FR2447719A1 - PROCESS FOR THE PREPARATION OF SUPPOSITORIES CONTAINING A SULFAMETHOXAZOLE / TRIMETHOPRIM COMPLEX AND NOVEL PRODUCTS THUS OBTAINED - Google Patents
PROCESS FOR THE PREPARATION OF SUPPOSITORIES CONTAINING A SULFAMETHOXAZOLE / TRIMETHOPRIM COMPLEX AND NOVEL PRODUCTS THUS OBTAINEDInfo
- Publication number
- FR2447719A1 FR2447719A1 FR8001854A FR8001854A FR2447719A1 FR 2447719 A1 FR2447719 A1 FR 2447719A1 FR 8001854 A FR8001854 A FR 8001854A FR 8001854 A FR8001854 A FR 8001854A FR 2447719 A1 FR2447719 A1 FR 2447719A1
- Authority
- FR
- France
- Prior art keywords
- sulfamethoxazole
- complex
- preparation
- novel products
- suppositories containing
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/02—Suppositories; Bougies; Bases therefor; Ovules
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/63—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide
- A61K31/635—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide having a heterocyclic ring, e.g. sulfadiazine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
- Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10S424/00—Drug, bio-affecting and body treating compositions
- Y10S424/15—Suppositories
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
DES SUPPOSITOIRES A ACTION BACTERICIDE CONTIENNENT UN COMPLEXE 11 DE SULFAMETHOXAZOLE ET DE TRIMETHOPRIM, DISPERSE DANS UN SUPPORT PHARMACEUTIQUEMENT ACCEPTABLE; ILS PEUVENT CONTENIR UNE QUANTITE SUPPLEMENTAIRE DE SULFAMETHOXAZOLE, EN PLUS DU COMPOSANT SULFAMETHOXAZOLE DANS LE COMPLEXE, ET, PAR RAPPORT AUX PRODUITS RESULTANT D'UN SIMPLE MELANGE, CES SUPPOSITOIRES PRESENTENT DE MEILLEURES PROPRIETES PHARMACOCINETIQUES.SUPPOSITORIES WITH BACTERICIDAL ACTION CONTAIN A COMPLEX 11 OF SULFAMETHOXAZOLE AND TRIMETHOPRIM, DISPERSE IN A PHARMACEUTICALLY ACCEPTABLE MEDIUM; THEY MAY CONTAIN AN ADDITIONAL QUANTITY OF SULFAMETHOXAZOLE, IN ADDITION TO THE SULFAMETHOXAZOLE COMPONENT IN THE COMPLEX, AND, IN RELATION TO PRODUCTS RESULTING FROM A SIMPLE MIXTURE, THESE SUPPOSITORIES HAVE BETTER PHARMACOKINETIC PROPERTIES.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP999279A JPS55102517A (en) | 1979-01-30 | 1979-01-30 | Preparation of sulfamethoxazole-trimethoprim complex for administration via body cavity |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2447719A1 true FR2447719A1 (en) | 1980-08-29 |
FR2447719B1 FR2447719B1 (en) | 1984-02-24 |
Family
ID=11735349
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR8001854A Granted FR2447719A1 (en) | 1979-01-30 | 1980-01-29 | PROCESS FOR THE PREPARATION OF SUPPOSITORIES CONTAINING A SULFAMETHOXAZOLE / TRIMETHOPRIM COMPLEX AND NOVEL PRODUCTS THUS OBTAINED |
Country Status (13)
Country | Link |
---|---|
US (1) | US4461765A (en) |
JP (1) | JPS55102517A (en) |
AR (1) | AR221525A1 (en) |
CA (1) | CA1136986A (en) |
CH (1) | CH641958A5 (en) |
DE (1) | DE3003147A1 (en) |
ES (1) | ES488367A0 (en) |
FR (1) | FR2447719A1 (en) |
GB (1) | GB2041749B (en) |
IT (1) | IT1133051B (en) |
MX (1) | MX5865E (en) |
NL (1) | NL8000515A (en) |
SE (1) | SE8000286L (en) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS57109713A (en) * | 1980-12-26 | 1982-07-08 | Shionogi & Co Ltd | Pharmaceutical preparation of combined agent of sulfamethoxazole and trimethoprim for medication through celom |
HU197670B (en) * | 1986-02-28 | 1989-05-29 | Egyt Gyogyszervegyeszeti Gyar | Process for producing composition comprising 2,4-diamino-5-(3,4-dimethoxybenzyl)-pyrimidine or pharmaceutically suitable acid addition salt thereof as active ingredient |
