FR2295933A1 - Cyclopentene-diols et leurs esters acyliques, utilisables pour la fabrication de medicaments, et preparation de ces composes - Google Patents

Cyclopentene-diols et leurs esters acyliques, utilisables pour la fabrication de medicaments, et preparation de ces composes

Info

Publication number
FR2295933A1
FR2295933A1 FR7539824A FR7539824A FR2295933A1 FR 2295933 A1 FR2295933 A1 FR 2295933A1 FR 7539824 A FR7539824 A FR 7539824A FR 7539824 A FR7539824 A FR 7539824A FR 2295933 A1 FR2295933 A1 FR 2295933A1
Authority
FR
France
Prior art keywords
cyclopentene
diols
compounds
manufacture
preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7539824A
Other languages
English (en)
Other versions
FR2295933B1 (fr
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Teijin Ltd
Original Assignee
Teijin Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP14826374A external-priority patent/JPS5176484A/ja
Priority claimed from JP14826674A external-priority patent/JPS5176486A/ja
Priority claimed from JP2948675A external-priority patent/JPS51106789A/ja
Priority claimed from JP4579375A external-priority patent/JPS51121595A/ja
Priority claimed from JP4652575A external-priority patent/JPS51123889A/ja
Priority claimed from JP4740875A external-priority patent/JPS51123890A/ja
Application filed by Teijin Ltd filed Critical Teijin Ltd
Publication of FR2295933A1 publication Critical patent/FR2295933A1/fr
Application granted granted Critical
Publication of FR2295933B1 publication Critical patent/FR2295933B1/fr
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12P—FERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P41/00—Processes using enzymes or microorganisms to separate optical isomers from a racemic mixture
    • C12P41/003—Processes using enzymes or microorganisms to separate optical isomers from a racemic mixture by ester formation, lactone formation or the inverse reactions
    • C12P41/004—Processes using enzymes or microorganisms to separate optical isomers from a racemic mixture by ester formation, lactone formation or the inverse reactions by esterification of alcohol- or thiol groups in the enantiomers or the inverse reaction
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C35/00—Compounds having at least one hydroxy or O-metal group bound to a carbon atom of a ring other than a six-membered aromatic ring
    • C07C35/02—Compounds having at least one hydroxy or O-metal group bound to a carbon atom of a ring other than a six-membered aromatic ring monocyclic
    • C07C35/06—Compounds having at least one hydroxy or O-metal group bound to a carbon atom of a ring other than a six-membered aromatic ring monocyclic containing a five-membered rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D309/08—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D309/10—Oxygen atoms
    • C07D309/12—Oxygen atoms only hydrogen atoms and one oxygen atom directly attached to ring carbon atoms, e.g. tetrahydropyranyl ethers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804—Compounds having Si-O-C linkages
    • C—CHEMISTRY; METALLURGY
    • C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12N—MICROORGANISMS OR ENZYMES; COMPOSITIONS THEREOF; PROPAGATING, PRESERVING, OR MAINTAINING MICROORGANISMS; MUTATION OR GENETIC ENGINEERING; CULTURE MEDIA
    • C12N9/00—Enzymes; Proenzymes; Compositions thereof; Processes for preparing, activating, inhibiting, separating or purifying enzymes
    • C12N9/14—Hydrolases (3)
    • C12N9/16—Hydrolases (3) acting on ester bonds (3.1)
    • C12N9/18—Carboxylic ester hydrolases (3.1.1)
    • C—CHEMISTRY; METALLURGY
    • C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12P—FERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P7/00—Preparation of oxygen-containing organic compounds
    • C12P7/24—Preparation of oxygen-containing organic compounds containing a carbonyl group
    • C12P7/26—Ketones
    • C12P7/38—Cyclopentanone- or cyclopentadione-containing products
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S435/00—Chemistry: molecular biology and microbiology
    • Y10S435/8215—Microorganisms
    • Y10S435/911—Microorganisms using fungi
    • Y10S435/913—Aspergillus
    • Y10S435/917—Aspergillus niger
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S435/00—Chemistry: molecular biology and microbiology
    • Y10S435/8215—Microorganisms
    • Y10S435/911—Microorganisms using fungi
    • Y10S435/94—Saccharomyces
    • Y10S435/942—Saccharomyces cerevisiae

