FR2361897A1 - Nouveaux derives de la cephalosporine, leurs intermediaires et procede pour les preparer - Google Patents

Nouveaux derives de la cephalosporine, leurs intermediaires et procede pour les preparer

Info

Publication number
FR2361897A1
FR2361897A1 FR7636974A FR7636974A FR2361897A1 FR 2361897 A1 FR2361897 A1 FR 2361897A1 FR 7636974 A FR7636974 A FR 7636974A FR 7636974 A FR7636974 A FR 7636974A FR 2361897 A1 FR2361897 A1 FR 2361897A1
Authority
FR
France
Prior art keywords
intermediaries
preparing
cephalosporin derivatives
new cephalosporin
new
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7636974A
Other languages
English (en)
French (fr)
Other versions
FR2361897B1 (en:Method
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
GlaxoSmithKline LLC
Original Assignee
SmithKline Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by SmithKline Corp filed Critical SmithKline Corp
Publication of FR2361897A1 publication Critical patent/FR2361897A1/fr
Application granted granted Critical
Publication of FR2361897B1 publication Critical patent/FR2361897B1/fr
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D257/00Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
    • C07D257/02Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D257/04Five-membered rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
FR7636974A 1975-12-09 1976-12-08 Nouveaux derives de la cephalosporine, leurs intermediaires et procede pour les preparer Granted FR2361897A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/639,033 US4025626A (en) 1975-12-09 1975-12-09 7-Acyl-3-(ureidoalkyl substituted tetrazolylthiomethyl)-cephalosporins

Publications (2)

Publication Number Publication Date
FR2361897A1 true FR2361897A1 (fr) 1978-03-17
FR2361897B1 FR2361897B1 (en:Method) 1982-10-29

Family

ID=24562451

Family Applications (3)

Application Number Title Priority Date Filing Date
FR7636974A Granted FR2361897A1 (fr) 1975-12-09 1976-12-08 Nouveaux derives de la cephalosporine, leurs intermediaires et procede pour les preparer
FR7713410A Granted FR2337730A1 (fr) 1975-12-09 1977-05-03 Nouveaux derives de cephalosporines
FR7713411A Granted FR2361376A1 (fr) 1975-12-09 1977-05-03 Nouveaux tetrazoles

Family Applications After (2)

Application Number Title Priority Date Filing Date
FR7713410A Granted FR2337730A1 (fr) 1975-12-09 1977-05-03 Nouveaux derives de cephalosporines
FR7713411A Granted FR2361376A1 (fr) 1975-12-09 1977-05-03 Nouveaux tetrazoles

Country Status (7)

Country Link
US (4) US4025626A (en:Method)
JP (1) JPS6053027B2 (en:Method)
BE (1) BE849003A (en:Method)
DE (1) DE2655692A1 (en:Method)
FR (3) FR2361897A1 (en:Method)
GB (3) GB1573004A (en:Method)
IE (1) IE44570B1 (en:Method)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK586175A (da) * 1974-12-28 1976-06-29 Asahi Chemical Ind Cephalosporin-forbindelser
US4198406A (en) * 1975-11-27 1980-04-15 Beecham Group Limited Carbamoyl heterocyclicthio cephalosporins and pharmaceutical compositions formulated therewith
AU498968B2 (en) * 1976-03-03 1979-03-29 Sumitomo Chemical Company, Limited Cephalosporins
JPS5321191A (en) * 1976-08-10 1978-02-27 Shionogi & Co Ltd 7-arylmalonamidocephem derivatives
US4117123A (en) * 1977-06-09 1978-09-26 Smithkline Corporation 7-Acylamino-3-[1-(2-sulfamidoethyl)tetrazol-5-ylthiomethyl]-3-cephem-4-carboxylic acids
US4148997A (en) * 1977-11-07 1979-04-10 Yeda Research And Development Co., Ltd. 7-[Sulfomethyl)phenyl]acetamidocephalosporin derivatives
US4226806A (en) * 1977-11-07 1980-10-07 Yeda Research And Development Co. Ltd. 7-[(Sulfomethyl)phenyl]acetamidocephalosporin derivatives
US4180658A (en) * 1978-02-24 1979-12-25 Bristol-Myers Company 7[-2-Alkoxyamino(acetamido)]cephalosporin derivatives
US4338452A (en) * 1980-09-17 1982-07-06 Eli Lilly And Company 1-and 2-(1-Alkyl-1H-tetrazol-5-yl-methyl)-1H-tetrazol-5-thiols and 1-cyanomethyl tetrazole-5-thiol
JPS59152385A (ja) * 1983-02-17 1984-08-31 Shionogi & Co Ltd ヒドロキサム酸系セフアロスポリン誘導体
JPS6361119A (ja) * 1986-09-01 1988-03-17 Ee & D:Kk 複数のロ−ドセルを用いた秤量装置
JPH0259446U (en:Method) * 1988-10-25 1990-05-01
US6903105B2 (en) * 2003-02-19 2005-06-07 Parion Sciences, Inc. Sodium channel blockers

