ID27035A - NEW SUBSTITUTED INDOLINONA, THEIR PRODUCTION AND USE AS A PHARMACY COMPOSITION - Google Patents
NEW SUBSTITUTED INDOLINONA, THEIR PRODUCTION AND USE AS A PHARMACY COMPOSITIONInfo
- Publication number
- ID27035A ID27035A IDW20002523A ID20002523A ID27035A ID 27035 A ID27035 A ID 27035A ID W20002523 A IDW20002523 A ID W20002523A ID 20002523 A ID20002523 A ID 20002523A ID 27035 A ID27035 A ID 27035A
- Authority
- ID
- Indonesia
- Prior art keywords
- indolinona
- production
- new substituted
- pharmacy composition
- pharmacy
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/32—Oxygen atoms
- C07D209/34—Oxygen atoms in position 2
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19824922A DE19824922A1 (en) | 1998-06-04 | 1998-06-04 | Novel substituted indolinones, their preparation and their use as pharmaceuticals |
Publications (1)
Publication Number | Publication Date |
---|---|
ID27035A true ID27035A (en) | 2001-02-22 |
Family
ID=7869856
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IDW20002523A ID27035A (en) | 1998-06-04 | 1999-05-28 | NEW SUBSTITUTED INDOLINONA, THEIR PRODUCTION AND USE AS A PHARMACY COMPOSITION |
Country Status (23)
Country | Link |
---|---|
EP (1) | EP1100779A1 (en) |
JP (1) | JP2002516906A (en) |
KR (1) | KR20010043973A (en) |
CN (1) | CN1303374A (en) |
AU (1) | AU764782B2 (en) |
BG (1) | BG104938A (en) |
BR (1) | BR9910898A (en) |
CA (1) | CA2328291A1 (en) |
CO (1) | CO5050294A1 (en) |
DE (1) | DE19824922A1 (en) |
EA (1) | EA003514B1 (en) |
EE (1) | EE200000723A (en) |
HR (1) | HRP20000831A2 (en) |
HU (1) | HUP0102210A3 (en) |
ID (1) | ID27035A (en) |
IL (1) | IL138702A0 (en) |
NO (1) | NO20006138L (en) |
PL (1) | PL344467A1 (en) |
SK (1) | SK18222000A3 (en) |
TR (1) | TR200003515T2 (en) |
WO (1) | WO1999062882A1 (en) |
YU (1) | YU73900A (en) |
ZA (1) | ZA200005435B (en) |
Families Citing this family (27)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE19816624A1 (en) * | 1998-04-15 | 1999-10-21 | Boehringer Ingelheim Pharma | Novel substituted indolinones, their preparation and their use as pharmaceuticals |
GB9904933D0 (en) * | 1999-03-04 | 1999-04-28 | Glaxo Group Ltd | Compounds |
US6624171B1 (en) | 1999-03-04 | 2003-09-23 | Smithkline Beecham Corporation | Substituted aza-oxindole derivatives |
US6762180B1 (en) | 1999-10-13 | 2004-07-13 | Boehringer Ingelheim Pharma Kg | Substituted indolines which inhibit receptor tyrosine kinases |
UA75054C2 (en) * | 1999-10-13 | 2006-03-15 | Бьорінгер Інгельхайм Фарма Гмбх & Ко. Кг | Substituted in position 6 indolinones, producing and use thereof as medicament |
EP1317446A1 (en) | 2000-09-01 | 2003-06-11 | Glaxo Group Limited | Oxindole derivatives |
JP2004517049A (en) | 2000-09-01 | 2004-06-10 | グラクソ グループ リミテッド | Substituted oxindole derivatives as tyrosine kinase inhibitors |
DE10117204A1 (en) * | 2001-04-06 | 2002-10-10 | Boehringer Ingelheim Pharma | Indolinones substituted in the 6-position, their preparation and their use as medicaments |
