HK1156032A1 - Quinuclidine carbonate derivatives and medicinal composition thereof - Google Patents

Quinuclidine carbonate derivatives and medicinal composition thereof

Info

Publication number
HK1156032A1
HK1156032A1 HK11110402.8A HK11110402A HK1156032A1 HK 1156032 A1 HK1156032 A1 HK 1156032A1 HK 11110402 A HK11110402 A HK 11110402A HK 1156032 A1 HK1156032 A1 HK 1156032A1
Authority
HK
Hong Kong
Prior art keywords
medicinal composition
carbonate derivatives
quinuclidine
quinuclidine carbonate
derivatives
Prior art date
Application number
HK11110402.8A
Other languages
English (en)
Inventor
Gabriele Amari
Maurizio Delcanale
Original Assignee
Chiesi Farma Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chiesi Farma Spa filed Critical Chiesi Farma Spa
Publication of HK1156032A1 publication Critical patent/HK1156032A1/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/04Drugs for disorders of the respiratory system for throat disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Pulmonology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)
HK11110402.8A 2008-08-08 2011-10-03 Quinuclidine carbonate derivatives and medicinal composition thereof HK1156032A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP08162066A EP2154136A1 (fr) 2008-08-08 2008-08-08 Dérivés de carbone de quinuclidine et ses compositions médicales
PCT/EP2009/005272 WO2010015324A1 (fr) 2008-08-08 2009-07-21 Dérivés de carbonate de quinuclidine et composition médicinale les comprenant

Publications (1)

Publication Number Publication Date
HK1156032A1 true HK1156032A1 (en) 2012-06-01

Family

ID=40228074

Family Applications (1)

Application Number Title Priority Date Filing Date
HK11110402.8A HK1156032A1 (en) 2008-08-08 2011-10-03 Quinuclidine carbonate derivatives and medicinal composition thereof

Country Status (32)

Country Link
US (3) US8039483B2 (fr)
EP (2) EP2154136A1 (fr)
JP (1) JP2011530489A (fr)
KR (1) KR20110044221A (fr)
CN (1) CN102112474B (fr)
AR (1) AR072994A1 (fr)
AT (1) ATE551341T1 (fr)
AU (1) AU2009278306B2 (fr)
CA (1) CA2733380A1 (fr)
CO (1) CO6351790A2 (fr)
CY (1) CY1112724T1 (fr)
DK (1) DK2313404T3 (fr)
EA (1) EA019166B1 (fr)
ES (1) ES2384914T3 (fr)
GE (1) GEP20135744B (fr)
HK (1) HK1156032A1 (fr)
HR (1) HRP20120394T1 (fr)
IL (1) IL211103A (fr)
JO (1) JO2831B1 (fr)
MA (1) MA32622B1 (fr)
ME (1) ME01283A (fr)
MX (1) MX2011001504A (fr)
MY (1) MY156332A (fr)
NZ (1) NZ590987A (fr)
PL (1) PL2313404T3 (fr)
PT (1) PT2313404E (fr)
RS (1) RS52370B (fr)
SI (1) SI2313404T1 (fr)
TW (1) TWI455938B (fr)
UA (1) UA102857C2 (fr)
WO (1) WO2010015324A1 (fr)
ZA (1) ZA201100963B (fr)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2009079078A1 (fr) 2007-12-14 2009-06-25 Labogroup S.A.S. Administration de produits alimentaires sous forme d'aérosols
EP2154136A1 (fr) 2008-08-08 2010-02-17 CHIESI FARMACEUTICI S.p.A. Dérivés de carbone de quinuclidine et ses compositions médicales
EP2206712A1 (fr) 2008-12-23 2010-07-14 CHIESI FARMACEUTICI S.p.A. Dérivés d'amino-ester d'alcaloïde et sa composition médicale
NO2560611T3 (fr) 2010-04-21 2018-06-02
CA2803433A1 (fr) 2010-06-22 2011-12-29 Chiesi Farmaceutici S.P.A. Derives aminoester d'alkaloides et composition medicinale les comprenant
WO2011161018A1 (fr) 2010-06-22 2011-12-29 Chiesi Farmaceutici S.P.A. Dérivés aminoester d'alcaloïdes et compositions médicinales les comprenant
KR20130111968A (ko) 2010-06-22 2013-10-11 키에시 파르마슈티시 엣스. 피. 에이. 알칼로이드 아미노에스테르 유도체 및 이의 의약 조성물
PL2621494T3 (pl) * 2010-09-30 2019-04-30 Chiesi Farm Spa Zastosowanie stearynianu magnezu w preparatach w postaci suchego proszku do inhalacji
RU2013118026A (ru) * 2010-10-20 2014-10-27 КЬЕЗИ ФАРМАЧЕУТИЧИ С.п.А. Карбонатные производные для лечения кашля
CA2820600A1 (fr) 2010-11-26 2012-05-31 Chiesi Farmaceutici S.P.A. Derives de glycine et leur utilisation en tant qu'antagonistes des recepteurs muscariniques
PT2685986T (pt) * 2011-03-18 2020-03-05 Genzyme Corp Inibidor de glicosilceramida-sintase
EP2702041A1 (fr) 2011-04-29 2014-03-05 Chiesi Farmaceutici S.p.A. Dérivés d'alcaloïde ester et carbamate, et compositions médicinales à base de ceux-ci
KR20140105746A (ko) 2011-12-30 2014-09-02 키에시 파르마슈티시 엣스. 피. 에이. 항무스카린제로서 1-아자헤테로시클릴아세트산의 퀴누클리딘 에스터, 이들의 제조 방법 및 이들의 의약 조성물
JOP20130273B1 (ar) 2012-09-11 2021-08-17 Genzyme Corp مثبطات انزيم (سينثاز) غلوكوسيل سيراميد
US9427376B2 (en) 2013-10-10 2016-08-30 Chiesi Farmaceutici S.P.A. Process for preparing pharmaceutical formulations for inhalation comprising a high-dosage strength active ingredient
EP4185267A1 (fr) 2020-07-24 2023-05-31 Genzyme Corporation Compositions pharmaceutiques comprenant du venglustat

