GR33806B - Μεθοδος δια την παρασκευην παραγωγων της βενζοδιαζεπινης. - Google Patents
Μεθοδος δια την παρασκευην παραγωγων της βενζοδιαζεπινης.Info
- Publication number
- GR33806B GR33806B GR670133806A GR670133806A GR33806B GR 33806 B GR33806 B GR 33806B GR 670133806 A GR670133806 A GR 670133806A GR 670133806 A GR670133806 A GR 670133806A GR 33806 B GR33806 B GR 33806B
- Authority
- GR
- Greece
- Prior art keywords
- alkyl
- preparation
- benzodiazepine
- producers
- lower alkylene
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/74—Quinazolines; Hydrogenated quinazolines with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached to ring carbon atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C249/00—Preparation of compounds containing nitrogen atoms doubly-bound to a carbon skeleton
- C07C249/04—Preparation of compounds containing nitrogen atoms doubly-bound to a carbon skeleton of oximes
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/74—Quinazolines; Hydrogenated quinazolines with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached to ring carbon atoms of the hetero ring
- C07D239/76—N-oxides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
- C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
- C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
- C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
- C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
- C07D243/20—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
- C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
- C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
- C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
- C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
- C07D243/24—Oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
έθοδος δια την παρασκευή παραγώγων της βενζοδιαζεπίνης χαρακτηριζόμενη εκ του ότι θερμαίνομε μιαν οξίμην του γενικού τύπου (1) εις τον οποίον τα R1 και R2 σημαίνουν έκαστο κατώτερο αλκύλιο ή ομού κατώτερο αλκυλένιο, άζα- κατώτερο αλκυλένιον, Ν-κατώτερο αλκυλο-άζα- κατώτερο αλκυλένιο, όξα- κατώτερο αλκυλένιο ή θεία-κατώτερο αλκυλένιο, τα R3 και R4και R5 σημαίνουν υδρογόνο, αλογόνο, κατώτερο αλκύλιο κατώτερο αλκόξυ, κυάνιο, τριφθορομεθύλιο ή νίτρο, τα R6 και R7σημιάνουν υδρογόνο ή κατώτερο αλκύλιο και το R10 σημαίνει κατώτερο αλκύλιο ή αραλκύλιον.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US52155166A | 1966-01-19 | 1966-01-19 |
Publications (1)
Publication Number | Publication Date |
---|---|
GR33806B true GR33806B (el) | 1968-02-06 |
Family
ID=24077176
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
GR670133806A GR33806B (el) | 1966-01-19 | 1967-01-17 | Μεθοδος δια την παρασκευην παραγωγων της βενζοδιαζεπινης. |
GR670135752A GR35752B (el) | 1966-01-19 | 1967-01-17 | Μεθοδος δια την παρασκευην παραγωγων της βενζοδιαζεπινης. |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
GR670135752A GR35752B (el) | 1966-01-19 | 1967-01-17 | Μεθοδος δια την παρασκευην παραγωγων της βενζοδιαζεπινης. |
Country Status (16)
Country | Link |
---|---|
US (1) | US3446806A (el) |
JP (1) | JPS4938814B1 (el) |
BE (2) | BE692378A (el) |
CH (3) | CH560692A5 (el) |
DE (2) | DE1695176A1 (el) |
DK (4) | DK114556B (el) |
ES (2) | ES335789A1 (el) |
FI (1) | FI47576C (el) |
FR (2) | FR1507878A (el) |
GB (2) | GB1144516A (el) |
GR (2) | GR33806B (el) |
IL (2) | IL27189A (el) |
MY (2) | MY6900383A (el) |
NL (3) | NL6700785A (el) |
OA (1) | OA02391A (el) |
SE (4) | SE321233B (el) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4601839A (en) * | 1978-06-19 | 1986-07-22 | The B. F. Goodrich Company | Stabilized polymers, novel stabilizers, and synthesis thereof |
US4310429A (en) * | 1978-06-19 | 1982-01-12 | The B. F. Goodrich Company | Stabilized polymers, novel stabilizers, and synthesis thereof |
