FR2252088A1 - Antibacterial 1,2,4-triazin-5-ones - of varying activity, some with tranquillizing activity - Google Patents

Antibacterial 1,2,4-triazin-5-ones - of varying activity, some with tranquillizing activity

Info

Publication number
FR2252088A1
FR2252088A1 FR7341846A FR7341846A FR2252088A1 FR 2252088 A1 FR2252088 A1 FR 2252088A1 FR 7341846 A FR7341846 A FR 7341846A FR 7341846 A FR7341846 A FR 7341846A FR 2252088 A1 FR2252088 A1 FR 2252088A1
Authority
FR
France
Prior art keywords
substd
opt
activity
atom
antibacterial
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7341846A
Other languages
French (fr)
Other versions
FR2252088B1 (en
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bpifrance Financement SA
Original Assignee
Agence National de Valorisation de la Recherche ANVAR
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Agence National de Valorisation de la Recherche ANVAR filed Critical Agence National de Valorisation de la Recherche ANVAR
Priority to FR7341846A priority Critical patent/FR2252088A1/en
Publication of FR2252088A1 publication Critical patent/FR2252088A1/en
Application granted granted Critical
Publication of FR2252088B1 publication Critical patent/FR2252088B1/fr
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D253/00—Heterocyclic compounds containing six-membered rings having three nitrogen atoms as the only ring hetero atoms, not provided for by group C07D251/00
    • C07D253/02—Heterocyclic compounds containing six-membered rings having three nitrogen atoms as the only ring hetero atoms, not provided for by group C07D251/00 not condensed with other rings
    • C07D253/06—1,2,4-Triazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D253/00—Heterocyclic compounds containing six-membered rings having three nitrogen atoms as the only ring hetero atoms, not provided for by group C07D251/00
    • C07D253/02—Heterocyclic compounds containing six-membered rings having three nitrogen atoms as the only ring hetero atoms, not provided for by group C07D251/00 not condensed with other rings
    • C07D253/06—1,2,4-Triazines
    • C07D253/065—1,2,4-Triazines having three double bonds between ring members or between ring members and non-ring members
    • C07D253/07—1,2,4-Triazines having three double bonds between ring members or between ring members and non-ring members with hetero atoms, or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D253/075—Two hetero atoms, in positions 3 and 5

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

of formula (I) and their tautomers (where A is O, S; when A is S, R1 and the H atom on N' are replaced by a second bond feature between N1 and C6; when a is O, R1 is H, opt. substd. phenyl 1-16C alkyl; R2 is opt. substd. phenyl 2-16C alkyl; when A is O, only one of R1, R2 is phenyl; R3 is H, opt. substd. benzyl, 1-16C opt. unsatd. aliphatic gp; when A is S, R2 is opt. substd. phenyl, 2-16C alkyl and the C atom of the chain next to the C6 atom of the triazine is substd. by -CO2H, an amide- CN or an ester; when A is S, and when R3 is opt. substd. benzyl, 1-16C opt. unsatd. aliphatic gp. the triazinone may be an isomer of I in which the S atom on C3 is substd. by R3 instead of the N4 atom) are antibacterial agents, but those with R1 = H, R2 = Me, R3 = H, A = O and are tranquillisers with no antibacterial activity.
FR7341846A 1973-11-23 1973-11-23 Antibacterial 1,2,4-triazin-5-ones - of varying activity, some with tranquillizing activity Granted FR2252088A1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FR7341846A FR2252088A1 (en) 1973-11-23 1973-11-23 Antibacterial 1,2,4-triazin-5-ones - of varying activity, some with tranquillizing activity

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7341846A FR2252088A1 (en) 1973-11-23 1973-11-23 Antibacterial 1,2,4-triazin-5-ones - of varying activity, some with tranquillizing activity

Publications (2)

Publication Number Publication Date
FR2252088A1 true FR2252088A1 (en) 1975-06-20
FR2252088B1 FR2252088B1 (en) 1977-04-22

Family

ID=9128189

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7341846A Granted FR2252088A1 (en) 1973-11-23 1973-11-23 Antibacterial 1,2,4-triazin-5-ones - of varying activity, some with tranquillizing activity

Country Status (1)

Country Link
FR (1) FR2252088A1 (en)

Also Published As

Publication number Publication date
FR2252088B1 (en) 1977-04-22

Similar Documents

Publication Publication Date Title
ES441673A1 (en) Biguanide salts
ATE269290T1 (en) BENZOYL DERIVATIVES
GB1457129A (en) Herbicidal antidote compositions with substituted oxazolidines and thiazolidines
IT1250749B (en) HETEROCYCLIC COMPOUNDS ACTIVATED IN II ANTAGONIST
ES428101A1 (en) 1-(1,2,4-Triazolyl-1{40 )-2-phenoxy-4,4-dimethyl-pentan-3-ones
ES422906A1 (en) Derivatives of 2-aminoindane, the preparation and use thereof
FR2252088A1 (en) Antibacterial 1,2,4-triazin-5-ones - of varying activity, some with tranquillizing activity
ES422386A1 (en) O-ethyl-S-n-propyl-0-2-cyanovinyl-thionothiol-phosphoric acid esters
GB1049064A (en) Preparation of aminopropylidenedibenzocycloheptenes
ES396035A1 (en) Triazole-coumarins
FR2071171A6 (en) 1,1-diphenyl-azaborolidines - with insecticidal acaricidal - herbicidal and fungicidal activity
BE816076A (en) N-cyclohexyl-N'-substd-phenyl-benzamides - having anti-inflammatory and analgesic activity with low toxicity
ES430676A1 (en) 2-Substituted -1,2,4-thiadiazolo-(2,3-a)benzimidazoles and process for their preparation
FR2078729A5 (en) Herbicidal 2,4-bis-trifluoromethyl-6-nitro-anilines
ES8207542A1 (en) Total synthesis of 1RS,4SR,5RS-4-(4,8-dimethyl-5-hydroxy-7-nonen-1-yl)-4-methyl-3,8-dioxabicyclo(3.2.1)octane-1-acetic acid and related compounds.
FR2400024A1 (en) NEW PENICILLIN DERIVATIVES
ES448065A1 (en) Nitropyrazole compounds and anti-microbial compositions
FR2085645A1 (en) 1-phenyl-2,3-benzodiazepin-4-ones - as tranquillizers
ES424835A1 (en) Alkyloxalyl amino-s-triazines
FR2191845A1 (en) Urea-triazine herbicidal compsn - showing synergistic effect for pre-emergence treatment of cereal crops
FR2201885A1 (en) 4-Aryl carbonyl methyl pyrimidine oxime carbamates - prepd. by treatment of the oxime with an isocyanate, used as sedatives, analgesics, vasodilators, diuretics
FR2070103A1 (en) Antiphlogistic 1- (hydroxy amido or amino) - acenaphthenes
FR2168185A1 (en) Dichloropyridyl dialkyl (thio) phosphates - eg insecticides
FR2242393A1 (en) N-(butyro or valerolactone)uracils prepn. - by reacting 2,4-bis(trimethylsilyl)uracil with alphabromobutyro or valerolactone
FR2021260A1 (en) Photographic fixer-developer with reduced fogging - tendency

Legal Events

Date Code Title Description
ST Notification of lapse