FR2197573A1 - 7-substd-phenylacetamido-cephalosporin derivs - - antibiotics active against streptococci and staphylococci - Google Patents

7-substd-phenylacetamido-cephalosporin derivs - - antibiotics active against streptococci and staphylococci

Info

Publication number
FR2197573A1
FR2197573A1 FR7231699A FR7231699A FR2197573A1 FR 2197573 A1 FR2197573 A1 FR 2197573A1 FR 7231699 A FR7231699 A FR 7231699A FR 7231699 A FR7231699 A FR 7231699A FR 2197573 A1 FR2197573 A1 FR 2197573A1
Authority
FR
France
Prior art keywords
substd
opt
phenylacetamido
staphylococci
active against
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7231699A
Other languages
French (fr)
Other versions
FR2197573B1 (en
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Aventis France
Original Assignee
Roussel Uclaf SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to BE793448D priority Critical patent/BE793448A/en
Priority to FR7231699A priority patent/FR2197573A1/en
Application filed by Roussel Uclaf SA filed Critical Roussel Uclaf SA
Priority to CH1867372A priority patent/CH563398A5/xx
Priority to CH1371974A priority patent/CH568328A5/xx
Priority to CH466575A priority patent/CH577519A5/xx
Priority to CH466675A priority patent/CH577516A5/xx
Priority to IL4839272A priority patent/IL48392A/en
Priority to IL41196A priority patent/IL41196A/en
Priority to PL1972159834A priority patent/PL94240B1/en
Priority to JP734409A priority patent/JPS599558B2/en
Priority to DD168202*A priority patent/DD106046A5/xx
Priority to SE7217182A priority patent/SE415564B/en
Priority to GB2357675A priority patent/GB1423743A/en
Priority to GB2611875A priority patent/GB1423742A/en
Priority to GB11473A priority patent/GB1423741A/en
Priority to US05/320,493 priority patent/US3962223A/en
Priority to DE2300009A priority patent/DE2300009C2/en
Priority to AT573*BA priority patent/AT324554B/en
Priority to CS7346A priority patent/CS201524B2/en
Priority to NL7300031A priority patent/NL7300031A/xx
Publication of FR2197573A1 publication Critical patent/FR2197573A1/en
Priority to SU742032631A priority patent/SU976853A3/en
Priority to US05/538,189 priority patent/US4016158A/en
Priority to IL48300A priority patent/IL48300A0/en
Application granted granted Critical
Publication of FR2197573B1 publication Critical patent/FR2197573B1/fr
Priority to IL48392A priority patent/IL48392A0/en
Priority to SE7606178A priority patent/SE417824B/en
Priority to SE7606177A priority patent/SE426816B/en
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/44—Iso-indoles; Hydrogenated iso-indoles
    • C07D209/48—Iso-indoles; Hydrogenated iso-indoles with oxygen atoms in positions 1 and 3, e.g. phthalimide
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J23/00—Catalysts comprising metals or metal oxides or hydroxides, not provided for in group B01J21/00
    • B01J23/38—Catalysts comprising metals or metal oxides or hydroxides, not provided for in group B01J21/00 of noble metals
    • B01J23/40—Catalysts comprising metals or metal oxides or hydroxides, not provided for in group B01J21/00 of noble metals of the platinum group metals
    • B01J23/44—Palladium

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Materials Engineering (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)

Abstract

Title cpds are of formula: (where R1 is phenyl opt. substd. by >=1 halogen atoms or 1 NO2 gp. or R1 is a heterocyclic radical, Y' is NHCOOR2, where R2 is 1-5C opt. branched alkyl, or Y' is Y", where Y" is H or OH, R2 is H or R2', where R2' is an ester gp. easily removable by acid hydrolysis or hydrogenolysis and A1 is 2-5C opt. branched alkyl or 3-7C cycloalkyl opt. contg. O or S as a heteroatom) together with their addn salts with mineral or org. acids, or bases. The cpds may be in the racemic form or as optically active isomers and may be in the cis or trans form, or as mixt. of these isomers.
FR7231699A 1971-12-31 1972-09-07 7-substd-phenylacetamido-cephalosporin derivs - - antibiotics active against streptococci and staphylococci Granted FR2197573A1 (en)

Priority Applications (26)

