UA99489C2 - Crystalline chemotherapeutic agent - Google Patents

Crystalline chemotherapeutic agent

Info

Publication number
UA99489C2
UA99489C2 UAA201006027A UAA201006027A UA99489C2 UA 99489 C2 UA99489 C2 UA 99489C2 UA A201006027 A UAA201006027 A UA A201006027A UA A201006027 A UAA201006027 A UA A201006027A UA 99489 C2 UA99489 C2 UA 99489C2
Authority
UA
Ukraine
Prior art keywords
chemotherapeutic agent
crystalline
crystalline chemotherapeutic
indazol
methylphenyl
Prior art date
Application number
UAA201006027A
Other languages
English (en)
Inventor
Майкл Дж. Розема
Original Assignee
Эбботт Леборетриз
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Эбботт Леборетриз filed Critical Эбботт Леборетриз
Publication of UA99489C2 publication Critical patent/UA99489C2/ru

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56Benzopyrazoles; Hydrogenated benzopyrazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
UAA201006027A 2007-10-19 2008-10-16 Crystalline chemotherapeutic agent UA99489C2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US98125307P 2007-10-19 2007-10-19

Publications (1)

Publication Number Publication Date
UA99489C2 true UA99489C2 (en) 2012-08-27

Family

ID=40174807

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA201006027A UA99489C2 (en) 2007-10-19 2008-10-16 Crystalline chemotherapeutic agent

Country Status (18)

Country Link
US (1) US7960564B2 (ru)
EP (1) EP2195301A1 (ru)
JP (1) JP2011500707A (ru)
KR (1) KR20100085987A (ru)
CN (1) CN101827824B (ru)
AU (1) AU2008312533A1 (ru)
BR (1) BRPI0818334A2 (ru)
CA (1) CA2699354A1 (ru)
CO (1) CO6280484A2 (ru)
CR (1) CR11443A (ru)
DO (1) DOP2010000112A (ru)
EC (1) ECSP10010176A (ru)
GT (1) GT201000100A (ru)
MX (1) MX2010004290A (ru)
PA (1) PA8800601A1 (ru)
RU (1) RU2010119919A (ru)
UA (1) UA99489C2 (ru)
WO (1) WO2009052230A1 (ru)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10166142B2 (en) 2010-01-29 2019-01-01 Forsight Vision4, Inc. Small molecule delivery with implantable therapeutic device
WO2012068549A2 (en) 2010-11-19 2012-05-24 Forsight Vision4, Inc. Therapeutic agent formulations for implanted devices
US9968603B2 (en) 2013-03-14 2018-05-15 Forsight Vision4, Inc. Systems for sustained intraocular delivery of low solubility compounds from a port delivery system implant
JP2017524034A (ja) 2014-08-08 2017-08-24 フォーサイト・ビジョン フォー・インコーポレーテッドForsight Vision4, Inc. 受容体型チロシンキナーゼ阻害剤の安定で可溶な製剤およびその調製の方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7297709B2 (en) * 2003-05-22 2007-11-20 Abbott Laboratories Indazole, benzisoxazole, and benzisothiazole kinase inhibitors
JP4810427B2 (ja) 2003-05-22 2011-11-09 アボット・ラボラトリーズ インダゾール、ベンズイソオキサゾールおよびベンズイソチアゾールキナーゼ阻害剤
DE102005033100B3 (de) * 2005-07-15 2007-01-25 Sanofi-Aventis Deutschland Gmbh Neues 1,4-Benzothiazepin-1,1-Dioxidderivat mit verbesserten Eigenschaften, diese Verbindung enthaltene Arzneimittel und Verfahren zu deren Herstellung
US20100105031A1 (en) * 2005-08-01 2010-04-29 Esai R & D Management Co., Ltd. Method for prediction of the efficacy of vascularization inhibitor
JP4989476B2 (ja) * 2005-08-02 2012-08-01 エーザイ・アール・アンド・ディー・マネジメント株式会社 血管新生阻害物質の効果を検定する方法
US20070104780A1 (en) 2005-10-25 2007-05-10 Lipari John M Formulation comprising a drug of low water solubility and method of use thereof
US20070173538A1 (en) * 2005-12-23 2007-07-26 Alcon, Inc. PHARMACEUTICAL FORMULATION FOR DELIVERY OF RECEPTOR TYROSINE KINASE INHIBITING (RTKi) COMPOUNDS TO THE EYE
JP2009521493A (ja) * 2005-12-23 2009-06-04 アルコン,インコーポレイテッド 眼への受容体チロシンキナーゼ阻害(RTKi)化合物の送達のための医薬製剤
EP2089003A1 (en) * 2006-11-09 2009-08-19 Abbott GmbH & Co. KG Pharmaceutical dosage form for oral administration of tyrosine kinase inhibitor

Also Published As

Publication number Publication date
US20090124815A1 (en) 2009-05-14
AU2008312533A1 (en) 2009-04-23
CR11443A (es) 2010-09-27
EP2195301A1 (en) 2010-06-16
PA8800601A1 (es) 2009-05-15
MX2010004290A (es) 2010-04-30
CN101827824A (zh) 2010-09-08
KR20100085987A (ko) 2010-07-29
GT201000100A (es) 2012-04-12
CO6280484A2 (es) 2011-05-20
CA2699354A1 (en) 2009-04-23
RU2010119919A (ru) 2011-11-27
BRPI0818334A2 (pt) 2017-05-16
ECSP10010176A (es) 2010-06-29
WO2009052230A1 (en) 2009-04-23
JP2011500707A (ja) 2011-01-06
CN101827824B (zh) 2012-10-03
US7960564B2 (en) 2011-06-14
DOP2010000112A (es) 2010-07-15

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