FR2450M - Nouvelles pyrimidines. - Google Patents
Nouvelles pyrimidines.Info
- Publication number
- FR2450M FR2450M FR928687A FR928687A FR2450M FR 2450 M FR2450 M FR 2450M FR 928687 A FR928687 A FR 928687A FR 928687 A FR928687 A FR 928687A FR 2450 M FR2450 M FR 2450M
- Authority
- FR
- France
- Prior art keywords
- new pyrimidines
- pyrimidines
- new
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 150000003230 pyrimidines Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DET21813A DE1197466B (de) | 1962-03-22 | 1962-03-22 | Verfahren zur Herstellung von neuen 5, 6, 7, 8-Tetrahydropyrido-[4, 3-d]pyrimidinen |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| FR2450M true FR2450M (fr) | 1964-04-06 |
Family
ID=7550280
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FR928687A Expired FR2450M (fr) | 1962-03-22 | 1963-03-20 | Nouvelles pyrimidines. |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US3248395A (fr) |
| CH (2) | CH462186A (fr) |
| DE (1) | DE1197466B (fr) |
| FR (1) | FR2450M (fr) |
| GB (1) | GB1033384A (fr) |
Cited By (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2005014558A1 (fr) * | 2003-08-05 | 2005-02-17 | Vertex Pharmaceuticals Incorporated | Composes de pyramidine condenses utilises comme inhibiteurs de canaux ioniques potentiel-dependants |
| US8163763B2 (en) | 2008-07-31 | 2012-04-24 | Genentech, Inc. | Pyrimidine compounds, compositions and methods of use |
| US8288381B2 (en) | 2009-11-12 | 2012-10-16 | Genentech, Inc. | N-9 substituted purine compounds, compositions and methods of use |
| US8828990B2 (en) | 2009-11-12 | 2014-09-09 | Genentech, Inc. | N-7 substituted purine and pyrazolopyrimine compounds, compositions and methods of use |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3725405A (en) * | 1970-06-18 | 1973-04-03 | American Home Prod | 2,4,7-TRISUBSTITUTED-{8 PYRIDO 2,3-d{9 PYRIMIDINE-6-CARBOXAMIDES |
| US3939268A (en) * | 1971-04-10 | 1976-02-17 | Boehringer Ingelheim Gmbh | 2,4-Diamino substituted pyridol(3,2-d)pyrimidine as antithrombotic agents |
| JPS5130077B2 (fr) * | 1971-12-28 | 1976-08-30 | ||
| US4085102A (en) * | 1974-11-25 | 1978-04-18 | E. R. Squibb & Sons, Inc. | 2-Amino-8-arylideno-3,4,5,6,7,8-hexahydro-4-arlypyrido[4,3-d]pyrimidines |
| US5137890A (en) * | 1990-02-14 | 1992-08-11 | Ortho Pharmaceutical Corporation | 4-phenyl tetrahydropyrido(4,3-d)pyrimidines |
| US5059602A (en) * | 1990-08-27 | 1991-10-22 | Hoechst-Roussel Pharmaceuticals Inc. | 4-substituted dihydropyrido(4,3-d)pyrimidines as analgesics and topical antiinflammatory agents for the treatment of skin disorders |
| US5212310A (en) * | 1991-12-19 | 1993-05-18 | Neurogen Corporation | Certain aryl fused imidazopyrimidines; a new class of GABA brain receptor ligands |
| EP1679668B1 (fr) * | 1996-09-04 | 2010-01-27 | Intertrust Technologies Corp. | Systèmes, procédés et techniques de support d'infrastructure sécurisée pour le commerce électronique sécurisé, transactions électroniques, contrôle et automatisation du processus de commerce, informatique distribuée et gestion des droits |
| WO2002088079A2 (fr) * | 2001-05-01 | 2002-11-07 | Bristol-Myers Squibb Company | Inhibiteurs doubles de pde 7 et pde 4 |
| US7105667B2 (en) * | 2001-05-01 | 2006-09-12 | Bristol-Myers Squibb Co. | Fused heterocyclic compounds and use thereof |
| AU2003242252A1 (en) * | 2002-06-07 | 2003-12-22 | Kyowa Hakko Kogyo Co., Ltd. | Bicyclic pyrimidine derivatives |
| MXPA06003150A (es) * | 2003-09-17 | 2006-08-31 | Johnson & Johnson | Compuestos heterociclicos fusionados. |
| CA2606760C (fr) * | 2005-05-04 | 2014-12-23 | Renovis, Inc. | Composes de tetrahydronaphthyridine et de tetrahydropyrido[4,3-d]pyrimidine et compositions de ceux-ci utiles dans lediraitement des conditions associees aux troubles et dysfonctions neurologiques et inflammatoires |
| US7598255B2 (en) * | 2005-08-04 | 2009-10-06 | Janssen Pharmaceutica Nv | Pyrimidine compounds as serotonin receptor modulators |
| US8071766B2 (en) | 2008-02-01 | 2011-12-06 | Takeda Pharmaceutical Company Limited | HSP90 inhibitors |
| WO2010120991A1 (fr) * | 2009-04-17 | 2010-10-21 | Wyeth Llc | Composés de 5,6,7,8-tétrahydropyrido[4,3-d]pyrimidine, leur utilisation en tant qu'inhibiteurs de kinase mtor, pi3, et hsmg-1, et leurs synthèses |