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2165768B1 (es) * 1999-07-14 2003-04-01 Almirall Prodesfarma Sa Nuevos derivados de quinuclidina y composiciones farmaceuticas que los contienen.
SK8002003A3 (en) 2000-12-22 2004-05-04 Almirall Prodesfarma Ag Quinuclidine carbamate derivatives and their use as M3 antagonists
EP1383730A2 (fr) * 2001-04-03 2004-01-28 Aryx Therapeutics Composes anticholinergiques et procedes d'utilisation
MXPA04006206A (es) 2001-12-20 2004-12-06 S A L V A T Lab Sa Derivados de 1-alquil-azoniabiciclo(2.2.2(octano carbamato y su uso como antagonistas del receptor musrcarinico.
EP1882691A1 (fr) 2006-07-26 2008-01-30 CHIESI FARMACEUTICI S.p.A. Dérivés de quinuclidine comme antagonistes M3
EP2154136A1 (fr) 2008-08-08 2010-02-17 CHIESI FARMACEUTICI S.p.A. Dérivés de carbone de quinuclidine et ses compositions médicales
EP2206712A1 (fr) 2008-12-23 2010-07-14 CHIESI FARMACEUTICI S.p.A. Dérivés d'amino-ester d'alcaloïde et sa composition médicale
BR112012032330A2 (pt) 2010-06-22 2016-11-08 Chiesi Farma Spa formulação em pó seco inalável, uso de uma formulação em pó seco, inalador de pó seco e embalagem
RU2013118026A (ru) 2010-10-20 2014-10-27 КЬЕЗИ ФАРМАЧЕУТИЧИ С.п.А. Карбонатные производные для лечения кашля
US20120220557A1 (en) 2011-02-17 2012-08-30 Chiesi Farmaceutici S.P.A. Liquid propellant-free formulation comprising an antimuscarinic drug
EP2702041A1 (fr) 2011-04-29 2014-03-05 Chiesi Farmaceutici S.p.A. Dérivés d'alcaloïde ester et carbamate, et compositions médicinales à base de ceux-ci

Also Published As

Publication number Publication date
US8440690B2 (en) 2013-05-14
IL211103A0 (en) 2011-04-28
ZA201100963B (en) 2012-05-30
PT2313404E (pt) 2012-07-02
EP2313404B1 (fr) 2012-03-28
AU2009278306A1 (en) 2010-02-11
TWI455938B (zh) 2014-10-11
US8404712B2 (en) 2013-03-26
MA32622B1 (fr) 2011-09-01
SI2313404T1 (sl) 2012-07-31
EP2313404A1 (fr) 2011-04-27
AR072994A1 (es) 2010-10-06
AU2009278306B2 (en) 2014-06-26
CN102112474A (zh) 2011-06-29
US20120004258A1 (en) 2012-01-05
ME01283A (fr) 2013-06-20
EP2154136A1 (fr) 2010-02-17
RS52370B (en) 2012-12-31
CY1112724T1 (el) 2016-02-10
US20110319444A1 (en) 2011-12-29
KR20110044221A (ko) 2011-04-28
GEP20135744B (en) 2013-02-11
EA201100161A1 (ru) 2011-10-31
CA2733380A1 (fr) 2010-02-11
CO6351790A2 (es) 2011-12-20
HRP20120394T1 (hr) 2012-06-30
NZ590987A (en) 2012-11-30
EA019166B1 (ru) 2014-01-30
PL2313404T3 (pl) 2012-09-28
ES2384914T3 (es) 2012-07-13
DK2313404T3 (da) 2012-06-04
WO2010015324A1 (fr) 2010-02-11
MX2011001504A (es) 2011-03-29
JO2831B1 (en) 2014-09-15
ATE551341T1 (de) 2012-04-15
US8039483B2 (en) 2011-10-18
JP2011530489A (ja) 2011-12-22
US20100035922A1 (en) 2010-02-11
IL211103A (en) 2014-04-30
MY156332A (en) 2016-02-15
TW201011022A (en) 2010-03-16
UA102857C2 (en) 2013-08-27
CN102112474B (zh) 2014-01-29

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