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Microbiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biochemistry (AREA)
  • General Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Biotechnology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Analytical Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Biomedical Technology (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
FR7539824A 1974-12-26 1975-12-26 Cyclopentene-diols et leurs esters acyliques, utilisables pour la fabrication de medicaments, et preparation de ces composes Granted FR2295933A1 (fr)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
JP14826374A JPS5176484A (en) 1974-12-26 1974-12-26 Shikuropentenooru mataha sonojudotaino seizoho
JP14826674A JPS5176486A (en) 1974-12-26 1974-12-26 Shikuropentenooru mataha sono judotaino seizoho
JP2948675A JPS51106789A (en) 1975-03-13 1975-03-13 44 haidorokishishikuropento 22 en 11 onnoseizoho
JP4579375A JPS51121595A (en) 1975-04-17 1975-04-17 Method for preparing cyclopentenol derivatives
JP4652575A JPS51123889A (en) 1975-04-18 1975-04-18 Process for preparing optically active 1-cyclopentene-3, 5-diol mono a nd or di-acyl esters
JP4740875A JPS51123890A (en) 1975-04-21 1975-04-21 Process for preparing optically active 1-cyclopentene-3, 5-diol and or its derivatives

Publications (2)

Publication Number Publication Date
FR2295933A1 true FR2295933A1 (fr) 1976-07-23
FR2295933B1 FR2295933B1 (fr) 1979-10-12

Family

ID=27549460

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7539824A Granted FR2295933A1 (fr) 1974-12-26 1975-12-26 Cyclopentene-diols et leurs esters acyliques, utilisables pour la fabrication de medicaments, et preparation de ces composes

Country Status (8)

Country Link
US (1) US4008125A (fr)
CA (1) CA1074240A (fr)
CH (1) CH619982A5 (fr)
DE (1) DE2552871C3 (fr)
FR (1) FR2295933A1 (fr)
GB (1) GB1528382A (fr)
IT (1) IT1048795B (fr)
NL (1) NL7513394A (fr)

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0080827A2 (fr) * 1981-11-28 1983-06-08 Sumitomo Chemical Company, Limited Procédé de préparation biotechnologique de l'alcool (S)-(-)- alpha-cyano-3-phénoxybenzylique
EP0118163A1 (fr) * 1983-01-10 1984-09-12 Sumitomo Chemical Company, Limited Procédé de préparation biotechnologique de l'alcool alpha-cyano-3-phénoxybenzylique optiquement actif
EP0148272A1 (fr) * 1983-05-09 1985-07-17 Sumitomo Chemical Company, Limited Procede de preparation de composes d'alcool benzylique optiquement actifs
EP0167759A1 (fr) * 1984-06-01 1986-01-15 Bayer Ag Procédé pour la préparation d'ester (1S,4R)-4-hydroxy-2-cyclopentényl
EP0576834A2 (fr) * 1992-05-29 1994-01-05 Kureha Kagaku Kogyo Kabushiki Kaisha Procédé de production de dérivés d'un 1,2-diol optiquement active

