FR2034605A1 - - Google Patents

Info

Publication number
FR2034605A1
FR2034605A1 FR7005100A FR7005100A FR2034605A1 FR 2034605 A1 FR2034605 A1 FR 2034605A1 FR 7005100 A FR7005100 A FR 7005100A FR 7005100 A FR7005100 A FR 7005100A FR 2034605 A1 FR2034605 A1 FR 2034605A1
Authority
FR
France
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7005100A
Other languages
French (fr)
Other versions
FR2034605B1 (el
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SOGERAS
Original Assignee
SOGERAS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by SOGERAS filed Critical SOGERAS
Publication of FR2034605A1 publication Critical patent/FR2034605A1/fr
Application granted granted Critical
Publication of FR2034605B1 publication Critical patent/FR2034605B1/fr
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FR7005100A 1969-03-03 1970-02-13 Expired FR2034605B1 (el)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB1124969 1969-03-03

Publications (2)

Publication Number Publication Date
FR2034605A1 true FR2034605A1 (el) 1970-12-11
FR2034605B1 FR2034605B1 (el) 1974-01-11

Family

ID=9982760

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7005100A Expired FR2034605B1 (el) 1969-03-03 1970-02-13

Country Status (9)

Country Link
AT (1) AT294114B (el)
BE (1) BE746034A (el)
CA (1) CA933925A (el)
CH (1) CH502378A (el)
DE (1) DE2009555A1 (el)
FR (1) FR2034605B1 (el)
GB (1) GB1250534A (el)
NL (1) NL7003014A (el)
SE (1) SE377803B (el)

Cited By (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2318638A2 (fr) * 1975-07-25 1977-02-18 Sogeras Nouveaux derives de la phenothiazine et procede pour leur preparation
FR2497806A1 (fr) * 1981-01-13 1982-07-16 Pharmindustrie Nouveau procede de preparation du n,n-dimethyl (aza-1 bicyclo (2,2,2) octyl-3)-10 10h-phenothiazinesulfonamide-2
FR2503165A1 (fr) * 1981-04-03 1982-10-08 Pharmindustrie Nouveaux derives de n,n-dimethyl(aza-1 bicyclo(2,2,2)octyl-3)-10 10h phenothiazinesulfonamide-2, procede pour leur preparation et utilisation comme medicaments
FR2509307A1 (fr) * 1981-07-10 1983-01-14 Pharmindustrie (aza-1 bicyclo-(2,2,2) octyl-3)-10 10h phenothiazine-sulfonamide-2, ses derives, procede pour leur preparation et leur utilisation comme medicaments
FR2522660A1 (fr) * 1982-03-05 1983-09-09 Pharmuka Lab Isomere levogyre de la mequitazine, son procede de preparation et medicaments le contenant
EP0093643A1 (fr) * 1982-05-04 1983-11-09 Pharmuka Laboratoires Isomères dextrogyres de dérivés de l'aza-1 bicyclo (2,2,2)octane, leur procédé de préparation et médicaments les contenant
FR2531955A1 (fr) * 1982-08-17 1984-02-24 Pharmuka Lab Nouveau procede de preparation de derives de la quinuclidine substitues en position 3
FR2772029A1 (fr) * 1997-12-08 1999-06-11 Pf Medicament Procede de preparation de la mequitazine et nouvel intermediaire de synthese
US7749982B2 (en) 2004-10-21 2010-07-06 Pierre Fabre Medicament Complex containing mequitazine, a cyclodextrin and an interaction agent
US8158784B2 (en) 2007-01-18 2012-04-17 Pierre Fabre Medicament Quinuclidine derivative useful in the preparation of mequitazine

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2117750A1 (en) * 1970-12-15 1972-07-28 Sogeras 10-(3-quinuclidinylmethyl)phenothiazine 5-oxide and 5,5 - -dioxide - with antihistamine,antidepressant and tranquillizing activ
IT1173445B (it) * 1984-03-16 1987-06-24 Guidotti & C Spa Labor Agenti ad attivita' antibroncospastica e composizioni farmaceutiche che li contengono
GB8510680D0 (en) * 1985-04-26 1985-06-05 Smith Kline French Lab Pyridine derivatives
GB9201751D0 (en) * 1992-01-28 1992-03-11 Smithkline Beecham Plc Compounds
CA2530444C (en) 2003-06-27 2012-03-13 Janssen Pharmaceutica, N.V. Tricyclic .delta. opioid modulators
AU2005335481A1 (en) 2004-08-05 2007-04-19 Janssen Pharmaceutica N.V. Tricyclic delta- opioid modulators
KR20070092293A (ko) 2004-12-22 2007-09-12 얀센 파마슈티카 엔.브이. 트리사이클릭 δ-오피오이드 모듈레이터
BRPI0519201A2 (pt) 2004-12-22 2008-12-30 Janssen Pharmaceutica Nv moduladores de delta-opiàide tricÍclico
EP1846400A2 (en) 2005-01-06 2007-10-24 Janssen Pharmaceutica N.V. Tricyclic delta-opioid modulators
WO2006138528A2 (en) 2005-06-16 2006-12-28 Janssen Pharmaceutica N.V Tricyclic opioid modulators

