FR2400526A2 - Procede de preparation de 3a, 5a-cyclo-6b-alkoxy-d22-25-oxy- ou -acyloxy-bisnorcholestanes et analogues - Google Patents
Procede de preparation de 3a, 5a-cyclo-6b-alkoxy-d22-25-oxy- ou -acyloxy-bisnorcholestanes et analoguesInfo
- Publication number
- FR2400526A2 FR2400526A2 FR7722815A FR7722815A FR2400526A2 FR 2400526 A2 FR2400526 A2 FR 2400526A2 FR 7722815 A FR7722815 A FR 7722815A FR 7722815 A FR7722815 A FR 7722815A FR 2400526 A2 FR2400526 A2 FR 2400526A2
- Authority
- FR
- France
- Prior art keywords
- cyclo
- alpha
- derivs
- hydroxy
- intermediates
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 239000000543 intermediate Substances 0.000 title abstract 2
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- JWUBBDSIWDLEOM-XHQRYOPUSA-N (3e)-3-[(2e)-2-[1-(6-hydroxy-6-methylheptan-2-yl)-7a-methyl-2,3,3a,5,6,7-hexahydro-1h-inden-4-ylidene]ethylidene]-4-methylidenecyclohexan-1-ol Chemical class C1CCC2(C)C(C(CCCC(C)(C)O)C)CCC2\C1=C\C=C1/CC(O)CCC1=C JWUBBDSIWDLEOM-XHQRYOPUSA-N 0.000 abstract 1
- INBGSXNNRGWLJU-ZHHJOTBYSA-N 25-hydroxycholesterol Chemical compound C1C=C2C[C@@H](O)CC[C@]2(C)[C@@H]2[C@@H]1[C@@H]1CC[C@H]([C@@H](CCCC(C)(C)O)C)[C@@]1(C)CC2 INBGSXNNRGWLJU-ZHHJOTBYSA-N 0.000 abstract 1
- INBGSXNNRGWLJU-UHFFFAOYSA-N 25epsilon-Hydroxycholesterin Natural products C1C=C2CC(O)CCC2(C)C2C1C1CCC(C(CCCC(C)(C)O)C)C1(C)CC2 INBGSXNNRGWLJU-UHFFFAOYSA-N 0.000 abstract 1
- IAYPIBMASNFSPL-UHFFFAOYSA-N Ethylene oxide Chemical compound C1CO1 IAYPIBMASNFSPL-UHFFFAOYSA-N 0.000 abstract 1
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 1
- DLEDOFVPSDKWEF-UHFFFAOYSA-N lithium butane Chemical compound [Li+].CCC[CH2-] DLEDOFVPSDKWEF-UHFFFAOYSA-N 0.000 abstract 1
- LSEFCHWGJNHZNT-UHFFFAOYSA-M methyl(triphenyl)phosphanium;bromide Chemical compound [Br-].C=1C=CC=CC=1[P+](C=1C=CC=CC=1)(C)C1=CC=CC=C1 LSEFCHWGJNHZNT-UHFFFAOYSA-M 0.000 abstract 1
- MZRVEZGGRBJDDB-UHFFFAOYSA-N n-Butyllithium Substances [Li]CCCC MZRVEZGGRBJDDB-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US05/708,821 US4058538A (en) | 1975-01-27 | 1976-07-26 | 3α,5α-Cyclo-6β-alkoxy-α22 -bis-nor cholestene derivatives |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| FR2400526A2 true FR2400526A2 (fr) | 1979-03-16 |
| FR2400526B2 FR2400526B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1982-07-09 |
Family
ID=24847311
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FR7722815A Granted FR2400526A2 (fr) | 1976-07-26 | 1977-07-25 | Procede de preparation de 3a, 5a-cyclo-6b-alkoxy-d22-25-oxy- ou -acyloxy-bisnorcholestanes et analogues |
Country Status (7)
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0019059A1 (de) * | 1979-05-18 | 1980-11-26 | F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft | Verfahren zur Herstellung von Cholestenderivaten und neue Zwischenprodukte in deren Herstellung |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2301537A1 (fr) * | 1975-01-27 | 1976-09-17 | Upjohn Co | Procédé de PREPARATION DE 3ALPHA,5ALPHA-CYCLO-6BETA-ALKOXY-DELTA22-25-OXY-OU-ACYLOXY-BISNORCHOLESTANES ET ANALOGUES |
-
1977
- 1977-07-01 IL IL52435A patent/IL52435A0/xx unknown
- 1977-07-08 NL NL7707612A patent/NL7707612A/xx not_active Application Discontinuation
- 1977-07-22 DE DE19772733116 patent/DE2733116A1/de not_active Withdrawn
- 1977-07-22 GB GB30845/77A patent/GB1537199A/en not_active Expired
- 1977-07-25 JP JP8845777A patent/JPS5318555A/ja active Pending
- 1977-07-25 FR FR7722815A patent/FR2400526A2/fr active Granted
- 1977-07-26 CH CH921977A patent/CH631186A5/de not_active IP Right Cessation
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2301537A1 (fr) * | 1975-01-27 | 1976-09-17 | Upjohn Co | Procédé de PREPARATION DE 3ALPHA,5ALPHA-CYCLO-6BETA-ALKOXY-DELTA22-25-OXY-OU-ACYLOXY-BISNORCHOLESTANES ET ANALOGUES |
Non-Patent Citations (1)
| Title |
|---|
| EXBK/74 * |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0019059A1 (de) * | 1979-05-18 | 1980-11-26 | F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft | Verfahren zur Herstellung von Cholestenderivaten und neue Zwischenprodukte in deren Herstellung |
Also Published As
| Publication number | Publication date |
|---|---|
| GB1537199A (en) | 1978-12-29 |
| CH631186A5 (en) | 1982-07-30 |
| FR2400526B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1982-07-09 |
| JPS5318555A (en) | 1978-02-20 |
| NL7707612A (nl) | 1978-01-30 |
| DE2733116A1 (de) | 1978-02-02 |
| IL52435A0 (en) | 1977-10-31 |
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