GB1445697A - 3-aminoisothiazolo-3,4-d-pyrimidines - Google Patents
3-aminoisothiazolo-3,4-d-pyrimidinesInfo
- Publication number
- GB1445697A GB1445697A GB4572573A GB4572573A GB1445697A GB 1445697 A GB1445697 A GB 1445697A GB 4572573 A GB4572573 A GB 4572573A GB 4572573 A GB4572573 A GB 4572573A GB 1445697 A GB1445697 A GB 1445697A
- Authority
- GB
- United Kingdom
- Prior art keywords
- aminoisothiazolo
- pyrimidines
- oct
- hydrogen
- optionally substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- 239000001257 hydrogen Substances 0.000 abstract 2
- 125000004435 hydrogen atom Chemical class [H]* 0.000 abstract 2
- 238000007243 oxidative cyclization reaction Methods 0.000 abstract 2
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 1
- RAHZWNYVWXNFOC-UHFFFAOYSA-N Sulphur dioxide Chemical group O=S=O RAHZWNYVWXNFOC-UHFFFAOYSA-N 0.000 abstract 1
- 125000002252 acyl group Chemical group 0.000 abstract 1
- 125000003342 alkenyl group Chemical group 0.000 abstract 1
- 239000002260 anti-inflammatory agent Substances 0.000 abstract 1
- 125000003710 aryl alkyl group Chemical group 0.000 abstract 1
- 239000003795 chemical substances by application Substances 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 239000002934 diuretic Substances 0.000 abstract 1
- 229940030606 diuretics Drugs 0.000 abstract 1
- AEOCXXJPGCBFJA-UHFFFAOYSA-N ethionamide Chemical compound CCC1=CC(C(N)=S)=CC=N1 AEOCXXJPGCBFJA-UHFFFAOYSA-N 0.000 abstract 1
- 239000000417 fungicide Substances 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- 239000012442 inert solvent Substances 0.000 abstract 1
- 239000000375 suspending agent Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19722248231 DE2248231A1 (de) | 1972-10-02 | 1972-10-02 | 3-aminoisothiazolo eckige klammer auf 3,4-d eckige klammer zu pyrimidine |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB1445697A true GB1445697A (en) | 1976-08-11 |
Family
ID=5857973
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB4572573A Expired GB1445697A (en) | 1972-10-02 | 1973-10-01 | 3-aminoisothiazolo-3,4-d-pyrimidines |
Country Status (4)
| Country | Link |
|---|---|
| CH (1) | CH578008A5 (enrdf_load_stackoverflow) |
| DE (1) | DE2248231A1 (enrdf_load_stackoverflow) |
| FR (1) | FR2201097B1 (enrdf_load_stackoverflow) |
| GB (1) | GB1445697A (enrdf_load_stackoverflow) |
Cited By (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1998005670A1 (de) * | 1996-07-31 | 1998-02-12 | Bayer Aktiengesellschaft | Substituierte n-isothiazolyl-(thio)amide |
| WO2005077959A1 (en) * | 2004-02-11 | 2005-08-25 | Smithkline Beecham Corporation | Pth agonists |
| WO2010109328A1 (en) * | 2009-03-23 | 2010-09-30 | Glenmark Pharmaceuticals, S.A. | Isothiazolo-pyrimidinedione derivatives as trpa1 modulators |
| US8507503B2 (en) | 2009-03-23 | 2013-08-13 | Glenmark Pharmaceuticals S.A. | Thienopyrimidinedione derivatives as TRPA1 modulators |
| US8623880B2 (en) | 2009-03-23 | 2014-01-07 | Glenmark Pharmaceuticals S.A. | Fused pyrimidine-dione derivatives as TRPA1 modulators |
| US9000159B2 (en) | 2009-03-23 | 2015-04-07 | Glenmark Pharmaceuticals S.A. | Fused pyrimidine-dione derivatives as TRPA1 modulators |
| US9458173B2 (en) | 2012-06-08 | 2016-10-04 | Glenmark Pharmaceuticals S.A. | Amides of 2-amino-4-arylthiazole compounds and their salts |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5826356B2 (ja) * | 1973-11-12 | 1983-06-02 | 武田薬品工業株式会社 | イソチアゾロ （３，４−ｄ） ピリミジンルイ ノ セイゾウホウ |
| JPS58152890A (ja) * | 1982-03-08 | 1983-09-10 | Takeda Chem Ind Ltd | イソキサゾロピリミジン誘導体 |
-
1972
- 1972-10-02 DE DE19722248231 patent/DE2248231A1/de not_active Withdrawn
-
1973
- 1973-09-28 CH CH1391773A patent/CH578008A5/xx not_active IP Right Cessation
- 1973-10-01 GB GB4572573A patent/GB1445697A/en not_active Expired
- 1973-10-01 FR FR7335018A patent/FR2201097B1/fr not_active Expired
Cited By (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1998005670A1 (de) * | 1996-07-31 | 1998-02-12 | Bayer Aktiengesellschaft | Substituierte n-isothiazolyl-(thio)amide |
| WO2005077959A1 (en) * | 2004-02-11 | 2005-08-25 | Smithkline Beecham Corporation | Pth agonists |
| EP1713815A4 (en) * | 2004-02-11 | 2009-03-11 | Smithkline Beecham Corp | PTH AGONISTS |
| WO2010109328A1 (en) * | 2009-03-23 | 2010-09-30 | Glenmark Pharmaceuticals, S.A. | Isothiazolo-pyrimidinedione derivatives as trpa1 modulators |
| CN102395592A (zh) * | 2009-03-23 | 2012-03-28 | 格兰马克药品股份有限公司 | 作为trpa1调节剂的异噻唑并嘧啶二酮衍生物 |
| US8507503B2 (en) | 2009-03-23 | 2013-08-13 | Glenmark Pharmaceuticals S.A. | Thienopyrimidinedione derivatives as TRPA1 modulators |
| US8575178B2 (en) | 2009-03-23 | 2013-11-05 | Glenmark Pharmaceuticals S.A. | Isothiazolo-pyrimidinedione derivatives as TRPA1 modulators |
| US8623880B2 (en) | 2009-03-23 | 2014-01-07 | Glenmark Pharmaceuticals S.A. | Fused pyrimidine-dione derivatives as TRPA1 modulators |
| US8987278B2 (en) | 2009-03-23 | 2015-03-24 | Glenmark Pharmaceuticals S.A. | Thienopyrimidinedione derivatives as TRPA1 modulators |
| US9000159B2 (en) | 2009-03-23 | 2015-04-07 | Glenmark Pharmaceuticals S.A. | Fused pyrimidine-dione derivatives as TRPA1 modulators |
| US9474758B2 (en) | 2009-03-23 | 2016-10-25 | Glenmark Pharmaceuticals, S.A. | Thienopyrimidinedione derivatives as TRPA1 modulators |
| US9458173B2 (en) | 2012-06-08 | 2016-10-04 | Glenmark Pharmaceuticals S.A. | Amides of 2-amino-4-arylthiazole compounds and their salts |
Also Published As
| Publication number | Publication date |
|---|---|
| FR2201097B1 (enrdf_load_stackoverflow) | 1976-10-22 |
| CH578008A5 (enrdf_load_stackoverflow) | 1976-07-30 |
| DE2248231A1 (de) | 1974-04-11 |
| FR2201097A1 (enrdf_load_stackoverflow) | 1974-04-26 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PS | Patent sealed | ||
| PCNP | Patent ceased through non-payment of renewal fee |