FR2792634B1 - Derives de 2-alcoxy-cyclobutene-3,4-dione leur preparation et leur application en therapeutique - Google Patents

Derives de 2-alcoxy-cyclobutene-3,4-dione leur preparation et leur application en therapeutique

Info

Publication number
FR2792634B1
FR2792634B1 FR9904945A FR9904945A FR2792634B1 FR 2792634 B1 FR2792634 B1 FR 2792634B1 FR 9904945 A FR9904945 A FR 9904945A FR 9904945 A FR9904945 A FR 9904945A FR 2792634 B1 FR2792634 B1 FR 2792634B1
Authority
FR
France
Prior art keywords
alcoxy
cyclobutene
preparation
therapeutic application
dione derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR9904945A
Other languages
English (en)
Other versions
FR2792634A1 (fr
Inventor
Philippe R Bovy
Claudie Gautier
Christophe Philippo
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Synthelabo SA
Original Assignee
Synthelabo SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo SA filed Critical Synthelabo SA
Priority to FR9904945A priority Critical patent/FR2792634B1/fr
Priority to PCT/FR2000/000926 priority patent/WO2000063160A1/fr
Priority to AU39718/00A priority patent/AU3971800A/en
Priority to CO00028248A priority patent/CO5160305A1/es
Priority to UY26110A priority patent/UY26110A1/es
Priority to ARP000101828A priority patent/AR023548A1/es
Publication of FR2792634A1 publication Critical patent/FR2792634A1/fr
Application granted granted Critical
Publication of FR2792634B1 publication Critical patent/FR2792634B1/fr
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C237/00Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
    • C07C237/24Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring of the carbon skeleton
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/08Drugs for disorders of the urinary system of the prostate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00Systems containing only non-condensed rings
    • C07C2601/02Systems containing only non-condensed rings with a three-membered ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00Systems containing only non-condensed rings
    • C07C2601/04Systems containing only non-condensed rings with a four-membered ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00Systems containing only non-condensed rings
    • C07C2601/12Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14The ring being saturated

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Vascular Medicine (AREA)
  • Emergency Medicine (AREA)
  • Reproductive Health (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FR9904945A 1999-04-20 1999-04-20 Derives de 2-alcoxy-cyclobutene-3,4-dione leur preparation et leur application en therapeutique Expired - Fee Related FR2792634B1 (fr)

Priority Applications (6)

Application Number Priority Date Filing Date Title
FR9904945A FR2792634B1 (fr) 1999-04-20 1999-04-20 Derives de 2-alcoxy-cyclobutene-3,4-dione leur preparation et leur application en therapeutique
PCT/FR2000/000926 WO2000063160A1 (fr) 1999-04-20 2000-04-11 Derives de 2-alcoxy-cyclobutane-3,4-dione leur preparation et leur application en therapeutique
AU39718/00A AU3971800A (en) 1999-04-20 2000-04-11 2-alkoxy-cyclobutene-3,4-dione derivatives, preparation and therapeutic use thereof
CO00028248A CO5160305A1 (es) 1999-04-20 2000-04-17 Derivados de 2-alcoxi-ciclobuten-3,4-diona su preparacion y su aplicacion en terapeutica
UY26110A UY26110A1 (es) 1999-04-20 2000-04-18 Derivados de 2-alcoxi-ciclobuten-3,4-diona, su preparación y su aplicación en terapéutica
ARP000101828A AR023548A1 (es) 1999-04-20 2000-04-19 Derivados de 2-alcoxi-ciclobuten-3,4-diona, su preparacion y su aplicacion en terapeutica

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9904945A FR2792634B1 (fr) 1999-04-20 1999-04-20 Derives de 2-alcoxy-cyclobutene-3,4-dione leur preparation et leur application en therapeutique

Publications (2)

Publication Number Publication Date
FR2792634A1 FR2792634A1 (fr) 2000-10-27
FR2792634B1 true FR2792634B1 (fr) 2001-06-01

Family

ID=9544620

Family Applications (1)

Application Number Title Priority Date Filing Date
FR9904945A Expired - Fee Related FR2792634B1 (fr) 1999-04-20 1999-04-20 Derives de 2-alcoxy-cyclobutene-3,4-dione leur preparation et leur application en therapeutique

Country Status (6)

Country Link
AR (1) AR023548A1 (fr)
AU (1) AU3971800A (fr)
CO (1) CO5160305A1 (fr)
FR (1) FR2792634B1 (fr)
UY (1) UY26110A1 (fr)
WO (1) WO2000063160A1 (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6495576B2 (en) 2001-02-07 2002-12-17 Abbott Laboratories Aminal diones as potassium channel openers
DE10135815A1 (de) * 2001-07-23 2003-02-06 Bayer Ag Verwendung von 2-Alkoxyphenyl-substituierten Imidazotriazinonen
AU2002361417A1 (en) * 2001-12-17 2003-06-30 Altana Pharma Ag Use of selective PDE5 inhibitors for treating partial and global respiratory failure
FR2842271B1 (fr) 2002-07-15 2004-09-10 Eurocopter France Boite de transmissiion de puissance basculante a transfert de charge par le carter

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9311282D0 (en) * 1993-06-01 1993-07-21 Rhone Poulenc Rorer Ltd New compositions of matter

Also Published As

Publication number Publication date
AU3971800A (en) 2000-11-02
CO5160305A1 (es) 2002-05-30
UY26110A1 (es) 2000-12-29
WO2000063160A1 (fr) 2000-10-26
AR023548A1 (es) 2002-09-04
FR2792634A1 (fr) 2000-10-27

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Legal Events

Date Code Title Description
TP Transmission of property
ST Notification of lapse