FR2396000A1 - Nouveaux derives a-acetyleniques d'histamine utiles notamment comme antihistaminiques et leur procede de preparation - Google Patents
Nouveaux derives a-acetyleniques d'histamine utiles notamment comme antihistaminiques et leur procede de preparationInfo
- Publication number
- FR2396000A1 FR2396000A1 FR7819354A FR7819354A FR2396000A1 FR 2396000 A1 FR2396000 A1 FR 2396000A1 FR 7819354 A FR7819354 A FR 7819354A FR 7819354 A FR7819354 A FR 7819354A FR 2396000 A1 FR2396000 A1 FR 2396000A1
- Authority
- FR
- France
- Prior art keywords
- antihistaminics
- histamine
- useful
- preparation
- new
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/68—Halogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/88—Nitrogen atoms, e.g. allantoin
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Les médicaments selon l'invention sont des dérivés de propargylamines de formule générale :
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US05/812,266 US4100349A (en) | 1977-07-01 | 1977-07-01 | α-Acetylenic derivatives of histamine and related compounds |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2396000A1 true FR2396000A1 (fr) | 1979-01-26 |
FR2396000B1 FR2396000B1 (fr) | 1980-07-18 |
Family
ID=25209057
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR7819354A Granted FR2396000A1 (fr) | 1977-07-01 | 1978-06-28 | Nouveaux derives a-acetyleniques d'histamine utiles notamment comme antihistaminiques et leur procede de preparation |
Country Status (8)
Country | Link |
---|---|
US (1) | US4100349A (fr) |
AU (1) | AU517270B2 (fr) |
BE (1) | BE868595A (fr) |
FR (1) | FR2396000A1 (fr) |
GB (1) | GB2001308B (fr) |
IT (1) | IT1105057B (fr) |
NZ (1) | NZ187544A (fr) |
ZA (1) | ZA783276B (fr) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
USRE31588E (en) * | 1977-06-03 | 1984-05-22 | Bristol-Myers Company | Imidazolylmethylthioethyl alkynyl guanidines |
FR2586562B1 (fr) * | 1985-09-02 | 1989-03-10 | Inst Nat Sante Rech Med | Composition pharmaceutique contenant de l'a-methylhistamine |
Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4088667A (en) * | 1977-07-01 | 1978-05-09 | Merrell Toraude Et Compagnie | Lower alkyl 2-tri-(lower)alkylsilylacetylene-N-carbethoxyglycinates and process for using same |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3169971A (en) * | 1965-02-16 | A-alkyl histidines | ||
GB715182A (en) * | 1951-09-19 | 1954-09-08 | Roche Products Ltd | A novel imidazole derivative and process for the manufacture thereof |
US3387031A (en) * | 1961-06-08 | 1968-06-04 | Union Carbide Corp | Synthesis of alpha-amino acid amide hydrohalides |
-
1977
- 1977-07-01 US US05/812,266 patent/US4100349A/en not_active Expired - Lifetime
-
1978
- 1978-06-07 ZA ZA00783276A patent/ZA783276B/xx unknown
- 1978-06-13 NZ NZ187544A patent/NZ187544A/xx unknown
- 1978-06-21 AU AU37323/78A patent/AU517270B2/en not_active Expired
- 1978-06-27 IT IT50049/78A patent/IT1105057B/it active
- 1978-06-27 GB GB787827969A patent/GB2001308B/en not_active Expired
- 1978-06-28 FR FR7819354A patent/FR2396000A1/fr active Granted
- 1978-06-29 BE BE188955A patent/BE868595A/fr not_active IP Right Cessation
Patent Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4088667A (en) * | 1977-07-01 | 1978-05-09 | Merrell Toraude Et Compagnie | Lower alkyl 2-tri-(lower)alkylsilylacetylene-N-carbethoxyglycinates and process for using same |
FR2396014A1 (fr) * | 1977-07-01 | 1979-01-26 | Merrell Toraude & Co | Esters d'acides silylacetyleniques et leurs utilisations therapeutiques, notamment comme antibacteriens |
Also Published As
Publication number | Publication date |
---|---|
AU517270B2 (en) | 1981-07-16 |
US4100349A (en) | 1978-07-11 |
GB2001308B (en) | 1982-01-13 |
FR2396000B1 (fr) | 1980-07-18 |
ZA783276B (en) | 1979-06-27 |
BE868595A (fr) | 1978-10-16 |
