FR2421614A1 - Composition pharmaceutique a base de 2-(7'-theophyllinomethyl)-1,3-dioxolane - Google Patents

Composition pharmaceutique a base de 2-(7'-theophyllinomethyl)-1,3-dioxolane

Info

Publication number
FR2421614A1
FR2421614A1 FR7818978A FR7818978A FR2421614A1 FR 2421614 A1 FR2421614 A1 FR 2421614A1 FR 7818978 A FR7818978 A FR 7818978A FR 7818978 A FR7818978 A FR 7818978A FR 2421614 A1 FR2421614 A1 FR 2421614A1
Authority
FR
France
Prior art keywords
theophyllinomethyl
dioxolane
pharmaceutical composition
composition based
antibronchospasmodic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7818978A
Other languages
English (en)
Other versions
FR2421614B1 (fr
Inventor
Jose Sebastian Franzone
Teresio Tamietto
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
ABC IST BIOLOG CHEM SpA
Original Assignee
ABC IST BIOLOG CHEM SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ABC IST BIOLOG CHEM SpA filed Critical ABC IST BIOLOG CHEM SpA
Publication of FR2421614A1 publication Critical patent/FR2421614A1/fr
Application granted granted Critical
Publication of FR2421614B1 publication Critical patent/FR2421614B1/fr
Granted legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52Purines, e.g. adenine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/14Antitussive agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/02Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
    • C07D473/06Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
    • C07D473/08Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3 with methyl radicals in positions 1 and 3, e.g. theophylline

Abstract

a. Nouvelle composition à effet antibronchospasmodique et antitussive. b. Cette composition contient à titre de principe la 2-(7'-théophyllinométhyl)-1,3-dioxolane. c. Application en thérapeutique.
FR7818978A 1978-04-06 1978-06-26 Composition pharmaceutique a base de 2-(7'-theophyllinomethyl)-1,3-dioxolane Granted FR2421614A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT22019/78A IT1113122B (it) 1978-04-06 1978-04-06 Composizione farmaceutica ad attivita' antibrocospastica e antitosse

Publications (2)

Publication Number Publication Date
FR2421614A1 true FR2421614A1 (fr) 1979-11-02
FR2421614B1 FR2421614B1 (fr) 1982-09-10

Family

ID=11190276

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7818978A Granted FR2421614A1 (fr) 1978-04-06 1978-06-26 Composition pharmaceutique a base de 2-(7'-theophyllinomethyl)-1,3-dioxolane

Country Status (8)

Country Link
US (1) US4187308A (fr)
JP (1) JPS54138127A (fr)
BE (1) BE868556A (fr)
DE (1) DE2827497C2 (fr)
FR (1) FR2421614A1 (fr)
GB (1) GB1582510A (fr)
IT (1) IT1113122B (fr)
NL (1) NL7807152A (fr)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2480286A1 (fr) * 1980-04-15 1981-10-16 Abc Ist Biolog Chem Spa Nouveaux derives de theophyllinylmethyldioxolane, leurs procedes de preparation et leur application en therapeutique
FR2531337A1 (fr) * 1982-08-04 1984-02-10 Hoechst Lab Nouvelles formes galeniques administrables par voie orale, des derives de la dimethylxanthine solubles

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL59664A0 (en) * 1979-04-05 1980-06-30 Wuelfing J Kg Xanthine derivatives,process for their preparation and their use in pharmaceutical compositions
IT1197516B (it) * 1986-12-24 1988-11-30 Abc Ist Biolog Chem Spa Derivati teofillinmetilanici e teofillinmetilditianici procedimento per la loro preparazione e composizioni farmaceutiche che li comprendono
HU198933B (en) * 1987-11-02 1989-12-28 Chinoin Gyogyszer Es Vegyeszet Process for producing new xanthine derivatives and pharmaceutical compositions comprising same as active ingredient
CN1037604C (zh) * 1994-08-09 1998-03-04 中国医学科学院药物研究所 一种制备平喘镇咳药物的新方法
HUP9700654A2 (hu) * 1997-03-26 1999-09-28 Dezső Korbonits Teobromin tartalmú köhögéscsillapító készítmények
US6423719B1 (en) 1999-02-16 2002-07-23 Upsher-Smith Laboratories, Inc. Method for treating benign prostate hyperplasia
US6313131B1 (en) 1999-02-16 2001-11-06 Upsher-Smith Laboratories, Inc. Method of kidney treatment
CN101647776B (zh) * 2009-09-02 2011-04-20 吴光彦 多索茶碱小容量静脉注射液及其制备方法和质量控制方法
WO2011146031A1 (fr) 2010-05-18 2011-11-24 Bilgic Mahmut Composition pharmaceutique contenant de la n- acétylcystéine et une xanthine
TR201104738A2 (tr) 2011-05-16 2012-12-21 Bi̇lgi̇ç Mahmut N-Asetilsistein içeren farmasötik kombinasyon.
CN102775405B (zh) * 2012-08-23 2014-03-12 天津梅花医药有限公司 一种高溶解度的多索茶碱化合物
CN109796454B (zh) * 2018-12-27 2020-10-23 北京鑫开元医药科技有限公司 多索茶碱杂质及其合成方法、用途、组合物及其制备方法
JP2022184639A (ja) 2021-06-01 2022-12-13 上村工業株式会社 銅エッチング液

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1523273A (fr) * 1967-03-13 1968-05-03 Soc Ind Fab Antibiotiques Sifa Nouveaux dérivés de théophylline et procédé de préparation
FR6106M (fr) * 1967-06-12 1968-06-10

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4085214A (en) * 1976-10-18 1978-04-18 Interx Research Corporation Stable pro-drug forms of theophylline

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1523273A (fr) * 1967-03-13 1968-05-03 Soc Ind Fab Antibiotiques Sifa Nouveaux dérivés de théophylline et procédé de préparation
FR6106M (fr) * 1967-06-12 1968-06-10

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
EXBK/62 *

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2480286A1 (fr) * 1980-04-15 1981-10-16 Abc Ist Biolog Chem Spa Nouveaux derives de theophyllinylmethyldioxolane, leurs procedes de preparation et leur application en therapeutique
FR2531337A1 (fr) * 1982-08-04 1984-02-10 Hoechst Lab Nouvelles formes galeniques administrables par voie orale, des derives de la dimethylxanthine solubles
EP0101963A1 (fr) * 1982-08-04 1984-03-07 Laboratoires Hoechst S.A. Formes galéniques administrables par voie orale des dérivés solubles de la diméthylxanthine

Also Published As

Publication number Publication date
FR2421614B1 (fr) 1982-09-10
NL7807152A (nl) 1979-10-09
DE2827497C2 (de) 1985-10-24
US4187308A (en) 1980-02-05
IT7822019A0 (it) 1978-04-06
IT1113122B (it) 1986-01-20
JPS54138127A (en) 1979-10-26
BE868556A (nl) 1978-10-16
DE2827497A1 (de) 1979-10-11
JPS5715088B2 (fr) 1982-03-29
GB1582510A (en) 1981-01-07

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