JP2004537542A (en) | 2001-06-29 | 2004-12-16 | アブ サイエンス | Use of a tyrosine kinase inhibitor for treating inflammatory bowel disease (IBD) |
ATE345839T1 (en) | 2001-06-29 | 2006-12-15 | Ab Science | THE USE OF TYROSINE KINASE INHIBITORS FOR THE TREATMENT OF ALLERGY DISEASES |
EP1434991B1 (en) | 2001-06-29 | 2007-10-17 | AB Science | New potent, selective and non toxic c-kit inhibitors |
EP1401415B1 (en) * | 2001-06-29 | 2006-06-21 | AB Science | Use of n-phenyl-2-pyrimidine-amine derivatives for treating inflammatory diseases |
EP1471907B1 (en) * | 2001-06-29 | 2008-07-16 | AB Science | Use of c-kit inhibitors for treating autoimmune diseases |
AU2002341881B2 (en) | 2001-09-27 | 2008-05-08 | Allergan, Inc. | 3-(arylamino)methylene-1, 3-dihydro-2h-indol-2-ones as kinase inhibitors |
US7169936B2 (en) | 2002-07-23 | 2007-01-30 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Indolinone derivatives substituted in the 6-position, their preparation and their use as medicaments |
JP4879492B2 (en) * | 2002-11-27 | 2012-02-22 | アラーガン、インコーポレイテッド | Kinase inhibitors for the treatment of diseases |
DE102004012070A1 (en) * | 2004-03-12 | 2005-09-29 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | New cycloalkyl-containing 5-acylindolinones, their preparation and their use as medicaments |
PE20060777A1 (en) * | 2004-12-24 | 2006-10-06 | Boehringer Ingelheim Int | INDOLINONE DERIVATIVES FOR THE TREATMENT OR PREVENTION OF FIBROTIC DISEASES |
EP2099743B1 (en) * | 2006-12-05 | 2014-08-27 | Arena Pharmaceuticals, Inc. | Processes for preparing (r)-8-chloro-1-methyl-2,3,4,5-tetrahydro-1h-3-benzazepine and intermediates thereof |
GB0706072D0 (en) * | 2007-03-28 | 2007-05-09 | Sterix Ltd | Compound |
US20170065529A1 (en) | 2015-09-09 | 2017-03-09 | Boehringer Ingelheim International Gmbh | Pharmaceutical dosage form for immediate release of an indolinone derivative |
CN101735071A (en) * | 2009-12-04 | 2010-06-16 | 大连凯飞精细化工有限公司 | Method for producing 4-N,N-dimethylamino methylaniline |
CN103102352B (en) * | 2011-11-15 | 2015-08-12 | 山东亨利医药科技有限责任公司 | Tyrosine kinase inhibitor indolinone derivative |
CN103130775B (en) * | 2011-11-22 | 2015-09-30 | 山东亨利医药科技有限责任公司 | As the dihydroindole ketone derivate of tyrosine kinase inhibitor |
GB201208775D0 (en) | 2012-05-18 | 2012-07-04 | Uni I Oslo | Chemical compounds |
CN103848814B (en) * | 2012-12-06 | 2016-08-17 | 山东亨利医药科技有限责任公司 | The full ketone derivatives of substituted indole as tyrosine kinase inhibitor |
WO2024050297A1 (en) * | 2022-09-02 | 2024-03-07 | Deciphera Pharmaceuticals, Llc | Ulk inhibitors and methods of use thereof |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BE838623A (en) * | 1976-02-16 | 1976-06-16 | 3-HYDROXYMETHYLENE-2-INDOLINONE DERIVATIVES AND PROCESS FOR THEIR PRODUCTION | |
US4145422A (en) * | 1977-09-06 | 1979-03-20 | Abbott Laboratories | Aminomethylene oxindoles |
