FR2967672B1 - Derives de nitrobenzothiazoles, leur preparation et leurs applications therapeutiques - Google Patents

Derives de nitrobenzothiazoles, leur preparation et leurs applications therapeutiques

Info

Publication number
FR2967672B1
FR2967672B1 FR1059602A FR1059602A FR2967672B1 FR 2967672 B1 FR2967672 B1 FR 2967672B1 FR 1059602 A FR1059602 A FR 1059602A FR 1059602 A FR1059602 A FR 1059602A FR 2967672 B1 FR2967672 B1 FR 2967672B1
Authority
FR
France
Prior art keywords
nitrobenzothiazole
derivatives
preparation
therapeutic applications
therapeutic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR1059602A
Other languages
English (en)
French (fr)
Other versions
FR2967672A1 (fr
Inventor
Alain Pellet
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Aventis France
Original Assignee
Sanofi Aventis France
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis France filed Critical Sanofi Aventis France
Priority to FR1059602A priority Critical patent/FR2967672B1/fr
Priority to EP11796759.6A priority patent/EP2643307B1/fr
Priority to PCT/FR2011/052699 priority patent/WO2012069743A1/fr
Priority to US13/988,868 priority patent/US8993561B2/en
Priority to JP2013539319A priority patent/JP5876885B2/ja
Publication of FR2967672A1 publication Critical patent/FR2967672A1/fr
Application granted granted Critical
Publication of FR2967672B1 publication Critical patent/FR2967672B1/fr
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62—Benzothiazoles
    • C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A61P31/06—Antibacterial agents for tuberculosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
FR1059602A 2010-11-22 2010-11-22 Derives de nitrobenzothiazoles, leur preparation et leurs applications therapeutiques Expired - Fee Related FR2967672B1 (fr)

Priority Applications (5)

Application Number Priority Date Filing Date Title
FR1059602A FR2967672B1 (fr) 2010-11-22 2010-11-22 Derives de nitrobenzothiazoles, leur preparation et leurs applications therapeutiques
EP11796759.6A EP2643307B1 (fr) 2010-11-22 2011-11-18 Derives de nitrobenzothiazoles et leur utilisation pour le traitment de la tubercolose
PCT/FR2011/052699 WO2012069743A1 (fr) 2010-11-22 2011-11-18 Derives de nitrobenzothiazoles et leur utilisation pour le traitment de la tubercolose
US13/988,868 US8993561B2 (en) 2010-11-22 2011-11-18 Nitrobenzothiazole derivatives, preparation thereof and therapeutic applications thereof
JP2013539319A JP5876885B2 (ja) 2010-11-22 2011-11-18 ニトロベンゾチアゾール誘導体および結核治療のためのこれらの使用

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR1059602A FR2967672B1 (fr) 2010-11-22 2010-11-22 Derives de nitrobenzothiazoles, leur preparation et leurs applications therapeutiques

Publications (2)

Publication Number Publication Date
FR2967672A1 FR2967672A1 (fr) 2012-05-25
FR2967672B1 true FR2967672B1 (fr) 2012-12-28

Family

ID=43498537

Family Applications (1)

Application Number Title Priority Date Filing Date
FR1059602A Expired - Fee Related FR2967672B1 (fr) 2010-11-22 2010-11-22 Derives de nitrobenzothiazoles, leur preparation et leurs applications therapeutiques

Country Status (5)

Country Link
US (1) US8993561B2 (enExample)
EP (1) EP2643307B1 (enExample)
JP (1) JP5876885B2 (enExample)
FR (1) FR2967672B1 (enExample)
WO (1) WO2012069743A1 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT2688403T (pt) 2011-03-23 2017-07-13 Trevena Inc Ligandos de recetores opioides e métodos de uso e fabrico dos mesmos
CN103204825B (zh) 2012-01-17 2015-03-04 上海科州药物研发有限公司 作为蛋白激酶抑制剂的苯并噻唑化合物及其制备方法和用途
HK1251472A1 (zh) 2015-12-14 2019-02-01 特维娜有限公司 治療痛覺過敏的方法
CN118660885A (zh) * 2022-01-06 2024-09-17 国家医疗保健研究所 降冰片烯类似物及其作为抗结核药物增效剂的用途

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2013434A1 (en) * 1970-03-20 1971-10-07 Farbenfabriken Bayer Ag, 5090 Lever Kusen Benzothiazole 3-oxides as concrementinhibitors
BE786520A (fr) * 1971-07-23 1973-01-22 Bayer Ag Nouveaux benzothiazoles substitues, leur preparation et leur application comme fongicides et bactericides
BE786521A (fr) 1971-07-23 1973-01-22 Bayer Ag Procede de preparation de 4-chloro-benzothiazoles
RU2227458C2 (ru) 1998-06-18 2004-04-27 Новартис Аг Применение бензазольных соединений в качестве репеллента, композиция их содержащая и способ получения композиции
CA2338328A1 (en) * 1998-07-21 2000-02-03 Thomas Jefferson University Small molecule inhibitors of bcl-2 proteins
JP2000086642A (ja) 1998-09-11 2000-03-28 Kyorin Pharmaceut Co Ltd ベンゾチアゾール誘導体及びその製造法
JP2000178248A (ja) 1998-12-14 2000-06-27 Japan Tobacco Inc 免疫賦活活性を有する化合物
GB0302220D0 (en) * 2003-01-30 2003-03-05 Cyclacel Ltd Use
GB0428173D0 (en) * 2004-12-23 2005-01-26 Astrazeneca Ab Compounds

Also Published As

Publication number Publication date
JP2013542976A (ja) 2013-11-28
US20130245008A1 (en) 2013-09-19
US8993561B2 (en) 2015-03-31
EP2643307B1 (fr) 2014-09-17
WO2012069743A1 (fr) 2012-05-31
JP5876885B2 (ja) 2016-03-02
EP2643307A1 (fr) 2013-10-02
FR2967672A1 (fr) 2012-05-25

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