Application Number Priority Date Filing Date Title
BE793448D BE793448A (en) 1971-12-31 PROCESS FOR PREPARATION OF NEW CEPHALOSPORIN DERIVATIVES AND PRODUCTS OBTAINED
FR7231699A FR2197573A1 (en) 1972-09-07 1972-09-07 7-substd-phenylacetamido-cephalosporin derivs - - antibiotics active against streptococci and staphylococci
CH1371974A CH568328A5 (en) 1971-12-31 1972-12-21
CH466575A CH577519A5 (en) 1971-12-31 1972-12-21
CH1867372A CH563398A5 (en) 1971-12-31 1972-12-21
CH466675A CH577516A5 (en) 1971-12-31 1972-12-21
IL4839272A IL48392A (en) 1971-12-31 1972-12-27 7-amino-3-alkyl-(or 3-cycloalkyl) ceph-3-eme-4-carboxylic acids and esters of these
IL41196A IL41196A (en) 1971-12-31 1972-12-27 Process for the preparation of 3-desacetoxymethyl-3-alkyl(or cycloalkyl) cephalosporins and some such compounds
PL1972159834A PL94240B1 (en) 1971-12-31 1972-12-28 Substituted cephene-4-carboxylates and their method of preparation[us3962223a]
DD168202*A DD106046A5 (en) 1971-12-31 1972-12-29
SE7217182A SE415564B (en) 1971-12-31 1972-12-29 SET TO MAKE NEW CEPHALOSPORINE DERIVATIVES
JP734409A JPS599558B2 (en) 1971-12-31 1972-12-29 Method for producing novel cephalosporin derivatives
GB2357675A GB1423743A (en) 1971-12-31 1973-01-01 Derivatives of cephalosporin processes for their preparation and compositions incorporating them
GB2611875A GB1423742A (en) 1971-12-31 1973-01-01 2-oxobut-3-enoates
GB11473A GB1423741A (en) 1971-12-31 1973-01-01 Derivatives of cephalosporin processes for their preparation and compositions incorporating them
US05/320,493 US3962223A (en) 1971-12-31 1973-01-02 Substituted cephene-4-carboxylates and their method of preparation
DE2300009A DE2300009C2 (en) 1971-12-31 1973-01-02 Process for the preparation of 7-aminocephalosporanic acid derivatives
AT573*BA AT324554B (en) 1971-12-31 1973-01-02 PROCESS FOR MANUFACTURING NEW CEPHALOSPORIN DERIVATIVES
CS7346A CS201524B2 (en) 1971-12-31 1973-01-02 Process for preparing new derivatives of 3-desacetoxycephalosporic acid
NL7300031A NL7300031A (en) 1971-12-31 1973-01-02
SU742032631A SU976853A3 (en) 1971-12-31 1974-06-13 Method of producing derivatives of cephalosporine or their salts in form of mixture of cys- or trans-isomers or one of these isomers
US05/538,189 US4016158A (en) 1971-12-31 1975-01-02 Cephalosporin derivatives
IL48300A IL48300A0 (en) 1971-12-31 1975-10-15 Process for preparing beta-methylene alpha-oxo carboxylic acid esters
IL48392A IL48392A0 (en) 1971-12-31 1975-10-31 7-amino-3-alkyl-(or cycloalkyl)ceph-3-em carboxylic acids and esters of these
SE7606178A SE417824B (en) 1971-12-31 1976-06-01 7-AMINOCEPHALOSPORANIC ACID DERIVATIVES FOR USE AS INTERMEDIATE FOR THE PRODUCTION OF CEPHALOSPORIN DERIVATIVES
SE7606177A SE426816B (en) 1971-12-31 1976-06-01 SET TO PREPARE BETA-METHYLENE-ALFA-OXO-CARBOXYLIC ACID ESTERS

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7231699A FR2197573A1 (en) 1972-09-07 1972-09-07 7-substd-phenylacetamido-cephalosporin derivs - - antibiotics active against streptococci and staphylococci

Publications (2)

Publication Number Publication Date
FR2197573A1 true FR2197573A1 (en) 1974-03-29
FR2197573B1 FR2197573B1 (en) 1975-10-17

Family

ID=9103962

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7231699A Granted FR2197573A1 (en) 1971-12-31 1972-09-07 7-substd-phenylacetamido-cephalosporin derivs - - antibiotics active against streptococci and staphylococci

Country Status (1)

Country Link
FR (1) FR2197573A1 (en)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1992001696A1 (en) * 1990-07-24 1992-02-06 Beecham Group Plc Cephalosporins and homologues, preparations and pharmaceutical compositions

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2102081A1 (en) * 1970-08-06 1972-04-07 Glaxo Lab Ltd
FR2102080A1 (en) * 1970-08-06 1972-04-07 Glaxo Lab Ltd

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2102081A1 (en) * 1970-08-06 1972-04-07 Glaxo Lab Ltd
FR2102080A1 (en) * 1970-08-06 1972-04-07 Glaxo Lab Ltd

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1992001696A1 (en) * 1990-07-24 1992-02-06 Beecham Group Plc Cephalosporins and homologues, preparations and pharmaceutical compositions

Also Published As

Publication number Publication date
FR2197573B1 (en) 1975-10-17

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Legal Events

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