US5880141A (en) * | 1995-06-07 | 1999-03-09 | Sugen, Inc. | Benzylidene-Z-indoline compounds for the treatment of disease |
AU4155697A (en) * | 1996-08-23 | 1998-03-06 | Sugen, Inc. | Indolinone combinatorial libraries and related products and methods for the treatment of disease |
GB9718913D0 (en) * | 1997-09-05 | 1997-11-12 | Glaxo Group Ltd | Substituted oxindole derivatives |
-
1998
- 1998-06-04 DE DE19824922A patent/DE19824922A1/en not_active Withdrawn
-
1999
- 1999-05-28 EP EP99926454A patent/EP1100779A1/en not_active Withdrawn
- 1999-05-28 KR KR1020007013597A patent/KR20010043973A/en not_active Application Discontinuation
- 1999-05-28 JP JP2000552094A patent/JP2002516906A/en active Pending
- 1999-05-28 HU HU0102210A patent/HUP0102210A3/en unknown
- 1999-05-28 EA EA200100001A patent/EA003514B1/en not_active IP Right Cessation
- 1999-05-28 WO PCT/EP1999/003692 patent/WO1999062882A1/en not_active Application Discontinuation
- 1999-05-28 IL IL13870299A patent/IL138702A0/en unknown
- 1999-05-28 PL PL99344467A patent/PL344467A1/en unknown
- 1999-05-28 TR TR2000/03515T patent/TR200003515T2/en unknown
- 1999-05-28 AU AU43707/99A patent/AU764782B2/en not_active Ceased
- 1999-05-28 CA CA002328291A patent/CA2328291A1/en not_active Abandoned
- 1999-05-28 ID IDW20002523A patent/ID27035A/en unknown
- 1999-05-28 BR BR9910898-4A patent/BR9910898A/en not_active IP Right Cessation
- 1999-05-28 EE EEP200000723A patent/EE200000723A/en unknown
- 1999-05-28 YU YU73900A patent/YU73900A/en unknown
- 1999-05-28 SK SK1822-2000A patent/SK18222000A3/en unknown
- 1999-05-28 CN CN99806884A patent/CN1303374A/en active Pending
- 1999-06-04 CO CO99035396A patent/CO5050294A1/en unknown
-
2000
- 2000-10-05 ZA ZA200005435A patent/ZA200005435B/en unknown
- 2000-11-13 BG BG104938A patent/BG104938A/en active Pending
- 2000-12-01 NO NO20006138A patent/NO20006138L/en not_active Application Discontinuation
- 2000-12-01 HR HR20000831A patent/HRP20000831A2/en not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
AU764782B2 (en) | 2003-08-28 |
SK18222000A3 (en) | 2001-08-06 |
YU73900A (en) | 2003-04-30 |
HUP0102210A2 (en) | 2001-11-28 |
BG104938A (en) | 2001-06-29 |
CO5050294A1 (en) | 2001-06-27 |
EE200000723A (en) | 2002-04-15 |
IL138702A0 (en) | 2001-10-31 |
EA003514B1 (en) | 2003-06-26 |
CN1303374A (en) | 2001-07-11 |
BR9910898A (en) | 2001-02-13 |
AU4370799A (en) | 1999-12-20 |
EA200100001A1 (en) | 2001-08-27 |
WO1999062882A1 (en) | 1999-12-09 |
NO20006138D0 (en) | 2000-12-01 |
KR20010043973A (en) | 2001-05-25 |
JP2002516906A (en) | 2002-06-11 |
NO20006138L (en) | 2001-02-01 |
ZA200005435B (en) | 2002-01-07 |
HUP0102210A3 (en) | 2002-12-28 |
CA2328291A1 (en) | 1999-12-09 |
TR200003515T2 (en) | 2001-06-21 |
DE19824922A1 (en) | 1999-12-09 |
EP1100779A1 (en) | 2001-05-23 |
HRP20000831A2 (en) | 2001-12-31 |
PL344467A1 (en) | 2001-11-05 |
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