GB1581015A - Benzylpyrimidines - Google Patents

Benzylpyrimidines Download PDF

Info

Publication number
GB1581015A
GB1581015A GB17757/78A GB1775778A GB1581015A GB 1581015 A GB1581015 A GB 1581015A GB 17757/78 A GB17757/78 A GB 17757/78A GB 1775778 A GB1775778 A GB 1775778A GB 1581015 A GB1581015 A GB 1581015A
Authority
GB
United Kingdom
Prior art keywords
acid
allyl
formula
group
benzylpyrimidine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB17757/78A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by F Hoffmann La Roche AG filed Critical F Hoffmann La Roche AG
Publication of GB1581015A publication Critical patent/GB1581015A/en
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • C07D239/49Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
GB17757/78A 1977-05-05 1978-05-04 Benzylpyrimidines Expired GB1581015A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
LU77268A LU77268A1 (US07714131-20100511-C00001.png) 1977-05-05 1977-05-05

Publications (1)

Publication Number Publication Date
GB1581015A true GB1581015A (en) 1980-12-10

Family

ID=19728558

Family Applications (1)

Application Number Title Priority Date Filing Date
GB17757/78A Expired GB1581015A (en) 1977-05-05 1978-05-04 Benzylpyrimidines

Country Status (13)

Country Link
US (1) US4191758A (US07714131-20100511-C00001.png)
JP (1) JPS53137977A (US07714131-20100511-C00001.png)
AU (1) AU3555378A (US07714131-20100511-C00001.png)
BE (1) BE866652A (US07714131-20100511-C00001.png)
CA (1) CA1075694A (US07714131-20100511-C00001.png)
DE (1) DE2819211A1 (US07714131-20100511-C00001.png)
DK (1) DK195478A (US07714131-20100511-C00001.png)
FR (1) FR2389612A1 (US07714131-20100511-C00001.png)
GB (1) GB1581015A (US07714131-20100511-C00001.png)
LU (1) LU77268A1 (US07714131-20100511-C00001.png)
NL (1) NL7804769A (US07714131-20100511-C00001.png)
SE (1) SE7805187L (US07714131-20100511-C00001.png)
ZA (1) ZA782454B (US07714131-20100511-C00001.png)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT99514B (pt) * 1990-11-14 1999-04-30 Chiron Corp Processo de preparacao de compostos para o tratamento de infeccoes fungicas

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3996356A (en) * 1969-07-02 1976-12-07 Hoffmann-La Roche Inc. Composition containing 5-sulfanilamido-3,4-dimethylisoxazole and a trimethoxybenzyl pyrimidine
BE795023A (fr) * 1972-02-07 1973-08-06 Hoffmann La Roche Nouvelles benzylpyrimidines
US3985876A (en) * 1973-01-05 1976-10-12 Burroughs Wellcome Co. Chemotherapeutic solutions containing a sulphur and a salt of a 2,4-diamino-5-benzylpyrimidine
US4033962A (en) * 1975-06-26 1977-07-05 Hoffman-La Roche Inc. 2,4-Diamino-pyrimidine derivatives and processes

Also Published As

Publication number Publication date
SE7805187L (sv) 1978-11-06
ZA782454B (en) 1979-04-25
DK195478A (da) 1978-11-06
LU77268A1 (US07714131-20100511-C00001.png) 1979-01-18
JPS53137977A (en) 1978-12-01
BE866652A (fr) 1978-11-03
DE2819211A1 (de) 1978-11-16
AU3555378A (en) 1979-11-01
FR2389612A1 (US07714131-20100511-C00001.png) 1978-12-01
NL7804769A (nl) 1978-11-07
US4191758A (en) 1980-03-04
CA1075694A (en) 1980-04-15

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Legal Events

Date Code Title Description
CSNS Application of which complete specification have been accepted and published, but patent is not sealed