| CA2766151A1 (fr) * | 2009-06-24 | 2010-12-29 | Genentech, Inc. | Composes pyrimidine fusionnes a oxo-heterocycles, compositions et procedes d'utilisation |
| WO2011022213A1 (fr) | 2009-08-17 | 2011-02-24 | Merck Sharp & Dohme Corp. | Inhibiteurs de pde10 damino-tétrahydro-pyridopyrimidine |
| UA112517C2 (uk) | 2010-07-06 | 2016-09-26 | Новартіс Аг | Тетрагідропіридопіримідинові похідні |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2697710A (en) * | 1953-01-02 | 1954-12-21 | Burroughs Wellcome Co | Pyrido (2,3-d) pyrimidines and method of preparing same |
| US2926166A (en) * | 1954-01-04 | 1960-02-23 | Burroughs Wellcome Co | Pyrido (2, 3-d) pyrimidine compounds and method of making |
| US2802826A (en) * | 1955-07-13 | 1957-08-13 | Hoffmann La Roche | Octahydro-pyrido [4, 3-d] pyrimidine compounds |
| US2890152A (en) * | 1956-11-29 | 1959-06-09 | Schering Corp | Topical anti-inflammatory compositions |
| US2994640A (en) * | 1957-02-22 | 1961-08-01 | Byk Gulden Lomberg Chem Fab | Anti-inflammatory therapy with purine molecular compounds |
| DE1110649B (de) * | 1957-11-22 | 1961-07-13 | Ciba Geigy | Verfahren zur Herstellung von 1-Isopropyl-pyrazolo[3, 4-d]pyrimidinen |
-
1962
- 1962-03-22 DE DET21813A patent/DE1197466B/de active Pending
-
1963
- 1963-03-11 CH CH1780166A patent/CH462186A/de unknown
- 1963-03-11 CH CH302963A patent/CH437327A/de unknown
- 1963-03-14 US US265059A patent/US3248395A/en not_active Expired - Lifetime
- 1963-03-18 GB GB10641/63A patent/GB1033384A/en not_active Expired
- 1963-03-20 FR FR928687A patent/FR2450M/fr not_active Expired
Cited By (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2005014558A1 (fr) * | 2003-08-05 | 2005-02-17 | Vertex Pharmaceuticals Incorporated | Composes de pyramidine condenses utilises comme inhibiteurs de canaux ioniques potentiel-dependants |
| US7968545B2 (en) | 2003-08-05 | 2011-06-28 | Vertex Pharmaceuticals Inc. | Compositions useful as inhibitors of voltage-gated ion channels |
| JP2011207914A (ja) * | 2003-08-05 | 2011-10-20 | Vertex Pharmaceuticals Inc | 電位依存型イオンチャネルの阻害剤としての縮合ピリミジン化合物 |
| JP4808156B2 (ja) * | 2003-08-05 | 2011-11-02 | バーテックス ファーマシューティカルズ インコーポレイテッド | 電位依存型イオンチャネルの阻害剤としての縮合ピリミジン化合物 |
| US8163763B2 (en) | 2008-07-31 | 2012-04-24 | Genentech, Inc. | Pyrimidine compounds, compositions and methods of use |
| US8288381B2 (en) | 2009-11-12 | 2012-10-16 | Genentech, Inc. | N-9 substituted purine compounds, compositions and methods of use |
| US8828990B2 (en) | 2009-11-12 | 2014-09-09 | Genentech, Inc. | N-7 substituted purine and pyrazolopyrimine compounds, compositions and methods of use |
Also Published As
| Publication number | Publication date |
|---|---|
| CH462186A (de) | 1968-09-15 |
| US3248395A (en) | 1966-04-26 |
| CH437327A (de) | 1967-06-15 |
| GB1033384A (en) | 1966-06-22 |
| DE1197466B (de) | 1965-07-29 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| FR2973M (fr) | Alpha-aminocétone. | |
| FR2450M (fr) | Nouvelles pyrimidines. | |
| FR3846M (fr) | Nouvelles 4-amino-pipéridines. | |
| FR2770M (fr) | Nouvelles dihalogéno-amino-benzylamines. | |
| FR3239M (fr) | Nouvelles amines substituées. | |
| DK105974C (da) | Lastpallemagasin. | |
| DK112125B (da) | Falstagsten. | |
| DK106882C (da) | Tagafdækning. | |
| NL143659B (nl) | Fluidum-en-afsluiting. | |
| FR3110M (fr) | Nouvelles benzamides. | |
| FR3046M (fr) | Nouvelles phényléthanolamines. | |
| FR2592M (fr) | Phénylbicyclononanes substitués. | |
| FR3546M (fr) | Azabenzocycloalcane-n-carboxamidines. | |
| OA01221A (fr) | Polythioformaldéhydes. | |
| FR3088M (fr) | 2-oxo-tétrahydroquinoléines substituées. | |
| FR3325M (fr) | Nouvelles 2-alcoyl-4-pyridine-aldéhyde-thiosemicarbazones. | |
| BE642025A (fr) | Nouvelles indolylalcoylguanidines. | |
| DK103099C (da) | Plov. | |
| FR2894M (fr) | Phénylalcanolamine. | |
| FR2503M (fr) | Nouvelles phénylhétéroalcoylamines. | |
| BE617318A (nl) | Bouwwerk. | |
| FR2953M (fr) | Nouvelles pénicillines. | |
| BE605579A (fr) | Nouvelles sulfonylurées. | |
| GR23071B (el) | Ειδικη κεραμος. | |
| FR2792M (fr) | Nouvelles tétrahydro-dibenzazocines substituées. |