FR2240225A1 - 3-Substd. cepham-4-carboxylic acids prodn. - by removal of carboxy protecting gps of corresp. protected cpd - Google Patents
3-Substd. cepham-4-carboxylic acids prodn. - by removal of carboxy protecting gps of corresp. protected cpdInfo
- Publication number
- FR2240225A1 FR2240225A1 FR7423877A FR7423877A FR2240225A1 FR 2240225 A1 FR2240225 A1 FR 2240225A1 FR 7423877 A FR7423877 A FR 7423877A FR 7423877 A FR7423877 A FR 7423877A FR 2240225 A1 FR2240225 A1 FR 2240225A1
- Authority
- FR
- France
- Prior art keywords
- cepham
- substd
- corresp
- cpd
- protected
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 title 1
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 2
- XBXGCAKAFVASIM-OPAIIUCXSA-N (6r)-3-anilino-3-methyl-8-oxo-7-[(2-phenoxyacetyl)amino]-5-thia-1-azabicyclo[4.2.0]octane-2-carboxylic acid Chemical compound C1([C@H]2SCC(C(N2C1=O)C(O)=O)(C)NC=1C=CC=CC=1)NC(=O)COC1=CC=CC=C1 XBXGCAKAFVASIM-OPAIIUCXSA-N 0.000 abstract 1
- ZDWICQDEBDSHSD-VTUJEPCUSA-N (6r)-3-bromo-3-methyl-8-oxo-7-[(2-phenoxyacetyl)amino]-5-thia-1-azabicyclo[4.2.0]octane-2-carboxylic acid Chemical compound C1([C@H]2SCC(C(N2C1=O)C(O)=O)(Br)C)NC(=O)COC1=CC=CC=C1 ZDWICQDEBDSHSD-VTUJEPCUSA-N 0.000 abstract 1
- RGUXHDLRDQTJBW-YTOPNPFISA-N 1-cyclopropylethyl (6r)-3-anilino-3-methyl-8-oxo-7-[(2-phenoxyacetyl)amino]-5-thia-1-azabicyclo[4.2.0]octane-2-carboxylate Chemical compound S([C@H]1N(C(C1NC(=O)COC=1C=CC=CC=1)=O)C1C(=O)OC(C)C2CC2)CC1(C)NC1=CC=CC=C1 RGUXHDLRDQTJBW-YTOPNPFISA-N 0.000 abstract 1
- DTQVDTLACAAQTR-UHFFFAOYSA-N Trifluoroacetic acid Chemical compound OC(=O)C(F)(F)F DTQVDTLACAAQTR-UHFFFAOYSA-N 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 238000001816 cooling Methods 0.000 abstract 1
- 125000001475 halogen functional group Chemical group 0.000 abstract 1
- 230000000269 nucleophilic effect Effects 0.000 abstract 1
- 238000003756 stirring Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
- C07D205/09—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a sulfur atom directly attached in position 4
- C07D205/095—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a sulfur atom directly attached in position 4 and with a nitrogen atom directly attached in position 3
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Cephalosporin Compounds (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP11738472A JPS5550955B2 (enrdf_load_stackoverflow) | 1972-11-22 | 1972-11-22 | |
| JP12557372A JPS5531791B2 (enrdf_load_stackoverflow) | 1972-12-13 | 1972-12-13 | |
| JP47128658A JPS5929597B2 (ja) | 1972-12-20 | 1972-12-20 | ２−置換アルキル−２−アルキルペナム−３−カルボン酸類の製造法 |
| JP12890272A JPS5641634B2 (enrdf_load_stackoverflow) | 1972-12-21 | 1972-12-21 | |
| JP731201A JPS5946950B2 (ja) | 1972-12-23 | 1972-12-23 | ３−置換セフアム−４−カルボン酸類を製造する方法 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| FR2240225A1 true FR2240225A1 (en) | 1975-03-07 |
| FR2240225B1 FR2240225B1 (enrdf_load_stackoverflow) | 1979-01-26 |
Family
ID=27518073
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FR7423877A Granted FR2240225A1 (en) | 1972-11-22 | 1974-07-09 | 3-Substd. cepham-4-carboxylic acids prodn. - by removal of carboxy protecting gps of corresp. protected cpd |
Country Status (1)
| Country | Link |
|---|---|
| FR (1) | FR2240225A1 (enrdf_load_stackoverflow) |
-
1974
- 1974-07-09 FR FR7423877A patent/FR2240225A1/fr active Granted
Also Published As
| Publication number | Publication date |
|---|---|
| FR2240225B1 (enrdf_load_stackoverflow) | 1979-01-26 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| ST | Notification of lapse |