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3305395A1 (de) * 1983-02-17 1984-08-23 Karl Dipl.-Ing. 6367 Karben Tesar Geraet zum auffinden von auf rollfilmen gespeichertem schriftgut
US5240835A (en) * 1989-10-10 1993-08-31 Genencor International, Inc. Methods for enzymatically preparing polymerizable monomers
US6448051B1 (en) * 2001-03-15 2002-09-10 Council Of Scientific And Industrial Research Process for the preparation of 4(R)-hydroxy cyclopent-2-en1(S)-acetate
ATE412061T1 (de) * 2002-12-13 2008-11-15 Archimica Gmbh Verfahren zur herstellung von (1s,4r)-(-)-4- hydroxycyclopent-2-enyl estern
DK2292743T3 (da) 2003-12-03 2013-11-25 Danisco Us Inc Perhydrolase
GT200500281A (es) * 2004-10-22 2006-04-24 Novartis Ag Compuestos organicos.
GB0500785D0 (en) * 2005-01-14 2005-02-23 Novartis Ag Organic compounds
WO2007133263A2 (fr) * 2005-12-09 2007-11-22 Genencor International, Inc. Acyle transférase utile pour la décontamination
US20080029130A1 (en) * 2006-03-02 2008-02-07 Concar Edward M Surface active bleach and dynamic pH
BRPI0709978A2 (pt) 2006-04-14 2011-08-02 Genencor Int tratamento em etapa única de produtos têxteis
GB0607944D0 (en) * 2006-04-21 2006-05-31 Novartis Ag Organic compounds
GB0607953D0 (en) * 2006-04-21 2006-05-31 Novartis Ag Organic compounds
AR060607A1 (es) 2006-04-21 2008-07-02 Novartis Ag Derivados de purina,composiciones farmaceuticas que los contienen, metodo de preparacion y usos en enfermedades obstructivas o inflamatorias de las vias respiratorias.
GB0607950D0 (en) * 2006-04-21 2006-05-31 Novartis Ag Organic compounds
EP1889846A1 (fr) 2006-07-13 2008-02-20 Novartis AG Dérivés de purine comme agonistes du recepteur A2a
EP1903044A1 (fr) * 2006-09-14 2008-03-26 Novartis AG Derivés de l'adénosine en tant qu' agonistes du récepteur A2A
MX2009004991A (es) * 2006-11-10 2009-05-20 Novartis Ag Derivados de monoacetato de ciclopenteno-diol.
KR102527797B1 (ko) 2012-12-21 2023-05-03 길리애드 사이언시즈, 인코포레이티드 폴리시클릭-카르바모일피리돈 화합물 및 그의 제약 용도
NO2865735T3 (fr) 2013-07-12 2018-07-21
CA2916993C (fr) 2013-07-12 2019-01-15 Gilead Sciences, Inc. Composes polycycliques-carbomoylpyridone et leur utilisation pharmaceutique
TW201613936A (en) 2014-06-20 2016-04-16 Gilead Sciences Inc Crystalline forms of(2R,5S,13aR)-8-hydroxy-7,9-dioxo-n-(2,4,6-trifluorobenzyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazepine-10-carboxamide
TWI744723B (zh) 2014-06-20 2021-11-01 美商基利科學股份有限公司 多環型胺甲醯基吡啶酮化合物之合成
NO2717902T3 (fr) 2014-06-20 2018-06-23

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3773622A (en) * 1972-09-29 1973-11-20 Wisconsin Alumni Res Found Method for preparing 2-substituted-4-hydroxy-cyclopentane-1,3-diones
JPS506779A (fr) * 1973-05-28 1975-01-23

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
NEANT *

Cited By (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0080827A2 (fr) * 1981-11-28 1983-06-08 Sumitomo Chemical Company, Limited Procédé de préparation biotechnologique de l'alcool (S)-(-)- alpha-cyano-3-phénoxybenzylique
EP0080827A3 (en) * 1981-11-28 1984-05-23 Sumitomo Chemical Company, Limited Method for biotechnologically preparing (s)-(-)-alpha-cyano-3-phenoxybenzyl alcohol
EP0118163A1 (fr) * 1983-01-10 1984-09-12 Sumitomo Chemical Company, Limited Procédé de préparation biotechnologique de l'alcool alpha-cyano-3-phénoxybenzylique optiquement actif
EP0148272A1 (fr) * 1983-05-09 1985-07-17 Sumitomo Chemical Company, Limited Procede de preparation de composes d'alcool benzylique optiquement actifs
EP0148272A4 (fr) * 1983-05-09 1987-02-03 Sumitomo Chemical Co Procede de preparation de composes d'alcool benzylique optiquement actifs.
EP0167759A1 (fr) * 1984-06-01 1986-01-15 Bayer Ag Procédé pour la préparation d'ester (1S,4R)-4-hydroxy-2-cyclopentényl
EP0576834A2 (fr) * 1992-05-29 1994-01-05 Kureha Kagaku Kogyo Kabushiki Kaisha Procédé de production de dérivés d'un 1,2-diol optiquement active
EP0576834A3 (fr) * 1992-05-29 1995-01-11 Kureha Chemical Ind Co Ltd Procédé de production de dérivés d'un 1,2-diol optiquement active.

Also Published As

Publication number Publication date
NL7513394A (nl) 1976-06-29
CH619982A5 (fr) 1980-10-31
CA1074240A (fr) 1980-03-25
FR2295933B1 (fr) 1979-10-12
DE2552871A1 (de) 1976-07-01
IT1048795B (it) 1980-12-20
GB1528382A (en) 1978-10-11
US4008125A (en) 1977-02-15
DE2552871C3 (de) 1979-07-05
DE2552871B2 (de) 1978-11-09

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Legal Events

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ST Notification of lapse