IT7850049A0 - Derivati alfa-acetilenici di istamina con attivita' farmaceutica e procedimento per la loro preparazione - Google Patents
Derivati alfa-acetilenici di istamina con attivita' farmaceutica e procedimento per la loro preparazioneInfo
- Publication number
- IT7850049A0 IT7850049A0 IT7850049A IT5004978A IT7850049A0 IT 7850049 A0 IT7850049 A0 IT 7850049A0 IT 7850049 A IT7850049 A IT 7850049A IT 5004978 A IT5004978 A IT 5004978A IT 7850049 A0 IT7850049 A0 IT 7850049A0
- Authority
- IT
- Italy
- Prior art keywords
- histamine
- alpha
- procedure
- preparation
- pharmaceutical activity
- Prior art date
Links
- HSFWRNGVRCDJHI-UHFFFAOYSA-N alpha-acetylene Natural products C#C HSFWRNGVRCDJHI-UHFFFAOYSA-N 0.000 title 1
- 229960001340 histamine Drugs 0.000 title 1
- NTYJJOPFIAHURM-UHFFFAOYSA-N histamine Natural products NCCC1=CN=CN1 NTYJJOPFIAHURM-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/68—Halogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/88—Nitrogen atoms, e.g. allantoin
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US05/812,266 US4100349A (en) | 1977-07-01 | 1977-07-01 | α-Acetylenic derivatives of histamine and related compounds |
Publications (2)
Publication Number | Publication Date |
---|---|
IT7850049A0 true IT7850049A0 (it) | 1978-06-27 |
IT1105057B IT1105057B (it) | 1985-10-28 |
Family
ID=25209057
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IT50049/78A IT1105057B (it) | 1977-07-01 | 1978-06-27 | Derivati alfa acetilenici di istamina con attivita' farmaceutica e procedimento per la loro preparazione |
Country Status (8)
Country | Link |
---|---|
US (1) | US4100349A (it) |
AU (1) | AU517270B2 (it) |
BE (1) | BE868595A (it) |
FR (1) | FR2396000A1 (it) |
GB (1) | GB2001308B (it) |
IT (1) | IT1105057B (it) |
NZ (1) | NZ187544A (it) |
ZA (1) | ZA783276B (it) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
USRE31588E (en) * | 1977-06-03 | 1984-05-22 | Bristol-Myers Company | Imidazolylmethylthioethyl alkynyl guanidines |
FR2586562B1 (fr) * | 1985-09-02 | 1989-03-10 | Inst Nat Sante Rech Med | Composition pharmaceutique contenant de l'a-methylhistamine |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3169971A (en) * | 1965-02-16 | A-alkyl histidines | ||
GB715182A (en) * | 1951-09-19 | 1954-09-08 | Roche Products Ltd | A novel imidazole derivative and process for the manufacture thereof |
US3387031A (en) * | 1961-06-08 | 1968-06-04 | Union Carbide Corp | Synthesis of alpha-amino acid amide hydrohalides |
US4088667A (en) * | 1977-07-01 | 1978-05-09 | Merrell Toraude Et Compagnie | Lower alkyl 2-tri-(lower)alkylsilylacetylene-N-carbethoxyglycinates and process for using same |
-
1977
- 1977-07-01 US US05/812,266 patent/US4100349A/en not_active Expired - Lifetime
-
1978
- 1978-06-07 ZA ZA00783276A patent/ZA783276B/xx unknown
- 1978-06-13 NZ NZ187544A patent/NZ187544A/xx unknown
- 1978-06-21 AU AU37323/78A patent/AU517270B2/en not_active Expired
- 1978-06-27 IT IT50049/78A patent/IT1105057B/it active
- 1978-06-27 GB GB787827969A patent/GB2001308B/en not_active Expired
- 1978-06-28 FR FR7819354A patent/FR2396000A1/fr active Granted
- 1978-06-29 BE BE188955A patent/BE868595A/xx not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
AU517270B2 (en) | 1981-07-16 |
US4100349A (en) | 1978-07-11 |
GB2001308B (en) | 1982-01-13 |
FR2396000B1 (it) | 1980-07-18 |
ZA783276B (en) | 1979-06-27 |
BE868595A (fr) | 1978-10-16 |
AU3732378A (en) | 1980-01-03 |
GB2001308A (en) | 1979-01-31 |
NZ187544A (en) | 1980-08-26 |
IT1105057B (it) | 1985-10-28 |
FR2396000A1 (fr) | 1979-01-26 |
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