HUP0104036A2 - Aril-piperidin-karbonil-származékok és közbenső termékeik, és eljárás előállításukra - Google Patents

Aril-piperidin-karbonil-származékok és közbenső termékeik, és eljárás előállításukra

Info

Publication number
HUP0104036A2
HUP0104036A2 HU0104036A HUP0104036A HUP0104036A2 HU P0104036 A2 HUP0104036 A2 HU P0104036A2 HU 0104036 A HU0104036 A HU 0104036A HU P0104036 A HUP0104036 A HU P0104036A HU P0104036 A2 HUP0104036 A2 HU P0104036A2
Authority
HU
Hungary
Prior art keywords
derivatives
preparing
arylpiperidine
intermediates
carbinol intermediates
Prior art date
Application number
HU0104036A
Other languages
English (en)
Inventor
Bruce Ronsen
Subhash P. Upadhyaya
Original Assignee
Pentech Pharmaceuticals, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pentech Pharmaceuticals, Inc. filed Critical Pentech Pharmaceuticals, Inc.
Publication of HUP0104036A2 publication Critical patent/HUP0104036A2/hu
Publication of HUP0104036A3 publication Critical patent/HUP0104036A3/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C07C255/01—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms
    • C07C255/32—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring
    • C07C255/41—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring the carbon skeleton being further substituted by carboxyl groups, other than cyano groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D211/72—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D211/78—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/07—Optical isomers

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Hydrogenated Pyridines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
HU0104036A 1998-12-22 1999-12-17 Process for preparing arylpiperidine carbinol intermediates and derivatives HUP0104036A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US21839398A 1998-12-22 1998-12-22
PCT/US1999/030365 WO2000037443A1 (en) 1998-12-22 1999-12-17 Process for preparing arylpiperidine carbinol intermediates and derivatives

Publications (2)

Publication Number Publication Date
HUP0104036A2 true HUP0104036A2 (hu) 2002-02-28
HUP0104036A3 HUP0104036A3 (en) 2003-04-28

Family

ID=22814930

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0104036A HUP0104036A3 (en) 1998-12-22 1999-12-17 Process for preparing arylpiperidine carbinol intermediates and derivatives

Country Status (5)

Country Link
EP (1) EP1140832A4 (hu)
JP (1) JP2002533325A (hu)
AU (1) AU2200400A (hu)
HU (1) HUP0104036A3 (hu)
WO (1) WO2000037443A1 (hu)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9930577D0 (en) * 1999-12-23 2000-02-16 Smithkline Beecham Plc Novel process
CN114437085B (zh) * 2020-11-03 2023-06-23 烟台弘邦医药科技有限公司 一种瑞卡帕布中间体的制备方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1422263A (en) * 1973-01-30 1976-01-21 Ferrosan As 4-phenyl-piperidine compounds
CH636858A5 (de) * 1977-01-17 1983-06-30 Ciba Geigy Ag Verfahren zur herstellung neuer phenylazacycloalkane.
EP0190496A3 (en) * 1984-12-13 1987-05-27 Beecham Group Plc Piperidine derivatives having a gastro-intestinal activity
JP3446468B2 (ja) * 1996-04-15 2003-09-16 旭硝子株式会社 ピペリジンカルビノール類の製造方法
JPH11240869A (ja) * 1997-12-22 1999-09-07 Sumika Fine Chemicals Co Ltd ラクタムカルボン酸誘導体およびその製法、ならびにそれを用いたピペリジン誘導体の製法
ES2137131B1 (es) * 1998-02-06 2000-09-16 Vita Invest Sa Derivado de piperidinona procedimiento de obtencion y procedimiento para su utilizacion.
WO2000026187A1 (en) * 1998-11-02 2000-05-11 Synthon B.V. Process for producing 4-arylpiperidine-3-carbinols and related compounds

Also Published As

Publication number Publication date
HUP0104036A3 (en) 2003-04-28
JP2002533325A (ja) 2002-10-08
WO2000037443A1 (en) 2000-06-29
EP1140832A1 (en) 2001-10-10
EP1140832A4 (en) 2004-11-03
AU2200400A (en) 2000-07-12

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