GB1141487A - Derivatives of 2-anilino-1,3-diazacyclopentene-(2) - Google Patents
Derivatives of 2-anilino-1,3-diazacyclopentene-(2)Info
- Publication number
- GB1141487A GB1141487A GB44068/66A GB4406866A GB1141487A GB 1141487 A GB1141487 A GB 1141487A GB 44068/66 A GB44068/66 A GB 44068/66A GB 4406866 A GB4406866 A GB 4406866A GB 1141487 A GB1141487 A GB 1141487A
- Authority
- GB
- United Kingdom
- Prior art keywords
- prepared
- formula
- compounds
- och
- hydrochloride
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/44—Nitrogen atoms not forming part of a nitro radical
- C07D233/50—Nitrogen atoms not forming part of a nitro radical with carbocyclic radicals directly attached to said nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
1,141,487. Substituted imidazolines. BOEHRINGER INGELHEIM G.m.b.H. 3 Oct., 1966 [1 Oct., 1965], No. 44068/66. Heading C2C. [Also in Division A5] Novel compounds of the formula (II) (wherein R<SP>1</SP> is F, Cl, Br, CH 3 or OCH 3 , and R<SP>2</SP> is F, Cl, Br, CF 3 , CN, CH 3 or OCH 3 ; one of R<SP>1</SP> and R<SP>2</SP> being CH 3 or OCH 3 , except that when R<SP>1</SP> is Cl, R<SP>2</SP> is not 4- or 6-CH 3 , and when R<SP>1</SP> is CH 3 , R<SP>2</SP> is not 3- or 4- Cl) and acidaddition salts thereof are prepared (1) by reaction of isothiouranium salts of the Formula (III) (wherein R<SP>3</SP> is lower alkyl and X is an anion) or corresponding thioureas with ethylenediamine; (2) by pyrolysis of compounds of the formula (V) (wherein Y is O or S). Compounds of the formula (III) are prepared by heating appropriately substituted anilines and ammonium thiocyanate to give the corresponding N-phenyl-thioureas and heating these with alkylating agents. Compounds of the formula (V) are prepared by reaction of appropriately substituted phenyl isocyanates or isothiocyanates with ethylenediamine. 3 - Bromo - 2 - methyl - aniline hydrochloride is prepared by hydrogenating 2 - bromo - 6 - nitro - toluene (prepared from the 2-amino compound and cuprous bromide) and converting the free base to the hydrochloride. Similarly are prepared 2-chloro-3-methyl-aniline and 3- amino - 4 - chloro - anisole hydrochloride.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DEB0083964 | 1965-10-01 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB1141487A true GB1141487A (en) | 1969-01-29 |
Family
ID=6982208
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB44068/66A Expired GB1141487A (en) | 1965-10-01 | 1966-10-03 | Derivatives of 2-anilino-1,3-diazacyclopentene-(2) |
Country Status (13)
| Country | Link |
|---|---|
| BE (1) | BE687656A (en) |
| CH (1) | CH484912A (en) |
| CS (2) | CS155146B2 (en) |
| DK (1) | DK115627B (en) |
| ES (1) | ES331789A1 (en) |
| FI (1) | FI46959C (en) |
| FR (2) | FR1506407A (en) |
| GB (1) | GB1141487A (en) |
| IL (1) | IL26613A (en) |
| IT (1) | IT7949465A0 (en) |
| NL (3) | NL156398B (en) |
| PL (1) | PL79137B1 (en) |
| SE (1) | SE331280B (en) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BE755270A (en) * | 1969-08-27 | 1971-02-25 | Sandoz Sa | NEW DERIVATIVES OF BENZO (CD) INDOLE, THEIR PREPARATION AND MEDICINAL PRODUCTS CONTAINING THESE DERIVATIVES |
| DE2806811A1 (en) * | 1978-02-17 | 1979-08-23 | Boehringer Sohn Ingelheim | NEW SUBSTITUTED 2-PHENYLIMINO-IMIDAZOLIDINE, THEIR ACID-ADDITIONAL SALTS, THESE MEDICINAL PRODUCTS AND METHOD FOR MANUFACTURING THE SAME |
| DE2854659A1 (en) * | 1978-12-18 | 1980-07-10 | Boehringer Sohn Ingelheim | NEW 3,4-DISUBSTITUTED 2-PHENYLIMINO IMIDAZOLIDINES, THEIR ACID ADDITION SALTS, THE MEDICINAL PRODUCTS CONTAINING THEM AND METHOD FOR THE PRODUCTION THEREOF |
