GT201000100A - Productos quimioterapéuticos cristalinos - Google Patents

Productos quimioterapéuticos cristalinos

Info

Publication number
GT201000100A
GT201000100A GT201000100A GT201000100A GT201000100A GT 201000100 A GT201000100 A GT 201000100A GT 201000100 A GT201000100 A GT 201000100A GT 201000100 A GT201000100 A GT 201000100A GT 201000100 A GT201000100 A GT 201000100A
Authority
GT
Guatemala
Prior art keywords
crystal
chemotherapeutic products
chemotherapeutic
products
indazol
Prior art date
Application number
GT201000100A
Other languages
English (en)
Inventor
Michael J Rozema
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of GT201000100A publication Critical patent/GT201000100A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56Benzopyrazoles; Hydrogenated benzopyrazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

FORMA CRISTALINA DE N-(4-(3-AMINO-1H-INDAZOL-4-IL)FENIL)-N'-(2-FLUORO-5-METILFENIL)UREA, MANERAS PARA ELABORARLA, FORMULACIONES QUE COMPRENDEN A LA MISMA Y ELABORADAS CON LA MISMA Y MÉTODOS DE TRATAMIENTO DE PACIENTES QUE PADECEN UNA ENFERMEDAD PARA USARLA.
GT201000100A 2007-10-19 2010-04-16 Productos quimioterapéuticos cristalinos GT201000100A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US98125307P 2007-10-19 2007-10-19

Publications (1)

Publication Number Publication Date
GT201000100A true GT201000100A (es) 2012-04-12

Family

ID=40174807

Family Applications (1)

Application Number Title Priority Date Filing Date
GT201000100A GT201000100A (es) 2007-10-19 2010-04-16 Productos quimioterapéuticos cristalinos

Country Status (18)

Country Link
US (1) US7960564B2 (es)
EP (1) EP2195301A1 (es)
JP (1) JP2011500707A (es)
KR (1) KR20100085987A (es)
CN (1) CN101827824B (es)
AU (1) AU2008312533A1 (es)
BR (1) BRPI0818334A2 (es)
CA (1) CA2699354A1 (es)
CO (1) CO6280484A2 (es)
CR (1) CR11443A (es)
DO (1) DOP2010000112A (es)
EC (1) ECSP10010176A (es)
GT (1) GT201000100A (es)
MX (1) MX2010004290A (es)
PA (1) PA8800601A1 (es)
RU (1) RU2010119919A (es)
UA (1) UA99489C2 (es)
WO (1) WO2009052230A1 (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10166142B2 (en) 2010-01-29 2019-01-01 Forsight Vision4, Inc. Small molecule delivery with implantable therapeutic device
CA2818612C (en) 2010-11-19 2020-12-29 Forsight Vision4, Inc. Therapeutic agent formulations for implanted devices
AU2014236455B2 (en) 2013-03-14 2018-07-12 Forsight Vision4, Inc. Systems for sustained intraocular delivery of low solubility compounds from a port delivery system implant
AU2015301054B2 (en) 2014-08-08 2020-05-14 Forsight Vision4, Inc. Stable and soluble formulations of receptor tyrosine kinase inhibitors, and methods of preparation thereof

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7297709B2 (en) * 2003-05-22 2007-11-20 Abbott Laboratories Indazole, benzisoxazole, and benzisothiazole kinase inhibitors
EP2246333B1 (en) 2003-05-22 2012-10-24 Abbott Laboratories Indazole, benzisoxazole, and benzisothiazole kinase inhibitors
DE102005033100B3 (de) * 2005-07-15 2007-01-25 Sanofi-Aventis Deutschland Gmbh Neues 1,4-Benzothiazepin-1,1-Dioxidderivat mit verbesserten Eigenschaften, diese Verbindung enthaltene Arzneimittel und Verfahren zu deren Herstellung
EP1925941B1 (en) * 2005-08-01 2012-11-28 Eisai R&D Management Co., Ltd. Method for prediction of the efficacy of vascularization inhibitor
US9006240B2 (en) * 2005-08-02 2015-04-14 Eisai R&D Management Co., Ltd. Method for assay on the effect of vascularization inhibitor
CN101346128B (zh) 2005-10-25 2013-10-02 雅培制药有限公司 包含低水溶解度药物的配方及其使用方法
WO2007076358A1 (en) * 2005-12-23 2007-07-05 Alcon, Inc. PHARMACEUTICAL FORMULATION FOR DELIVERY OF RECEPTOR TYROSINE KINASE INHIBITING (RTKi) COMPOUNDS TO THE EYE
US20070173538A1 (en) * 2005-12-23 2007-07-26 Alcon, Inc. PHARMACEUTICAL FORMULATION FOR DELIVERY OF RECEPTOR TYROSINE KINASE INHIBITING (RTKi) COMPOUNDS TO THE EYE
MX2009004861A (es) * 2006-11-09 2009-05-21 Abbott Gmbh & Co Kg Forma de dosificacion farmaceutica para la administracion oral de inhibidor de tirosina quinasa.

Also Published As

Publication number Publication date
CO6280484A2 (es) 2011-05-20
CN101827824A (zh) 2010-09-08
EP2195301A1 (en) 2010-06-16
PA8800601A1 (es) 2009-05-15
CA2699354A1 (en) 2009-04-23
KR20100085987A (ko) 2010-07-29
MX2010004290A (es) 2010-04-30
ECSP10010176A (es) 2010-06-29
WO2009052230A1 (en) 2009-04-23
US20090124815A1 (en) 2009-05-14
AU2008312533A1 (en) 2009-04-23
RU2010119919A (ru) 2011-11-27
US7960564B2 (en) 2011-06-14
BRPI0818334A2 (pt) 2017-05-16
CN101827824B (zh) 2012-10-03
DOP2010000112A (es) 2010-07-15
UA99489C2 (en) 2012-08-27
JP2011500707A (ja) 2011-01-06
CR11443A (es) 2010-09-27

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