FR2882263B1 - Utilisation d'un derive du pyrazole pour la preparation de medicaments utiles dans la prevention et le traitement des maladies renales - Google Patents

Utilisation d'un derive du pyrazole pour la preparation de medicaments utiles dans la prevention et le traitement des maladies renales

Info

Publication number
FR2882263B1
FR2882263B1 FR0504798A FR0504798A FR2882263B1 FR 2882263 B1 FR2882263 B1 FR 2882263B1 FR 0504798 A FR0504798 A FR 0504798A FR 0504798 A FR0504798 A FR 0504798A FR 2882263 B1 FR2882263 B1 FR 2882263B1
Authority
FR
France
Prior art keywords
prevention
preparation
treatment
renal diseases
pyrazole derivative
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR0504798A
Other languages
English (en)
Other versions
FR2882263A1 (fr
Inventor
Mohammed Bensaid
Jean Marc Herbert
Philip Janiak
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Aventis France
Original Assignee
Sanofi Aventis France
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR0501919A external-priority patent/FR2882262B1/fr
Application filed by Sanofi Aventis France filed Critical Sanofi Aventis France
Priority to FR0504798A priority Critical patent/FR2882263B1/fr
Priority to AU2006217794A priority patent/AU2006217794A1/en
Priority to BRPI0607894-0A priority patent/BRPI0607894A2/pt
Priority to MX2007009995A priority patent/MX2007009995A/es
Priority to EA200701800A priority patent/EA011655B1/ru
Priority to JP2007556630A priority patent/JP2008531526A/ja
Priority to KR1020077019170A priority patent/KR20070104916A/ko
Priority to CA002597802A priority patent/CA2597802A1/fr
Priority to PCT/FR2006/000369 priority patent/WO2006090047A1/fr
Priority to EP06709339A priority patent/EP1855675A1/fr
Priority to ARP060100612A priority patent/AR054003A1/es
Priority to TW095105981A priority patent/TW200640458A/zh
Publication of FR2882263A1 publication Critical patent/FR2882263A1/fr
Publication of FR2882263B1 publication Critical patent/FR2882263B1/fr
Application granted granted Critical
Priority to CR9270A priority patent/CR9270A/es
Priority to TNP2007000291A priority patent/TNSN07291A1/en
Priority to US11/832,861 priority patent/US7622488B2/en
Priority to IL185165A priority patent/IL185165A0/en
Priority to MA30159A priority patent/MA29263B1/fr
Priority to NO20074768A priority patent/NO20074768L/no
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FR0504798A 2005-02-23 2005-05-12 Utilisation d'un derive du pyrazole pour la preparation de medicaments utiles dans la prevention et le traitement des maladies renales Expired - Fee Related FR2882263B1 (fr)

Priority Applications (18)

Application Number Priority Date Filing Date Title
FR0504798A FR2882263B1 (fr) 2005-02-23 2005-05-12 Utilisation d'un derive du pyrazole pour la preparation de medicaments utiles dans la prevention et le traitement des maladies renales
AU2006217794A AU2006217794A1 (en) 2005-02-23 2006-02-17 Use of a pyrazole derivative for preparing medicines useful for preventing or treating renal diseases
BRPI0607894-0A BRPI0607894A2 (pt) 2005-02-23 2006-02-17 utilização de um derivado de pirazol para a preparação de medicamentos úteis na prevenção e no tratamento das doenças renais
MX2007009995A MX2007009995A (es) 2005-02-23 2006-02-17 Utilizacion de un derivado de pirazol para la preparacion de medicamentos utiles en la prevencion y el tratamiento de las enfermedades renales.
EA200701800A EA011655B1 (ru) 2005-02-23 2006-02-17 Применение производного пиразола для получения лекарственных средств, подходящих для профилактики и лечения заболеваний почек
JP2007556630A JP2008531526A (ja) 2005-02-23 2006-02-17 腎臓病の予防または治療に有用な薬物を調製するためのピラゾール誘導体の使用
KR1020077019170A KR20070104916A (ko) 2005-02-23 2006-02-17 신장병의 예방 또는 치료에 유용한 의약의 제조를 위한피라졸 유도체의 용도
CA002597802A CA2597802A1 (fr) 2005-02-23 2006-02-17 Utilisation d'un derive du pyrazole pour la preparation de medicaments utiles dans la prevention et le traitement des maladies renales
PCT/FR2006/000369 WO2006090047A1 (fr) 2005-02-23 2006-02-17 Utilisation d'un derive du pyrazole pour la preparation de medicaments utiles dans la prevention et le traitement des maladies renales
EP06709339A EP1855675A1 (fr) 2005-02-23 2006-02-17 Utilisation d'un derive du pyrazole pour la preparation de medicaments utiles dans la prevention et le traitement des maladies renales
ARP060100612A AR054003A1 (es) 2005-02-23 2006-02-21 Utilizacion de un derivado de pirazol para la preparacion de medicamentos utiles en la prevencion y el tratamiento de las enfermedades renales
TW095105981A TW200640458A (en) 2005-02-23 2006-02-22 Use of a pyrazole derivative for preparing medicinal products that are of use in the prevention and treatment of kidney diseases
CR9270A CR9270A (es) 2005-02-23 2007-07-20 Utilizacion de un derivado de pirazol para la preparacion de medicamentos utiles en la prevencion y el tratamiento de enfermedades renales
TNP2007000291A TNSN07291A1 (en) 2005-02-23 2007-07-24 Use of a pyrazole derivative for preparing medicines useful for preventing or treating renal diseases
US11/832,861 US7622488B2 (en) 2005-02-23 2007-08-02 Use of a pyrazole derivative for preparing medicines useful for treating renal diseases
IL185165A IL185165A0 (en) 2005-02-23 2007-08-09 Use of a pyrazole derivative for preparing medicines useful for preventing or treating renal diseases
MA30159A MA29263B1 (fr) 2005-02-23 2007-08-23 Utilisation d'un derive du pyrazole pour la preparation de medicaments utiles dans la prevention et le traitement des maladies renales
NO20074768A NO20074768L (no) 2005-02-23 2007-09-18 Anvendelse av pyrazolderivater for fremstilling av medisiner nyttige for a forebygge eller behandle nyresykdommer