| HU192986B (en) | 1984-05-23 | 1987-08-28 | Egyt Gyogyszervegyeszeti Gyar | Process for production of imidasodiline derivatives |
-
1966
- 1966-09-30 NL NL6613829.A patent/NL156398B/en not_active IP Right Cessation
- 1966-09-30 FR FR78365A patent/FR1506407A/en not_active Expired
- 1966-09-30 FR FR78361A patent/FR6998M/fr not_active Expired
- 1966-09-30 CH CH1414166A patent/CH484912A/en not_active IP Right Cessation
- 1966-09-30 ES ES0331789A patent/ES331789A1/en not_active Expired
- 1966-09-30 SE SE13242/66A patent/SE331280B/xx unknown
- 1966-09-30 DK DK506966AA patent/DK115627B/en unknown
- 1966-09-30 BE BE687656D patent/BE687656A/xx not_active IP Right Cessation
- 1966-10-01 CS CS486672*1A patent/CS155146B2/cs unknown
- 1966-10-01 PL PL1966116712A patent/PL79137B1/en unknown
- 1966-10-01 FI FI662577A patent/FI46959C/en active
- 1966-10-01 CS CS629466A patent/CS155145B2/cs unknown
- 1966-10-02 IL IL26613A patent/IL26613A/en unknown
- 1966-10-03 GB GB44068/66A patent/GB1141487A/en not_active Expired
-
1977
- 1977-09-14 NL NL7710062A patent/NL7710062A/en not_active Application Discontinuation
- 1977-09-14 NL NL7710061A patent/NL7710061A/en not_active Application Discontinuation
-
1979
- 1979-06-19 IT IT7949465A patent/IT7949465A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| FI46959B (en) | 1973-05-02 |
| FI46959C (en) | 1973-08-10 |
| IT7949465A0 (en) | 1979-06-19 |
| FR1506407A (en) | 1967-12-22 |
| NL7710062A (en) | 1978-01-31 |
| NL156398B (en) | 1978-04-17 |
| NL6613829A (en) | 1967-04-03 |
| ES331789A1 (en) | 1967-11-01 |
| SE331280B (en) | 1970-12-21 |
| IL26613A (en) | 1970-07-19 |
| DK115627B (en) | 1969-10-27 |
| NL7710061A (en) | 1978-01-31 |
| PL79137B1 (en) | 1975-06-30 |
| FR6998M (en) | 1969-06-02 |
| BE687656A (en) | 1967-03-30 |
| CS155145B2 (en) | 1974-05-30 |
| CH484912A (en) | 1970-01-31 |
| CS155146B2 (en) | 1974-05-30 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| GB1048888A (en) | Cyanine dyestuffs | |
| GB1290388A (en) | ||
| GB1206764A (en) | Poultry feeds containing 5-nitro furyl compounds | |
| GB1141487A (en) | Derivatives of 2-anilino-1,3-diazacyclopentene-(2) | |
| GB1202299A (en) | Imidazoline derivatives | |
| GB1053163A (en) | ||
| GB1144230A (en) | Derivatives of 2-anilino-1,3-diazacyclopentene-(2) | |
| GB1131799A (en) | Substituted thiazolidines | |
| GB1138714A (en) | Pesticidal preparations | |
| GB1230663A (en) | ||
| GB971245A (en) | Method of preparation of heterocyclic compounds | |
| GB1341863A (en) | Thiazole derivatives and their use as plant growth control agents | |
| ES317623A1 (en) | A procedure for the preparation of heterociclic compounds. (Machine-translation by Google Translate, not legally binding) | |
| GB1369386A (en) | Glycidyl-urethane compounds processes for their manufacture and their use | |
| GB1173679A (en) | Water-Insoluble Styryl Dyestuffs and processes for their manufacture and use | |
| ES352647A1 (en) | 2-(4'-chloro-naphthyl(1')-methyl)-imidazoline | |
| GB1199680A (en) | Triazole Compounds, processes for their manufacture and use | |
| GB1143263A (en) | Desyl amines and compositions thereof | |
| ES385424A1 (en) | Thiocarbamoylalkylamino-s-triazine | |
| GB1309274A (en) | Merocyanin dyes | |
| GB1074433A (en) | Merocyanine dyestuffs | |
| GB1103410A (en) | Preparation of 3-amino-1,2,5-thiadiazole | |
| GB1108060A (en) | Indole derivatives and a process for their production | |
| GB1048812A (en) | Substituted amino-guanidines | |
| GB1363038A (en) | Bolism |