FR2578544A1 - Antihypertension spirocyclic compounds - Google Patents

Antihypertension spirocyclic compounds Download PDF

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Publication number
FR2578544A1
FR2578544A1 FR8503531A FR8503531A FR2578544A1 FR 2578544 A1 FR2578544 A1 FR 2578544A1 FR 8503531 A FR8503531 A FR 8503531A FR 8503531 A FR8503531 A FR 8503531A FR 2578544 A1 FR2578544 A1 FR 2578544A1
Authority
FR
France
Prior art keywords
salts
chloro
spiro
dihydro
dioxide
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR8503531A
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English (en)
French (fr)
Other versions
FR2578544B1 (hu
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
USV Pharmaceutical Corp
Original Assignee
USV Pharmaceutical Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by USV Pharmaceutical Corp filed Critical USV Pharmaceutical Corp
Priority to FR8503531A priority Critical patent/FR2578544A1/fr
Publication of FR2578544A1 publication Critical patent/FR2578544A1/fr
Application granted granted Critical
Publication of FR2578544B1 publication Critical patent/FR2578544B1/fr
Granted legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/022—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
    • C07K5/0222—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2 with the first amino acid being heterocyclic, e.g. Pro, Trp
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
FR8503531A 1985-03-11 1985-03-11 Antihypertension spirocyclic compounds Granted FR2578544A1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FR8503531A FR2578544A1 (en) 1985-03-11 1985-03-11 Antihypertension spirocyclic compounds

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8503531A FR2578544A1 (en) 1985-03-11 1985-03-11 Antihypertension spirocyclic compounds

Publications (2)

Publication Number Publication Date
FR2578544A1 true FR2578544A1 (en) 1986-09-12
FR2578544B1 FR2578544B1 (hu) 1988-07-01

Family

ID=9317059

Family Applications (1)

Application Number Title Priority Date Filing Date
FR8503531A Granted FR2578544A1 (en) 1985-03-11 1985-03-11 Antihypertension spirocyclic compounds

Country Status (1)

Country Link
FR (1) FR2578544A1 (hu)

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2487341A1 (fr) * 1980-07-24 1982-01-29 Squibb & Sons Inc Tripeptides inhibiteurs de l'enzyme de transformation de l'angiotensine
GB2123834A (en) * 1982-07-19 1984-02-08 Squibb & Sons Inc Substituted peptide compounds
EP0121830A2 (en) * 1983-03-16 1984-10-17 Usv Pharmaceutical Corporation Substituted dipeptides as antihypertensives
EP0132304A2 (en) * 1983-07-21 1985-01-30 E.R. Squibb & Sons, Inc. Hydroxy substituted peptide compounds

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2487341A1 (fr) * 1980-07-24 1982-01-29 Squibb & Sons Inc Tripeptides inhibiteurs de l'enzyme de transformation de l'angiotensine
GB2123834A (en) * 1982-07-19 1984-02-08 Squibb & Sons Inc Substituted peptide compounds
EP0121830A2 (en) * 1983-03-16 1984-10-17 Usv Pharmaceutical Corporation Substituted dipeptides as antihypertensives
EP0132304A2 (en) * 1983-07-21 1985-01-30 E.R. Squibb & Sons, Inc. Hydroxy substituted peptide compounds

Also Published As

Publication number Publication date
FR2578544B1 (hu) 1988-07-01

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