FR2911874B1 - Derives d'urees de tropane, leur preparation et leur application en therapeutique - Google Patents
Derives d'urees de tropane, leur preparation et leur application en therapeutiqueInfo
- Publication number
- FR2911874B1 FR2911874B1 FR0700507A FR0700507A FR2911874B1 FR 2911874 B1 FR2911874 B1 FR 2911874B1 FR 0700507 A FR0700507 A FR 0700507A FR 0700507 A FR0700507 A FR 0700507A FR 2911874 B1 FR2911874 B1 FR 2911874B1
- Authority
- FR
- France
- Prior art keywords
- urees
- tropane
- derivatives
- preparation
- therapeutic application
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Physical Education & Sports Medicine (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Rheumatology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Immunology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (25)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0700507A FR2911874B1 (fr) | 2007-01-25 | 2007-01-25 | Derives d'urees de tropane, leur preparation et leur application en therapeutique |
TW096122891A TW200811170A (en) | 2006-06-27 | 2007-06-25 | Urea derivatives of tropane, their preparation and their therapeutic application |
PE2007000811A PE20080344A1 (es) | 2006-06-27 | 2007-06-25 | Compuestos 8-azabiciclo[3.2.1]oct-8-il-1,2,3,4-tetrahidroquinolina sustituidos como inhibidores 11b-hsd1 |
DK07803782.7T DK2046791T3 (da) | 2006-06-27 | 2007-06-26 | Ureaderivater af tropan, fremstilling deraf og terepeutisk anvendelse deraf |
ES07803782T ES2342793T3 (es) | 2006-06-27 | 2007-06-26 | Derivados de ureas de tropano, su preparacion y su aplicacion en terapeutica. |
EP07803782A EP2046791B1 (fr) | 2006-06-27 | 2007-06-26 | Dérivés d'urees de tropane, leur préparation et leur application en thérapeutique |
CL2007001885A CL2007001885A1 (es) | 2006-06-27 | 2007-06-26 | Compuestos derivados de urea de tropano, moduladores de la actividad de la 11betahsd1; procedimiento de preparacion; composicion farmaceutica; y uso para el tratamiento de enfermedades tales como obesidad, diabetes, hipertension, aterosclerosis, demencia y osteoporosis. |
PL07803782T PL2046791T3 (pl) | 2006-06-27 | 2007-06-26 | Mocznikowe pochodne tropanu, ich wytwarzanie i ich zastosowanie w lecznictwie |
RU2009102535/04A RU2009102535A (ru) | 2006-06-27 | 2007-06-26 | Производные карбамидов тропана, их получение и их применение в терапии |
KR1020087031631A KR20090021193A (ko) | 2006-06-27 | 2007-06-26 | 트로판의 우레아 유도체, 그의 제법 및 그의 치료 용도 |
PT07803782T PT2046791E (pt) | 2006-06-27 | 2007-06-26 | Derivados de ureias de tropano, sua preparação e sua aplicação em terapêutica |
CA002648769A CA2648769A1 (fr) | 2006-06-27 | 2007-06-26 | Derives d'urees de tropane, leur preparation et leur application en therapeutique |
JP2009517319A JP2009541464A (ja) | 2006-06-27 | 2007-06-26 | トロパンの尿素誘導体、その調製およびその治療用途 |
ARP070102821A AR061642A1 (es) | 2006-06-27 | 2007-06-26 | Derivados de ureas de tropano, su preparacion y su aplicacion en terapeu-tica, procesos de obtencion y composiciones farmaceuticas |
MX2008016492A MX277822B (es) | 2006-06-27 | 2007-06-26 | Derivados de urea de tropano, su preparacion y su aplicacion terapeutica. |
AT07803782T ATE461930T1 (de) | 2006-06-27 | 2007-06-26 | Harnstoffderivate von tropan, ihre herstellung und ihre therapeutische anwendung |
SI200730258T SI2046791T1 (sl) | 2006-06-27 | 2007-06-26 | Sečninski derivati tropana, njihova priprava in njihova terapevtska uporaba |
PCT/FR2007/001070 WO2008000951A2 (fr) | 2006-06-27 | 2007-06-26 | Dérivés d'urees de tropane, leur préparation et leur application en thérapeutique |
AU2007264792A AU2007264792A1 (en) | 2006-06-27 | 2007-06-26 | Urea derivatives of tropane, their preparation and their therapeutic application |
DE602007005487T DE602007005487D1 (de) | 2006-06-27 | 2007-06-26 | Harnstoffderivate von tropan, ihre herstellung und ihre therapeutische anwendung |
UY30447A UY30447A1 (es) | 2006-06-27 | 2007-06-27 | Derivados de ureas de tropano, su preparacion y su aplicacion en terapéutica |
IL195510A IL195510A0 (en) | 2006-06-27 | 2008-11-25 | Urea derivatives of tropane, their preparation and their therapeutic application |
US12/332,547 US7897773B2 (en) | 2006-06-27 | 2008-12-11 | Urea derivatives of tropane, their preparation and their therapeutic application |
CY20101100571T CY1110132T1 (el) | 2006-06-27 | 2010-06-21 | Παραγωγα ουριας τροπανιου, η παρασκευη τους και οι εφαρμογες τους στη θεραπευτικη |
US12/871,403 US20100324084A1 (en) | 2006-06-27 | 2010-08-30 | Urea derivatives of tropane, their preparation and their therapeutic application |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0700507A FR2911874B1 (fr) | 2007-01-25 | 2007-01-25 | Derives d'urees de tropane, leur preparation et leur application en therapeutique |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2911874A1 FR2911874A1 (fr) | 2008-08-01 |
FR2911874B1 true FR2911874B1 (fr) | 2009-03-06 |
Family
ID=38283192
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR0700507A Expired - Fee Related FR2911874B1 (fr) | 2006-06-27 | 2007-01-25 | Derives d'urees de tropane, leur preparation et leur application en therapeutique |
Country Status (1)
Country | Link |
---|---|
FR (1) | FR2911874B1 (fr) |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1263758A2 (fr) * | 2000-03-03 | 2002-12-11 | Ortho-McNeil Pharmaceutical, Inc. | Derives de 3-(diarylmethylene)-8-azabicyclo 3.2.1]octane |
ATE474577T1 (de) * | 2003-03-26 | 2010-08-15 | Merck Sharp & Dohme | Bicyclische piperidin-derivate als melanocortin-4 rezeptor-agonisten |
EP1809626A2 (fr) * | 2004-10-13 | 2007-07-25 | Neurogen Corporation | Composes de 8-azabicyclo[3.2.1]octane a substitution aryle comme ligands du recepteur de l'hormone de concentration de la melanine |
JP5042028B2 (ja) * | 2004-11-05 | 2012-10-03 | セラヴァンス, インコーポレーテッド | キノリノン−カルボキサミド化合物 |
-
2007
- 2007-01-25 FR FR0700507A patent/FR2911874B1/fr not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
FR2911874A1 (fr) | 2008-08-01 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PLFP | Fee payment |
Year of fee payment: 9 |
|
ST | Notification of lapse |
Effective date: 20160930 |