AU2200400A - Process for preparing arylpiperidine carbinol intermediates and derivatives - Google Patents

Process for preparing arylpiperidine carbinol intermediates and derivatives

Info

Publication number
AU2200400A
AU2200400A AU22004/00A AU2200400A AU2200400A AU 2200400 A AU2200400 A AU 2200400A AU 22004/00 A AU22004/00 A AU 22004/00A AU 2200400 A AU2200400 A AU 2200400A AU 2200400 A AU2200400 A AU 2200400A
Authority
AU
Australia
Prior art keywords
derivatives
preparing
arylpiperidine
intermediates
carbinol intermediates
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU22004/00A
Inventor
Bruce Ronsen
Subhash P. Upadhyaya
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pentech Pharmaceuticals Inc
Original Assignee
Pentech Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pentech Pharmaceuticals Inc filed Critical Pentech Pharmaceuticals Inc
Publication of AU2200400A publication Critical patent/AU2200400A/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C07C255/01—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms
    • C07C255/32—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring
    • C07C255/41—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring the carbon skeleton being further substituted by carboxyl groups, other than cyano groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D211/72—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D211/78—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/07—Optical isomers

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Hydrogenated Pyridines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
AU22004/00A 1998-12-22 1999-12-17 Process for preparing arylpiperidine carbinol intermediates and derivatives Abandoned AU2200400A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US21839398A 1998-12-22 1998-12-22
US09218393 1998-12-22
PCT/US1999/030365 WO2000037443A1 (en) 1998-12-22 1999-12-17 Process for preparing arylpiperidine carbinol intermediates and derivatives

Publications (1)

Publication Number Publication Date
AU2200400A true AU2200400A (en) 2000-07-12

Family

ID=22814930

Family Applications (1)

Application Number Title Priority Date Filing Date
AU22004/00A Abandoned AU2200400A (en) 1998-12-22 1999-12-17 Process for preparing arylpiperidine carbinol intermediates and derivatives

Country Status (5)

Country Link
EP (1) EP1140832A4 (en)
JP (1) JP2002533325A (en)
AU (1) AU2200400A (en)
HU (1) HUP0104036A3 (en)
WO (1) WO2000037443A1 (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9930577D0 (en) * 1999-12-23 2000-02-16 Smithkline Beecham Plc Novel process
CN114437085B (en) * 2020-11-03 2023-06-23 烟台弘邦医药科技有限公司 Preparation method of rebamipa intermediate

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1422263A (en) * 1973-01-30 1976-01-21 Ferrosan As 4-phenyl-piperidine compounds
CH636858A5 (en) * 1977-01-17 1983-06-30 Ciba Geigy Ag METHOD FOR PRODUCING NEW PHENYLAZACYCLOAL CHANES.
EP0190496A3 (en) * 1984-12-13 1987-05-27 Beecham Group Plc Piperidine derivatives having a gastro-intestinal activity
JP3446468B2 (en) * 1996-04-15 2003-09-16 旭硝子株式会社 Method for producing piperidine carbinols
JPH11240869A (en) * 1997-12-22 1999-09-07 Sumika Fine Chemicals Co Ltd Lactam carboxylic acid derivative, its production and production of piperidine derivative using the same
ES2137131B1 (en) * 1998-02-06 2000-09-16 Vita Invest Sa DERIVATIVE OF PIPERIDINONE PROCEDURE FOR OBTAINING AND PROCEDURE FOR ITS USE.
WO2000026187A1 (en) * 1998-11-02 2000-05-11 Synthon B.V. Process for producing 4-arylpiperidine-3-carbinols and related compounds

Also Published As

Publication number Publication date
WO2000037443A1 (en) 2000-06-29
EP1140832A1 (en) 2001-10-10
JP2002533325A (en) 2002-10-08
HUP0104036A3 (en) 2003-04-28
HUP0104036A2 (en) 2002-02-28
EP1140832A4 (en) 2004-11-03

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Legal Events

Date Code Title Description
MK6 Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase