HK1061973B - 内醯胺类-含其化合物及衍生物并作为因子xa的抑制剂 - Google Patents
内醯胺类-含其化合物及衍生物并作为因子xa的抑制剂 Download PDFInfo
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- HK1061973B HK1061973B HK04105041.4A HK04105041A HK1061973B HK 1061973 B HK1061973 B HK 1061973B HK 04105041 A HK04105041 A HK 04105041A HK 1061973 B HK1061973 B HK 1061973B
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Abstract
本申请描述了式I的含内酰胺的化合物及其衍生物：P4-P-M-M-4或其药学上可接受的盐形式，其中环P，如果存在，是5-7元碳环或杂环，环M是5-7元碳环或杂环。本发明的化合物可用作胰蛋白酶样丝氨酸蛋白酶，特别是因子Xa的抑制剂。
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US324165 | 1981-11-23 | ||
| US32416501P | 2001-09-21 | 2001-09-21 | |
| PCT/US2002/029491 WO2003026652A1 (en) | 2001-09-21 | 2002-09-17 | Lactam-containing compounds and derivatives thereof as factor xa inhibitors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| HK1061973A1 HK1061973A1 (zh) | 2004-10-15 |
| HK1061973B true HK1061973B (zh) | 2010-02-05 |
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