Cited By (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2318638A2 (fr) * 1975-07-25 1977-02-18 Sogeras Nouveaux derives de la phenothiazine et procede pour leur preparation
FR2497806A1 (fr) * 1981-01-13 1982-07-16 Pharmindustrie Nouveau procede de preparation du n,n-dimethyl (aza-1 bicyclo (2,2,2) octyl-3)-10 10h-phenothiazinesulfonamide-2
EP0056201A1 (fr) * 1981-01-13 1982-07-21 Pharmuka Laboratoires Nouveau procédé de préparation du N,N-diméthyl aza-1 bicyclo 2,2,2 octyl-3 -10 10H-phénothiazinesulfonamide-2
FR2503165A1 (fr) * 1981-04-03 1982-10-08 Pharmindustrie Nouveaux derives de n,n-dimethyl(aza-1 bicyclo(2,2,2)octyl-3)-10 10h phenothiazinesulfonamide-2, procede pour leur preparation et utilisation comme medicaments
US4451461A (en) * 1981-07-10 1984-05-29 Pharmindustrie 10-(1-Aza-[2,2,2)-bicyclo-3-octyl]-10H-2-phenothiazinesulfonamide and derivatives thereof
EP0070753A1 (fr) * 1981-07-10 1983-01-26 Pharmuka Laboratoires (Aza-1 bicyclo-(2,2,2) octyl-3) -10 10H phénothiazine-sulfonamide-2 et dérivés
FR2509307A1 (fr) * 1981-07-10 1983-01-14 Pharmindustrie (aza-1 bicyclo-(2,2,2) octyl-3)-10 10h phenothiazine-sulfonamide-2, ses derives, procede pour leur preparation et leur utilisation comme medicaments
FR2522660A1 (fr) * 1982-03-05 1983-09-09 Pharmuka Lab Isomere levogyre de la mequitazine, son procede de preparation et medicaments le contenant
EP0089860A1 (fr) * 1982-03-05 1983-09-28 Pharmuka Laboratoires Isomère lévogyre de la méquitazine, son procédé de préparation et médicaments le contenant
EP0093643A1 (fr) * 1982-05-04 1983-11-09 Pharmuka Laboratoires Isomères dextrogyres de dérivés de l'aza-1 bicyclo (2,2,2)octane, leur procédé de préparation et médicaments les contenant
FR2526433A1 (fr) * 1982-05-04 1983-11-10 Pharmuka Lab Isomeres dextrogyres de derives de l'aza-1 bicyclo (2,2,2) octane, leur procede de preparation et medicaments les contenant
EP0102283A1 (fr) * 1982-08-17 1984-03-07 Pharmuka Laboratoires Nouveau procédé de préparation de dérivés de la quinuclidine substitués en position 3
FR2531955A1 (fr) * 1982-08-17 1984-02-24 Pharmuka Lab Nouveau procede de preparation de derives de la quinuclidine substitues en position 3
FR2772029A1 (fr) * 1997-12-08 1999-06-11 Pf Medicament Procede de preparation de la mequitazine et nouvel intermediaire de synthese
WO1999029692A1 (fr) * 1997-12-08 1999-06-17 Pierre Fabre Medicament Procede de preparation de la mequitazine et nouvel intermediaire de synthese
US7749982B2 (en) 2004-10-21 2010-07-06 Pierre Fabre Medicament Complex containing mequitazine, a cyclodextrin and an interaction agent
US8158784B2 (en) 2007-01-18 2012-04-17 Pierre Fabre Medicament Quinuclidine derivative useful in the preparation of mequitazine
US8304545B2 (en) 2007-01-18 2012-11-06 Pierre Fabre Medicament Quinuclidine derivative useful in the preparation of mequitazine

Also Published As

Publication number Publication date
CH502378A (fr) 1971-01-31
NL7003014A (el) 1970-09-07
DE2009555A1 (de) 1970-10-08
BE746034A (fr) 1970-07-31
SE377803B (el) 1975-07-28
AT294114B (de) 1971-11-10
GB1250534A (el) 1971-10-20
FR2034605B1 (el) 1974-01-11
CA933925A (en) 1973-09-18

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Legal Events

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