FR2281758A1 - 3-methyl-pyrazole-5-carboxylates, procede pour leur fabrication et preparations pharmaceutiques contenant ces composes - Google Patents

3-methyl-pyrazole-5-carboxylates, procede pour leur fabrication et preparations pharmaceutiques contenant ces composes

Info

Publication number
FR2281758A1
FR2281758A1 FR7525251A FR7525251A FR2281758A1 FR 2281758 A1 FR2281758 A1 FR 2281758A1 FR 7525251 A FR7525251 A FR 7525251A FR 7525251 A FR7525251 A FR 7525251A FR 2281758 A1 FR2281758 A1 FR 2281758A1
Authority
FR
France
Prior art keywords
carboxylates
pyrazole
methyl
compounds
manufacture
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7525251A
Other languages
English (en)
Other versions
FR2281758B1 (fr
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
JOHANN A WULFING
Original Assignee
JOHANN A WULFING
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by JOHANN A WULFING filed Critical JOHANN A WULFING
Publication of FR2281758A1 publication Critical patent/FR2281758A1/fr
Application granted granted Critical
Publication of FR2281758B1 publication Critical patent/FR2281758B1/fr
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/02Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
    • C07D473/06Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
    • C07D473/08Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3 with methyl radicals in positions 1 and 3, e.g. theophylline
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FR7525251A 1974-08-14 1975-08-13 3-methyl-pyrazole-5-carboxylates, procede pour leur fabrication et preparations pharmaceutiques contenant ces composes Granted FR2281758A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2439137A DE2439137A1 (de) 1974-08-14 1974-08-14 3-methyl-pyrazol-5-carboxylate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneipraeparate

Publications (2)

Publication Number Publication Date
FR2281758A1 true FR2281758A1 (fr) 1976-03-12
FR2281758B1 FR2281758B1 (fr) 1978-09-08

Family

ID=5923236

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7525251A Granted FR2281758A1 (fr) 1974-08-14 1975-08-13 3-methyl-pyrazole-5-carboxylates, procede pour leur fabrication et preparations pharmaceutiques contenant ces composes

Country Status (12)

Country Link
US (1) US3980646A (fr)
JP (1) JPS51104019A (fr)
AR (1) AR211100A1 (fr)
AT (1) AT338287B (fr)
BE (1) BE832389A (fr)
CA (1) CA1062258A (fr)
DE (1) DE2439137A1 (fr)
FI (1) FI752070A (fr)
FR (1) FR2281758A1 (fr)
GB (1) GB1481147A (fr)
NL (1) NL7509706A (fr)
SE (1) SE7509123L (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2373283A1 (fr) * 1976-12-10 1978-07-07 Wuelfing Johann A Composes derives de l'isoxazole, utilisables comme medicament

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4092417A (en) * 1976-12-08 1978-05-30 Johann A. Wulfing Theophylline salts of 5-methylisoxazole-3-carboxylic acid
US20060167270A1 (en) * 2002-10-10 2006-07-27 Arena Pharmaceuticals Inc. 5-substituted 2h-pyrazone-3-carbixylic acid derivatives as antilipolytic agents for the treatment of metabolic-related disorders such as dyslipidemia
EP1633351A1 (fr) * 2003-06-13 2006-03-15 Arena Pharmaceuticals, Inc. Derives d'acide 2h-pyrazol-3- carboxylique substitues en 5 utilises comme agonistes du recepteur de l'acide nicotinique rup25 pour le traitement des dyslipidemies et des pathologies apparentees
JP4348440B2 (ja) 2005-09-01 2009-10-21 有洙 安 透過性補強材と発泡体を利用したベッド用マットレス及びその製造方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2924598A (en) * 1960-02-09 Methods of preparing same
DE1089763B (de) * 1957-10-26 1960-09-29 Wuelfing J A Fa Verfahren zur Herstellung des 7-[ª‰-Oxy-ª†-(methyl-ª‰-oxyaethylamino)-propyl]-theophyllin-nikotinats
DE1102750B (de) * 1958-07-17 1961-03-23 Wuelfing J A Fa Verfahren zur Herstellung eines Salzes von Theophyllinbasen
US3728346A (en) * 1971-07-16 1973-04-17 Degussa Hydroxyphenylhydroxyalkylaminoalkyltheophyllines
AT313916B (de) * 1971-10-28 1974-03-11 Degussa Verfahren zur Herstellung von neuen basisch substituierten Theophyllinen und deren Säureadditionssalzen

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2373283A1 (fr) * 1976-12-10 1978-07-07 Wuelfing Johann A Composes derives de l'isoxazole, utilisables comme medicament

Also Published As

Publication number Publication date
CA1062258A (fr) 1979-09-11
GB1481147A (en) 1977-07-27
AT338287B (de) 1977-08-10
US3980646A (en) 1976-09-14
BE832389A (fr) 1976-02-13
SE7509123L (sv) 1976-02-16
FI752070A (fr) 1976-02-15
AR211100A1 (es) 1977-10-31
NL7509706A (nl) 1976-02-17
DE2439137A1 (de) 1976-08-12
FR2281758B1 (fr) 1978-09-08
ATA618075A (de) 1976-12-15
JPS51104019A (en) 1976-09-14

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Legal Events

Date Code Title Description
ST Notification of lapse