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3819623A (en) * 1968-04-12 1974-06-25 Fujisawa Pharmaceutical Co 3,7-disubstituted cephalosporin compounds
US3867380A (en) * 1971-02-18 1975-02-18 Smithkline Corp 3-Heterocyclic thiomethylcephalosporins
US3828037A (en) * 1972-07-20 1974-08-06 Smithkline Corp Trifluoromethylmercaptoacetamidocephalosporins
GB1478055A (en) 1973-07-27 1977-06-29 Erba Carlo Spa Cephalosporin compounds
JPS57873B2 (en:Method) 1973-12-25 1982-01-08

Also Published As

Publication number Publication date
IE44570L (en) 1977-06-09
FR2337730A1 (fr) 1977-08-05
FR2361376A1 (fr) 1978-03-10
US4025626A (en) 1977-05-24
JPS5273891A (en) 1977-06-21
GB1573006A (en) 1980-08-13
IE44570B1 (en) 1982-01-13
US4068073A (en) 1978-01-10
BE849003A (fr) 1977-06-02
US4066761A (en) 1978-01-03
US4096256A (en) 1978-06-20
FR2361897B1 (en:Method) 1982-10-29
GB1573005A (en) 1980-08-13
FR2361376B1 (en:Method) 1981-03-27
FR2337730B1 (en:Method) 1981-01-09
GB1573004A (en) 1980-08-13
JPS6053027B2 (ja) 1985-11-22
DE2655692A1 (de) 1977-06-16

Similar Documents

Publication Publication Date Title
FR2384765A1 (fr) Derives amino-substitues du furanne et procede pour leur preparation
FR2387234A1 (fr) Derives de cephalosporine, leur procede de preparation et leurs applications en therapeutique
FR2357541A1 (fr) Composes polyeniques et leur procede de preparation
FR2446289A1 (fr) Compose de 2-penem, procede de preparation et composition pharmaceutique obtenue
FR2381052A1 (fr) Derives de cephalosporine, leur procede de preparation et leur utilisation
FR2361897A1 (fr) Nouveaux derives de la cephalosporine, leurs intermediaires et procede pour les preparer
FR2389629A1 (en:Method)
FR2428042A1 (fr) Procede de preparation d'analogues de cephalosporine et nouveaux produits ainsi obtenus, a activite antimicrobienne
FR2390433A1 (fr) Composes utiles pour la preparation de derives d'acide penicillanique
FR2370028A1 (fr) Hydroxylamines alkylees, leur procede de preparation et leur emploi comme medicaments
FR2386544A1 (fr) Procede pour la preparation de derives d'imidazodiazepine
FR2406630A1 (fr) 2-phenoxy-5-trifluoromethylpyridines et leur procede de preparation
FR2375239A1 (fr) Derives d'acide 7-amino-8-oxo-3-oxa-1-azabicyclo-(4.2.0)octane-2-carboxylique
FR2373546A1 (fr) Derives thio-oxime de cephalosporines et de penicillines, utiles comme inhibiteurs de b-lactamases
FR2366284A1 (fr) Derives de benzimidazole, leur procede de leur preparation et leur utilisation comme anthelmintiques
FR2356626A1 (fr) Acides ureidoacetohydroxamiques substitues
FR2355020A1 (fr) Antibiotiques de b-lactames et leur procede de preparation
FR2383152A1 (fr) Procede de preparation du 2-methyl-3-prenyl-4,5,6-trimethoxyphenol
FR2375206A1 (fr) Nouvelles isothiourees, procede pour les preparer et compositions pharmaceutiques les contenant
FR2429211A1 (fr) Procede de production de derives de n-methylbenzothiazolone substitues en position 4
FR2433009A1 (fr) Procede pour la preparation de dicyclopentylene(2,2'-bis(4-alkyl-6-t-butylphenols))
FR2359133A1 (fr) Procede de preparation de (vinyl 2,2-disubstitue)-g-butyrolactones
FR2374322A1 (fr) Procede pour la preparation de nouveaux derives de la piperazine et leur utilisation comme vasodilatateurs et produits anti-arythmiques
FR2361876A1 (fr) 2,9-dioxatricyclo(4,3,1,03,7)decanes, procede pour leur preparation ainsi que les produits intermediaires convenant a cet effet
FR2362808A1 (fr) Procede de preparation de 2-alkyl-2-methylpropane-1,3-diols

Legal Events

Date Code Title Description
ST Notification of lapse