GB1272527A - Propanolamine derivatives - Google Patents

Propanolamine derivatives

Info

Publication number
GB1272527A
GB1272527A GB1739670A GB1739670A GB1272527A GB 1272527 A GB1272527 A GB 1272527A GB 1739670 A GB1739670 A GB 1739670A GB 1739670 A GB1739670 A GB 1739670A GB 1272527 A GB1272527 A GB 1272527A
Authority
GB
United Kingdom
Prior art keywords
alkyl
april
propanolamine derivatives
compounds
frosst
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB1739670A
Inventor
Ronald Stiles Stuart
Burton Kendall Wasson
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck Frosst Canada and Co
Original Assignee
Charles E Frosst and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Charles E Frosst and Co filed Critical Charles E Frosst and Co
Publication of GB1272527A publication Critical patent/GB1272527A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/08—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
    • C07D295/096—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

1,272,527. Propanolamine derivatives. CHARLES E. FROSST & CO. 13 April, 1970 [18 April, 1969], No. 17396/70. Heading C2C. Compounds of the general formula (R<SP>1</SP>, R<SP>2</SP>. R<SP>4</SP>=H, C 1-3 alkyl; R<SP>3</SP>=H, PhCO, C 2-4 alkanoyl; R<SP>5</SP> = C 1-20 alkyl, C 3-10 cycloalkyl, polycycloalkyl, C 2-6 alkenyl or alkynyl, phenyl- (C 1-5 alkyl) optionally substituted by one or more substituents selected from Cl, Br, OH, C 1-3 alkyl or alkoxy) and their salts are prepared by the following routes optionally followed by esterification, salt formation and/or resolution. The above compounds are #-adrenergic blocking agents, and may be administered in the form of pharmaceutical preparations containing them in association with a carrier.
GB1739670A 1969-04-18 1970-04-13 Propanolamine derivatives Expired GB1272527A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CA049,141A CA954861A (en) 1969-04-18 1969-04-18 1-(morpholino-phenoxy)-3-(substituted amino) propan-2-01s

Publications (1)

Publication Number Publication Date
GB1272527A true GB1272527A (en) 1972-05-03

Family

ID=4085157

Family Applications (1)

Application Number Title Priority Date Filing Date
GB1739670A Expired GB1272527A (en) 1969-04-18 1970-04-13 Propanolamine derivatives

Country Status (6)

Country Link
CA (1) CA954861A (en)
CH (1) CH542869A (en)
DE (1) DE2018522A1 (en)
FR (1) FR2042344B1 (en)
GB (1) GB1272527A (en)
NL (1) NL7005505A (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE402764B (en) 1975-06-04 1978-07-17 Haessle Ab PROCEDURE FOR PRODUCING NEW HEART ACTIVE ASSOCIATIONS

Also Published As

Publication number Publication date
CA954861A (en) 1974-09-17
FR2042344B1 (en) 1973-12-21
NL7005505A (en) 1970-10-20
CH542869A (en) 1973-10-15
DE2018522A1 (en) 1970-11-12
FR2042344A1 (en) 1971-02-12

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Legal Events

Date Code Title Description
PS Patent sealed
PCNP Patent ceased through non-payment of renewal fee
PCNP Patent ceased through non-payment of renewal fee
PCNP Patent ceased through non-payment of renewal fee

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