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0501919A FR2882262B1 (fr) 2005-02-23 2005-02-23 Utilisation d'un derive du pyrazole pour la preparation de medicaments utiles dans la prevention et le traitement des maladies renales
FR0504798A FR2882263B1 (fr) 2005-02-23 2005-05-12 Utilisation d'un derive du pyrazole pour la preparation de medicaments utiles dans la prevention et le traitement des maladies renales

Publications (2)

Publication Number Publication Date
FR2882263A1 FR2882263A1 (fr) 2006-08-25
FR2882263B1 true FR2882263B1 (fr) 2007-04-06

Family

ID=36603585

Family Applications (1)

Application Number Title Priority Date Filing Date
FR0504798A Expired - Fee Related FR2882263B1 (fr) 2005-02-23 2005-05-12 Utilisation d'un derive du pyrazole pour la preparation de medicaments utiles dans la prevention et le traitement des maladies renales

Country Status (18)

Country Link
US (1) US7622488B2 (fr)
EP (1) EP1855675A1 (fr)
JP (1) JP2008531526A (fr)
KR (1) KR20070104916A (fr)
AR (1) AR054003A1 (fr)
AU (1) AU2006217794A1 (fr)
BR (1) BRPI0607894A2 (fr)
CA (1) CA2597802A1 (fr)
CR (1) CR9270A (fr)
EA (1) EA011655B1 (fr)
FR (1) FR2882263B1 (fr)
IL (1) IL185165A0 (fr)
MA (1) MA29263B1 (fr)
MX (1) MX2007009995A (fr)
NO (1) NO20074768L (fr)
TN (1) TNSN07291A1 (fr)
TW (1) TW200640458A (fr)
WO (1) WO2006090047A1 (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2010079241A1 (fr) 2009-01-12 2010-07-15 Fundacion Hospital Nacional De Paraplejicos Para La Investigacion Y La Integracion Utilisation d'antagonistes et/ou d'agonistes inverses des récepteurs cb1 pour la préparation de médicaments qui augmentent l'excitabilité des motoneurones
FR2958850B1 (fr) * 2010-04-14 2012-07-06 Centre Nat Rech Scient Medicaments pour la prevention ou le traitement des addictions aux drogues

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2692575B1 (fr) * 1992-06-23 1995-06-30 Sanofi Elf Nouveaux derives du pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.
FR2713225B1 (fr) * 1993-12-02 1996-03-01 Sanofi Sa N-pipéridino-3-pyrazolecarboxamide substitué.
FR2789079B3 (fr) 1999-02-01 2001-03-02 Sanofi Synthelabo Derive d'acide pyrazolecarboxylique, sa preparation, les compositions pharmaceutiques en contenant
US20040122033A1 (en) * 2002-12-10 2004-06-24 Nargund Ravi P. Combination therapy for the treatment of obesity
US20040214804A1 (en) * 2003-04-25 2004-10-28 Pharmacia Corporation Combination of an aldosterone receptor antagonist and an anti-obesity agent
AR051446A1 (es) * 2004-09-23 2007-01-17 Bristol Myers Squibb Co Glucosidos de c-arilo como inhibidores selectivos de transportadores de glucosa (sglt2)

Also Published As

Publication number Publication date
NO20074768L (no) 2007-11-23
CR9270A (es) 2007-10-01
MA29263B1 (fr) 2008-02-01
EA200701800A1 (ru) 2008-02-28
TNSN07291A1 (en) 2008-12-31
KR20070104916A (ko) 2007-10-29
TW200640458A (en) 2006-12-01
WO2006090047A1 (fr) 2006-08-31
US20080015228A1 (en) 2008-01-17
IL185165A0 (en) 2008-06-05
EA011655B1 (ru) 2009-04-28
FR2882263A1 (fr) 2006-08-25
BRPI0607894A2 (pt) 2009-10-20
MX2007009995A (es) 2007-10-10
AU2006217794A1 (en) 2006-08-31
EP1855675A1 (fr) 2007-11-21
JP2008531526A (ja) 2008-08-14
CA2597802A1 (fr) 2006-08-31
AR054003A1 (es) 2007-05-30
US7622488B2 (en) 2009-11-24

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Legal Events

Date Code Title Description
ST Notification of lapse

Effective date: 20110131