FR2338930A1 - Procede de preparation de composes d'azetidinone et nouveaux produits ainsi obtenus, a activite antibacterienne - Google Patents

Procede de preparation de composes d'azetidinone et nouveaux produits ainsi obtenus, a activite antibacterienne

Info

Publication number
FR2338930A1
FR2338930A1 FR7701767A FR7701767A FR2338930A1 FR 2338930 A1 FR2338930 A1 FR 2338930A1 FR 7701767 A FR7701767 A FR 7701767A FR 7701767 A FR7701767 A FR 7701767A FR 2338930 A1 FR2338930 A1 FR 2338930A1
Authority
FR
France
Prior art keywords
preparation
antibacterial activity
new products
azetidinone compounds
azetidinone
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7701767A
Other languages
English (en)
Other versions
FR2338930B1 (fr
Inventor
Shoichiro Uyeo
Tsutomu Aoki
Wataru Nagata
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Shionogi and Co Ltd
Original Assignee
Shionogi and Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shionogi and Co Ltd filed Critical Shionogi and Co Ltd
Publication of FR2338930A1 publication Critical patent/FR2338930A1/fr
Application granted granted Critical
Publication of FR2338930B1 publication Critical patent/FR2338930B1/fr
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • C07D205/09—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a sulfur atom directly attached in position 4
    • C07D205/095—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a sulfur atom directly attached in position 4 and with a nitrogen atom directly attached in position 3
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FR7701767A 1976-01-23 1977-01-21 Procede de preparation de composes d'azetidinone et nouveaux produits ainsi obtenus, a activite antibacterienne Granted FR2338930A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP51006960A JPS6019315B2 (ja) 1976-01-23 1976-01-23 アゼチジノン化合物

Publications (2)

Publication Number Publication Date
FR2338930A1 true FR2338930A1 (fr) 1977-08-19
FR2338930B1 FR2338930B1 (fr) 1979-03-09

Family

ID=11652774

Family Applications (2)

Application Number Title Priority Date Filing Date
FR7701767A Granted FR2338930A1 (fr) 1976-01-23 1977-01-21 Procede de preparation de composes d'azetidinone et nouveaux produits ainsi obtenus, a activite antibacterienne
FR7725950A Granted FR2355845A1 (fr) 1976-01-23 1977-08-25 Procede de preparation de derives de penam et nouveaux produits ainsi obtenus, a activite antibacterienne

Family Applications After (1)

Application Number Title Priority Date Filing Date
FR7725950A Granted FR2355845A1 (fr) 1976-01-23 1977-08-25 Procede de preparation de derives de penam et nouveaux produits ainsi obtenus, a activite antibacterienne

Country Status (8)

Country Link
US (1) US4058521A (fr)
JP (1) JPS6019315B2 (fr)
CA (1) CA1070672A (fr)
CH (1) CH632271A5 (fr)
DE (1) DE2702527A1 (fr)
FR (2) FR2338930A1 (fr)
GB (1) GB1529662A (fr)
NL (1) NL7700712A (fr)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1136132A (fr) * 1975-02-17 1982-11-23 Teruji Tsuji Cyclisation pour fermer des noyaux cephem et intermediaires ainsi obtenus
US4024152A (en) * 1975-09-19 1977-05-17 Eli Lilly And Company 4-Dithio-3-imido-azetidin-2-ones
US4195021A (en) * 1977-10-26 1980-03-25 Eli Lilly And Company 1,3-Disubstituted 2-azetidinone antibitotics
US4168314A (en) * 1977-11-17 1979-09-18 Merck & Co., Inc. 6-(1'-Hydroxyethyl)-2-aminoethylthio-pen-2-em-3-carboxylic acid
US4340539A (en) * 1980-01-21 1982-07-20 Bristol-Myers Company Derivatives of 6-bromo penicillanic acid
JPS5738769A (en) * 1980-08-18 1982-03-03 Sankyo Co Ltd Azetidinone derivative and its preparation
US4380512A (en) * 1980-12-11 1983-04-19 Bristol-Myers Company 2β-Chloromethyl-2α-methylpenam-3α-carboxylic acid sulfone and salts and esters thereof
GB2099817B (en) * 1981-04-10 1985-05-15 Otsuka Kagaku Yakuhin Azetidinone derivatives and process for the preparation of the same
US4482491A (en) * 1981-05-01 1984-11-13 Otsuka Kagaku Yakuhin Kabushiki Kaisha Thiazolinoazetidinone derivatives and process for the preparation of the same
EP0065488B1 (fr) * 1981-05-19 1985-08-14 Ciba-Geigy Ag Procédé de préparation de dérivés de 4-thio-azétidinone
AU541028B2 (en) * 1982-06-21 1984-12-13 Taiho Pharmaceutical Co., Ltd. 6-unsubstituted penicillin derivatives
US4532077A (en) * 1982-08-25 1985-07-30 Otsuka Kagaku Yakuhin Kabushiki Kaisha Thiazolineazetidinone-type compounds
JPS59101485A (ja) * 1982-11-29 1984-06-12 Otsuka Chem Co Ltd アセチジノン誘導体
JPS60204893A (ja) * 1984-03-27 1985-10-16 Otsuka Chem Co Ltd ２，２−ビスハロメチルペナム誘導体の製造法
JPS61178961A (ja) * 1985-02-01 1986-08-11 Otsuka Chem Co Ltd アゼチジノン誘導体の製造法
EP0206000A1 (fr) * 1985-06-01 1986-12-30 F. Hoffmann-La Roche Ag Acides (2,3)-alpha-méthylènepénam-3-carboxyliques et leurs dérivés
JPS6212783A (ja) * 1985-06-01 1987-01-21 エフ・ホフマン―ラ　ロシユ　アーゲー （２，３）−α−メチレンペナム−３−カルボン酸及びその誘導体
KR100370291B1 (ko) * 1996-08-23 2003-08-21 주식회사 코오롱 2-브로모설피닐 아제티디논 유도체의 제조방법
CN101525340B (zh) * 2008-03-04 2011-05-18 山东方兴科技开发有限公司 7-苯乙酰氨基-3-氯甲基头孢烷烯酸对甲氧基苄酯的合成方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3275626A (en) * 1962-07-31 1966-09-27 Lilly Co Eli Penicillin conversion via sulfoxide
FR2143211B1 (fr) * 1971-06-24 1975-10-31 Fujisawa Pharmaceutical Co
SE417968B (sv) * 1972-10-20 1981-04-27 Fujisawa Pharmaceutical Co Forfarande for framstellning av penamderivat
JPS5535394B2 (fr) * 1972-12-23 1980-09-12

Also Published As

Publication number Publication date
JPS6019315B2 (ja) 1985-05-15
GB1529662A (en) 1978-10-25
FR2355845B1 (fr) 1980-12-05
CA1070672A (fr) 1980-01-29
US4058521A (en) 1977-11-15
DE2702527A1 (de) 1977-07-28
NL7700712A (nl) 1977-07-26
JPS5291852A (en) 1977-08-02
CH632271A5 (de) 1982-09-30
FR2355845A1 (fr) 1978-01-20
FR2338930B1 (fr) 1979-03-09

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Legal Events

Date Code Title Description
ST Notification of lapse