US4472435A (en) * | 1980-07-31 | 1984-09-18 | Hoffman-La Roche Inc. | Benzophenone derivatives useful in treating heart failure |
WO1995024394A1 (en) * | 1994-03-08 | 1995-09-14 | Takeda Chemical Industries, Ltd. | Quinoline or quinazoline derivatives as anti-inflammatory agents, in particular for treating arthritis |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3267110A (en) * | 1960-06-03 | 1966-08-16 | Smith Kline French Lab | Trifluoromethyl substituted o-aminophenyl ketones |
US3321467A (en) * | 1963-11-27 | 1967-05-23 | Hoffmann La Roche | 3-halo-1, 4-benzodiazepin-2-ones |
-
0
- NL NL131198D patent/NL131198C/xx active
-
1966
- 1966-01-19 US US521551A patent/US3446806A/en not_active Expired - Lifetime
- 1966-12-27 CH CH438369A patent/CH560692A5/xx not_active IP Right Cessation
- 1966-12-27 CH CH1862266A patent/CH553193A/de not_active IP Right Cessation
- 1966-12-29 IL IL27189A patent/IL27189A/xx unknown
- 1966-12-29 DE DE19661695176 patent/DE1695176A1/de active Pending
-
1967
- 1967-01-04 IL IL27212A patent/IL27212A/xx unknown
- 1967-01-06 CH CH20067A patent/CH461517A/de unknown
- 1967-01-10 BE BE692378D patent/BE692378A/xx unknown
- 1967-01-10 DE DE19671618486 patent/DE1618486A1/de active Pending
- 1967-01-11 GB GB1581/67A patent/GB1144516A/en not_active Expired
- 1967-01-11 GB GB1580/67A patent/GB1144515A/en not_active Expired
- 1967-01-12 FI FI670076A patent/FI47576C/fi active
- 1967-01-13 FR FR90972A patent/FR1507878A/fr not_active Expired
- 1967-01-13 BE BE692558D patent/BE692558A/xx unknown
- 1967-01-16 FR FR91188A patent/FR1508490A/fr not_active Expired
- 1967-01-17 GR GR670133806A patent/GR33806B/el unknown
- 1967-01-17 GR GR670135752A patent/GR35752B/el unknown
- 1967-01-18 DK DK29967AA patent/DK114556B/da unknown
- 1967-01-18 DK DK29867AA patent/DK120347B/da unknown
- 1967-01-18 NL NL6700785A patent/NL6700785A/xx unknown
- 1967-01-18 NL NL6700786A patent/NL6700786A/xx unknown
- 1967-01-18 ES ES0335789A patent/ES335789A1/es not_active Expired
- 1967-01-18 ES ES335788A patent/ES335788A1/es not_active Expired
- 1967-01-19 SE SE811/67A patent/SE321233B/xx unknown
- 1967-01-19 SE SE02828/69A patent/SE353717B/xx unknown
- 1967-01-19 SE SE00810/67A patent/SE335858B/xx unknown
- 1967-01-19 SE SE7008427A patent/SE386168B/xx unknown
- 1967-03-30 OA OA52856A patent/OA02391A/xx unknown
- 1967-10-27 DK DK537067AA patent/DK120392B/da unknown
- 1967-11-21 DK DK582367AA patent/DK119656B/da unknown
-
1969
- 1969-02-08 JP JP44009665A patent/JPS4938814B1/ja active Pending
- 1969-12-31 MY MY1969383A patent/MY6900383A/xx unknown
- 1969-12-31 MY MY1969384A patent/MY6900384A/xx unknown
Also Published As
Publication number | Publication date |
---|---|
DK120392B (da) | 1971-05-24 |
GR35752B (el) | 1968-10-25 |
CH553193A (en) | 1974-08-30 |
FI47576B (el) | 1973-10-01 |
DK120347B (da) | 1971-05-17 |
DK119656B (da) | 1971-02-08 |
FR1507878A (fr) | 1967-12-29 |
BE692378A (el) | 1967-07-10 |
FR1508490A (fr) | 1968-01-05 |
DE1695176A1 (de) | 1970-04-16 |
ES335789A1 (es) | 1967-12-16 |
MY6900384A (en) | 1969-12-31 |
IL27212A (en) | 1971-04-28 |
ES335788A1 (es) | 1968-03-16 |
OA02391A (fr) | 1970-05-05 |
JPS4938814B1 (el) | 1974-10-21 |
US3446806A (en) | 1969-05-27 |
MY6900383A (en) | 1969-12-31 |
SE335858B (el) | 1971-06-14 |
CH461517A (de) | 1968-08-31 |
DE1618486A1 (de) | 1971-04-01 |
NL131198C (el) | |
SE386168B (sv) | 1976-08-02 |
NL6700785A (el) | 1967-07-20 |
GB1144515A (en) | 1969-03-05 |
CH560692A5 (el) | 1975-04-15 |
GB1144516A (en) | 1969-03-05 |
BE692558A (el) | 1967-07-13 |
SE353717B (el) | 1973-02-12 |
NL6700786A (el) | 1967-07-20 |
FI47576C (fi) | 1974-01-10 |
DK114556B (da) | 1969-07-14 |
IL27189A (en) | 1971-01-28 |
SE321233B (el) | 1970-03-02 |
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