclic compounds |
US8933105B2 (en) * | 2007-02-28 | 2015-01-13 | Takeda Pharmaceutical Company Limited | Pyrrole compounds |
NZ591793A (en) * | 2008-08-27 | 2012-11-30 | Takeda Pharmaceutical | Substituted 1-(4-fluoro-5-(2-fluoropyridin-3-yl)-1-((pyrindin-2-yl)sulfonyl)-1H-pyrrol-3-yl)-N-methylmethanamine compounds |
CN103626747B (zh) * | 2013-10-22 | 2015-04-08 | 湖南大学 | N-(2,3-二氢苯并呋喃-5-基)苯并吡喃-4-酰胺及其制备方法与应用 |
JPWO2016104630A1 (ja) * | 2014-12-26 | 2017-10-05 | 武田薬品工業株式会社 | 縮合複素環化合物 |
GB2542064B (en) * | 2015-01-20 | 2020-11-18 | Univ California | Unit aerosol doses for anticoagulation |
CN113214199B (zh) * | 2021-04-28 | 2023-03-10 | 江西师范大学 | 一种苯并呋喃-3-氧代羧酸酯类化合物的合成方法 |
CN114057720B (zh) * | 2021-12-13 | 2024-02-23 | 陶金辉 | 一种靶向p2x7r的小分子抑制剂及其在治疗结肠癌中的应用 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0350163A3 (en) * | 1988-06-09 | 1990-11-22 | Beecham Group Plc | Renin inhibitory peptides |
ZA928276B (en) * | 1991-10-31 | 1993-05-06 | Daiichi Seiyaku Co | Aromatic amidine derivates and salts thereof. |
WO1997045424A1 (en) * | 1996-05-31 | 1997-12-04 | C & C Research Laboratories | Aromatic amidine derivatives useful as selective thrombin inhibitors |
WO1998001428A1 (en) * | 1996-07-08 | 1998-01-15 | Du Pont Pharmaceuticals Company | AMIDINOINDOLES, AMIDINOAZOLES, AND ANALOGS THEREOF AS INHIBITORS OF FACTOR Xa AND OF THROMBIN |
US5886191A (en) * | 1997-08-18 | 1999-03-23 | Dupont Pharmaceuticals Company | Amidinoindoles, amidinoazoles, and analogs thereof |
-
2000
- 2000-08-12 CA CA2383257A patent/CA2383257C/en not_active Expired - Fee Related
- 2000-08-12 AT AT00968181T patent/ATE309995T1/de not_active IP Right Cessation
- 2000-08-12 DE DE60024120T patent/DE60024120T2/de not_active Expired - Lifetime
- 2000-08-12 ES ES00968181T patent/ES2250196T3/es not_active Expired - Lifetime
- 2000-08-12 IL IL14808400A patent/IL148084A0/xx unknown
- 2000-08-12 WO PCT/IB2000/001562 patent/WO2001014358A2/en active IP Right Grant
- 2000-08-12 EP EP00968181A patent/EP1222182B1/en not_active Expired - Lifetime
- 2000-08-12 MX MXPA02001735A patent/MXPA02001735A/es active IP Right Grant
- 2000-08-12 AU AU78129/00A patent/AU7812900A/en not_active Abandoned
-
2002
- 2002-02-22 US US10/081,113 patent/US6599918B2/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
EP1222182B1 (en) | 2005-11-16 |
WO2001014358A2 (en) | 2001-03-01 |
CA2383257C (en) | 2010-09-28 |
ATE309995T1 (de) | 2005-12-15 |
EP1222182A2 (en) | 2002-07-17 |
DE60024120D1 (de) | 2005-12-22 |
ES2250196T3 (es) | 2006-04-16 |
WO2001014358A3 (en) | 2001-05-17 |
AU7812900A (en) | 2001-03-19 |
MXPA02001735A (es) | 2002-08-06 |
US6599918B2 (en) | 2003-07-29 |
US20020193410A1 (en) | 2002-12-19 |
CA2383257A1 (en) | 2001-03-01 |
DE60024120T2 (de) | 2006-07-27 |
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