HU199683B (en) * | 1987-07-22 | 1990-03-28 | Egyt Gyogyszervegyeszeti Gyar | Process for producing pharmaceutical compositions analgesic, antiphlogistic, antipyretic, antianginic and/or antioxidative activity |
Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2415660A1 (en) * | 1973-04-19 | 1974-11-14 | Paolo Chiesi | SUPPOSITORIES CONTAINING A TRIMETHOPRIM-SULFAMETHOXAZOLE COMBINATION AND PROCESS FOR THEIR PRODUCTION |
FR2361103A1 (en) * | 1976-07-15 | 1978-03-10 | Basf Ag | SULFONAMIDE-TRIMETHOPRIME SOLUTIONS |
JPS54101415A (en) * | 1978-01-27 | 1979-08-10 | Gea As | Stable suspension containing sulfamethoxal and trimetoprim and production thereof |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3197369A (en) * | 1962-02-15 | 1965-07-27 | Scherer Gmbh R P | Coated gelatin capsules |
BE633957A (en) * | 1962-06-22 | |||
US3485840A (en) * | 1964-11-12 | 1969-12-23 | Hoffmann La Roche | 2,4-diamino - 5 - (2',4',5'-substituted benzyl) pyrimidines,intermediates and processes |
JPS555379A (en) * | 1978-03-27 | 1980-01-16 | Muscarella James Allen | Capturing apparatus |
-
1979
- 1979-01-30 JP JP999279A patent/JPS55102517A/en active Pending
-
1980
- 1980-01-04 CA CA000343059A patent/CA1136986A/en not_active Expired
- 1980-01-14 SE SE8000286A patent/SE8000286L/en not_active Application Discontinuation
- 1980-01-28 MX MX808609U patent/MX5865E/en unknown
- 1980-01-28 NL NL8000515A patent/NL8000515A/en not_active Application Discontinuation
- 1980-01-29 DE DE19803003147 patent/DE3003147A1/en not_active Withdrawn
- 1980-01-29 FR FR8001854A patent/FR2447719A1/en active Granted
- 1980-01-29 CH CH70580A patent/CH641958A5/en not_active IP Right Cessation
- 1980-01-29 IT IT67127/80A patent/IT1133051B/en active
- 1980-01-29 ES ES488367A patent/ES488367A0/en active Granted
- 1980-01-30 AR AR279801A patent/AR221525A1/en active
- 1980-01-30 GB GB8003152A patent/GB2041749B/en not_active Expired
-
1981
- 1981-07-31 US US06/288,795 patent/US4461765A/en not_active Expired - Lifetime
Patent Citations (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2415660A1 (en) * | 1973-04-19 | 1974-11-14 | Paolo Chiesi | SUPPOSITORIES CONTAINING A TRIMETHOPRIM-SULFAMETHOXAZOLE COMBINATION AND PROCESS FOR THEIR PRODUCTION |
FR2226156A1 (en) * | 1973-04-19 | 1974-11-15 | Chiesi Paolo | Suppositories contg. trimethoprim and sulphamethoxazole - in two separate layers |
FR2361103A1 (en) * | 1976-07-15 | 1978-03-10 | Basf Ag | SULFONAMIDE-TRIMETHOPRIME SOLUTIONS |
JPS54101415A (en) * | 1978-01-27 | 1979-08-10 | Gea As | Stable suspension containing sulfamethoxal and trimetoprim and production thereof |
Non-Patent Citations (5)
Title |
---|
CA1973 * |
CA1979 * |
CA1980 * |
EXBK/71 * |
EXBK/73 * |
Also Published As
Publication number | Publication date |
---|---|
CH641958A5 (en) | 1984-03-30 |
GB2041749B (en) | 1983-05-05 |
NL8000515A (en) | 1980-08-01 |
GB2041749A (en) | 1980-09-17 |
CA1136986A (en) | 1982-12-07 |
ES8100076A1 (en) | 1980-11-01 |
ES488367A0 (en) | 1980-11-01 |
AR221525A1 (en) | 1981-02-13 |
IT1133051B (en) | 1986-07-09 |
IT8067127A0 (en) | 1980-01-29 |
SE8000286L (en) | 1980-07-31 |
US4461765A (en) | 1984-07-24 |
MX5865E (en) | 1984-08-13 |
DE3003147A1 (en) | 1980-08-07 |
JPS55102517A (en) | 1980-08-05 |
FR2447719B1 (en) | 1984-02-24 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
ST | Notification of lapse |