FR2465735A1 - Composes intermediaires pour la preparation de derives de la morphine, et leur procede de preparation - Google Patents

Composes intermediaires pour la preparation de derives de la morphine, et leur procede de preparation Download PDF

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Publication number
FR2465735A1
FR2465735A1 FR8017530A FR8017530A FR2465735A1 FR 2465735 A1 FR2465735 A1 FR 2465735A1 FR 8017530 A FR8017530 A FR 8017530A FR 8017530 A FR8017530 A FR 8017530A FR 2465735 A1 FR2465735 A1 FR 2465735A1
Authority
FR
France
Prior art keywords
boron
amide
preparation
compounds
nalbuphine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
FR8017530A
Other languages
English (en)
French (fr)
Inventor
Dennis J Malfer
Donald F Loncrini
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Mallinckrodt Inc
Original Assignee
Mallinckrodt Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mallinckrodt Inc filed Critical Mallinckrodt Inc
Publication of FR2465735A1 publication Critical patent/FR2465735A1/fr
Withdrawn legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D489/00Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula:
    • C07D489/06Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: with a hetero atom directly attached in position 14
    • C07D489/08Oxygen atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
FR8017530A 1979-08-09 1980-08-08 Composes intermediaires pour la preparation de derives de la morphine, et leur procede de preparation Withdrawn FR2465735A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US6527579A 1979-08-09 1979-08-09

Publications (1)

Publication Number Publication Date
FR2465735A1 true FR2465735A1 (fr) 1981-03-27

Family

ID=22061564

Family Applications (1)

Application Number Title Priority Date Filing Date
FR8017530A Withdrawn FR2465735A1 (fr) 1979-08-09 1980-08-08 Composes intermediaires pour la preparation de derives de la morphine, et leur procede de preparation

Country Status (16)

Country Link
JP (1) JPS56501010A (online.php)
AU (1) AU6116580A (online.php)
BE (1) BE884671A (online.php)
DD (1) DD154541A5 (online.php)
DK (1) DK151781A (online.php)
ES (1) ES494122A0 (online.php)
FI (1) FI802479A7 (online.php)
FR (1) FR2465735A1 (online.php)
GB (1) GB2066256A (online.php)
IL (1) IL60783A0 (online.php)
IT (1) IT8068267A0 (online.php)
NL (1) NL8020319A (online.php)
NO (1) NO802139L (online.php)
PL (1) PL226162A1 (online.php)
SE (1) SE8102214L (online.php)
WO (1) WO1981000409A1 (online.php)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4795813A (en) * 1981-08-17 1989-01-03 The Florida Board Of Regents On Behalf Of The Florida State University Synthesis of derivatives of codeine and other 3-O-alkylmorphines
US5668285A (en) * 1986-10-31 1997-09-16 The United States Of America As Represented By The Department Of Health And Human Services Total synthesis of northebaine, normophine, noroxymorphone enantiomers and derivatives via N-Nor intermediates
CA2067200C (en) * 1989-10-16 1998-06-30 Kenner C. Rice Total synthesis of northebaine, normorphine, noroxymorphone enantiomers and derivatives via n-nor intermediates

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3332950A (en) * 1963-03-23 1967-07-25 Endo Lab 14-hydroxydihydronormorphinone derivatives
NL7106612A (en) * 1971-05-13 1972-11-15 N-cycloalkylalkyl-14-hydroxy-dihydronormorphines - - by o-demethylation of 14-methoxy cpds
US4161597A (en) * 1976-12-20 1979-07-17 Research Corporation N-alkyl-14-hydroxymorphinans and derivatives

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA913077A (en) * 1972-10-24 J. Pachter Irwin Process of preparing n-substituted 14-hydroxydihydronormorphines
US3249616A (en) * 1966-05-03 Ix-dfflydroxy-g-oxo-n-phenethylmor- phinan (cis) and production thereof
US2772270A (en) * 1954-10-21 1956-11-27 M J Lewenstein 14-hydroxymorphinone and 8, 14-dihydroxydihydromorphinone
US2806033A (en) * 1955-08-03 1957-09-10 Lewenstein Morphine derivative
BE638369A (online.php) * 1962-10-10
US3775414A (en) * 1972-05-10 1973-11-27 Bristol Myers Co Process for the preparation of 14-hydroxymorphinan derivatives

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3332950A (en) * 1963-03-23 1967-07-25 Endo Lab 14-hydroxydihydronormorphinone derivatives
NL7106612A (en) * 1971-05-13 1972-11-15 N-cycloalkylalkyl-14-hydroxy-dihydronormorphines - - by o-demethylation of 14-methoxy cpds
US4161597A (en) * 1976-12-20 1979-07-17 Research Corporation N-alkyl-14-hydroxymorphinans and derivatives

Also Published As

Publication number Publication date
JPS56501010A (online.php) 1981-07-23
NL8020319A (nl) 1981-07-01
GB2066256A (en) 1981-07-08
BE884671A (fr) 1980-12-01
ES8104296A1 (es) 1981-04-16
WO1981000409A1 (en) 1981-02-19
PL226162A1 (online.php) 1981-04-24
AU6116580A (en) 1981-02-12
ES494122A0 (es) 1981-04-16
IT8068267A0 (it) 1980-08-07
DD154541A5 (de) 1982-03-31
DK151781A (da) 1981-04-03
SE8102214L (sv) 1981-04-07
FI802479A7 (fi) 1981-01-01
IL60783A0 (en) 1980-10-26
NO802139L (no) 1981-02-10

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