AU3732378A (en) | 1980-01-03 |
GB2001308A (en) | 1979-01-31 |
NZ187544A (en) | 1980-08-26 |
IT1105057B (it) | 1985-10-28 |
IT7850049A0 (it) | 1978-06-27 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
FR2378521A1 (fr) | Derives du carbostyrile, utiles notamment comme stimulants des centres b- adrenorecepteurs, et leur procede de preparation | |
FR2360587A1 (fr) | Nouveaux derives d'amino-alcoyl-furannes utiles comme medicaments | |
FR2434154A1 (fr) | Nouveaux derives d'imidazole, utiles notamment comme anticonvulsivants, et leur procede de preparation | |
FR2395990A1 (fr) | Derives a-acetyleniques d'amines utiles notamment comme inhibiteurs de certaines decarboxylases et leur procede de preparation | |
FR2376147A1 (fr) | Prostaglandines bicycliques, utiles notamment comme anti-agglutinants des plaquettes sanguines et leur procede de preparation | |
FR2416227A1 (fr) | Nouveaux derives de 2h-benzofuranne-3-one, utiles notamment comme anti-allergiques, et leur procede de preparation | |
FR2364219A1 (fr) | Derives de thiazolidine, leur procede de preparation et leur application en therapeutique | |
FR2387980A1 (fr) | Nouveaux 2-(2,2-diarylalkyl)-1-azabicyclo (2.2.2) octanes, utiles notamment comme antidiarrheiques, et leur procede de preparation | |
FR2431505A1 (fr) | Nouveaux n-(diaminophosphinyl)arylcarboxamides, utiles notamment comme inhibiteurs de l'urease | |
FR2380285A1 (fr) | Nouveaux derives insatures d'acides 7-acylamido-3-cephem-4-carboxyliques, utiles notamment comme agents antibacteriens, et leur procede de preparation | |
FR2360558A1 (fr) | Nouveaux esters de l'epinine, utiles notamment en cardiotherapie, et leur procede de preparation | |
FR2400018A1 (fr) | Nouveaux acides imidazolinylbenzoiques, leurs esters et leurs sels, leur procede de preparation et leur application comme insecticides | |
FR2443471A1 (fr) | Derives du type thiazolidine de la progesterone utiles notamment comme precurseurs de medicaments antiacne et antiseborrhee | |
FR2394522A1 (fr) | Nouveaux derives d'acides (s-phenenyl tris(carbonylimino))-5,5',5''tri-benzene-carboxyliques utiles notamment comme inhibiteurs du complement, et leur procede de preparation | |
FR2361879A2 (fr) | Nouvelles 4,5,6,7- tetrahydro-7-oxo (ou hydroxy)benzo (b)thienyl-4-amines utiles notamment comme agents de croissance pour animaux et leur procede de preparation | |
FR2358388A1 (fr) | Nouvelles 1,2,3,4-tetrahydro-4-imino-1-naphtylurees substituees, utiles notamment comme agents de croissance pour animaux, et leur procede de preparation | |
FR2430232A1 (fr) | Nouveaux acides arylaminobenzoiques utiles notamment comme agents hypoglycemiants | |
FR2446829A1 (fr) | Derives de polymethylene disubstitues en alpha, omega, procede pour leur preparation et compositions pharmaceutiques les contenant | |
FR2403994A1 (fr) | Nouvelles 1-(2-chloroethyl)-1-nitrosourees utiles notamment comme agents antitumoraux et leur procede de preparation | |
FR2401935A1 (fr) | Nouveaux 25-alkylcholesterols utiles notamment comme hypocholesterolemiants et leur procede de preparation | |
FR2422638A1 (fr) | Nouveaux derives de 3,3-dichloro-2-azetidinone, utiles notamment comme agents anti-inflammatoires | |
FR2357574A1 (fr) | Nouveaux derives 16-acylthio de l'acide fusidique, utiles notamment comme antimicrobiens et leur procede de preparation | |
FR2396000A1 (fr) | Nouveaux derives a-acetyleniques d'histamine utiles notamment comme antihistaminiques et leur procede de preparation | |
FR2361382A1 (fr) | 2-vinyl-chromones substituees, utiles notamment comme anti-allergiques, et leur procede de preparation | |
FR2414494A1 (fr) | Nouveaux derives d'acide 1,5-cyclohexadienecarboxyliques substitues, utiles notamment comme antiepileptiques, et leur procede de preparation |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
ST | Notification of lapse |