HK1073243A1 - Use of N-(indolecarbonyl-) piperazine derivatives - Google Patents

Use of N-(indolecarbonyl-) piperazine derivatives

Info

Publication number
HK1073243A1
HK1073243A1 HK05105839A HK05105839A HK1073243A1 HK 1073243 A1 HK1073243 A1 HK 1073243A1 HK 05105839 A HK05105839 A HK 05105839A HK 05105839 A HK05105839 A HK 05105839A HK 1073243 A1 HK1073243 A1 HK 1073243A1
Authority
HK
Hong Kong
Prior art keywords
indolecarbonyl
piperazine derivatives
piperazine
derivatives
Prior art date
Application number
HK05105839A
Other languages
English (en)
Inventor
Christoph Van Amsterdam
Ewen Sedman
Gard Bartoszyk
Jurgen Hellmann
Van F Landengerb
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of HK1073243A1 publication Critical patent/HK1073243A1/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Child & Adolescent Psychology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
HK05105839A 2001-11-24 2005-07-11 Use of N-(indolecarbonyl-) piperazine derivatives HK1073243A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10157673A DE10157673A1 (de) 2001-11-24 2001-11-24 Verwendung von N-(Indolcarbonyl-)piperazinderivaten
PCT/EP2002/012009 WO2003045392A2 (de) 2001-11-24 2002-10-28 Verwendung von n-(indolcarbonyl-)piperazinderivaten

Publications (1)

Publication Number Publication Date
HK1073243A1 true HK1073243A1 (en) 2005-09-30

Family

ID=7706831

Family Applications (1)

Application Number Title Priority Date Filing Date
HK05105839A HK1073243A1 (en) 2001-11-24 2005-07-11 Use of N-(indolecarbonyl-) piperazine derivatives

Country Status (23)

Country Link
US (1) US20050014766A1 (zh)
EP (1) EP1448201B1 (zh)
JP (1) JP2005511640A (zh)
KR (1) KR100953172B1 (zh)
CN (1) CN1319532C (zh)
AR (1) AR037404A1 (zh)
AU (1) AU2002349012B2 (zh)
BR (1) BR0214347A (zh)
CA (1) CA2468380A1 (zh)
DE (2) DE10157673A1 (zh)
ES (1) ES2297018T3 (zh)
HK (1) HK1073243A1 (zh)
HU (1) HUP0402388A3 (zh)
IL (2) IL162125A0 (zh)
MX (1) MXPA04004766A (zh)
MY (1) MY141210A (zh)
NZ (1) NZ533667A (zh)
PE (1) PE20030710A1 (zh)
PL (1) PL207565B1 (zh)
RU (1) RU2317083C2 (zh)
UA (1) UA77468C2 (zh)
WO (1) WO2003045392A2 (zh)
ZA (1) ZA200404967B (zh)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10246357A1 (de) * 2002-10-04 2004-04-15 Merck Patent Gmbh Verwendung von 5-HT2Rezeptorantagonisten
DE102004047517A1 (de) * 2004-09-28 2006-03-30 Merck Patent Gmbh Neuartige Kristallform von (3-Cyan-1H-indol-7-yl)-[4-(4-fluorphenethyl)-piperazin-1-yl]-methanon, Hydrochlorid

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3582371D1 (de) * 1984-07-06 1991-05-08 Otsuka Pharma Co Ltd Oxindolverbindungen, diese enthaltende zusammensetzungen sowie verfahren zur herstellung derselben.
GB9718712D0 (en) * 1997-09-03 1997-11-12 Merck Sharp & Dohme Theraputic Agents
EP1076644B1 (en) * 1998-04-29 2004-06-23 Ortho-McNeil Pharmaceutical, Inc. N-substituted aminotetralins as ligands for the neuropeptide y y5 receptor useful in the treatment of obesity and other disorders
GB9825413D0 (en) * 1998-11-19 1999-01-13 Lilly Co Eli Pharmaceutical compounds
DE19934433A1 (de) * 1999-07-22 2001-01-25 Merck Patent Gmbh N-(Indolcarbonyl-)piperazinderivate
DE19934432A1 (de) * 1999-07-22 2001-02-01 Merck Patent Gmbh Indolderivate
US6372743B1 (en) * 1999-09-30 2002-04-16 Neurogen Corporation Certain alkylene diamine-substituted pyrazlo (1,5-a)-1,5-pyrimidines and pyrazolo (1,5-a) 1,3,5-triazines

Also Published As

Publication number Publication date
MXPA04004766A (es) 2004-07-30
AU2002349012A1 (en) 2003-06-10
KR100953172B1 (ko) 2010-04-20
BR0214347A (pt) 2004-10-26
IL162125A (en) 2010-12-30
WO2003045392A8 (de) 2004-12-29
AU2002349012B2 (en) 2008-01-24
MY141210A (en) 2010-03-31
DE50211298D1 (de) 2008-01-10
RU2004119303A (ru) 2005-04-20
CA2468380A1 (en) 2003-06-05
US20050014766A1 (en) 2005-01-20
AR037404A1 (es) 2004-11-10
EP1448201A2 (de) 2004-08-25
HUP0402388A2 (hu) 2005-03-29
CN1589147A (zh) 2005-03-02
PE20030710A1 (es) 2003-08-21
KR20040072624A (ko) 2004-08-18
JP2005511640A (ja) 2005-04-28
IL162125A0 (en) 2005-11-20
ES2297018T3 (es) 2008-05-01
HUP0402388A3 (en) 2009-08-28
CN1319532C (zh) 2007-06-06
DE10157673A1 (de) 2003-06-05
EP1448201B1 (de) 2007-11-28
WO2003045392A3 (de) 2003-09-18
NZ533667A (en) 2006-11-30
WO2003045392A2 (de) 2003-06-05
RU2317083C2 (ru) 2008-02-20
PL207565B1 (pl) 2011-01-31
ZA200404967B (en) 2005-08-05
PL369675A1 (en) 2005-05-02
UA77468C2 (en) 2006-12-15

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Legal Events

Date Code Title Description
PC Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)

Effective date: 20111028