FI960940A - Alkoxy-substituted beta-carbolines with effect on AMPA receptor - Google Patents
Alkoxy-substituted beta-carbolines with effect on AMPA receptor Download PDFInfo
- Publication number
- FI960940A FI960940A FI960940A FI960940A FI960940A FI 960940 A FI960940 A FI 960940A FI 960940 A FI960940 A FI 960940A FI 960940 A FI960940 A FI 960940A FI 960940 A FI960940 A FI 960940A
- Authority
- FI
- Finland
- Prior art keywords
- carbolines
- alkoxy
- effect
- ampa receptor
- substituted beta
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE4330175A DE4330175A1 (en) | 1993-08-31 | 1993-08-31 | Alkoxy substituted beta carbolines |
PCT/DE1994/001009 WO1995006647A1 (en) | 1993-08-31 | 1994-08-29 | ALKOXY-SUBSTITUTED β-CARBOLINES ACTING ON THE AMPA-RECEPTOR |
Publications (2)
Publication Number | Publication Date |
---|---|
FI960940A true FI960940A (en) | 1996-02-28 |
FI960940A0 FI960940A0 (en) | 1996-02-28 |
Family
ID=6497015
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FI960940A FI960940A0 (en) | 1993-08-31 | 1996-02-28 | Alkoxy-substituted beta-carbolines acting on the AMPA receptor |
Country Status (17)
Country | Link |
---|---|
EP (1) | EP0716657A1 (en) |
JP (1) | JPH09501938A (en) |
KR (1) | KR960704888A (en) |
CN (1) | CN1129938A (en) |
AU (1) | AU7530394A (en) |
CA (1) | CA2170615A1 (en) |
CZ (1) | CZ50596A3 (en) |
DE (1) | DE4330175A1 (en) |
FI (1) | FI960940A0 (en) |
HU (1) | HUT73845A (en) |
IL (1) | IL110745A0 (en) |
NO (1) | NO960812L (en) |
NZ (1) | NZ271615A (en) |
PL (1) | PL313230A1 (en) |
SK (1) | SK23896A3 (en) |
WO (1) | WO1995006647A1 (en) |
ZA (1) | ZA946670B (en) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MY125942A (en) | 1999-09-07 | 2006-09-29 | Upjohn Co | Aminoalkoxy carbazoles for the treatment of cns diseases |
CN111093662B (en) | 2017-06-20 | 2023-10-03 | 安布里亚制药公司 | Compositions and methods for improving cardiac metabolic efficiency |
US11780811B2 (en) | 2020-06-30 | 2023-10-10 | Imbria Pharmaceuticals, Inc. | Methods of synthesizing 2-[4-[(2,3,4-trimethoxyphenyl)methyl]piperazin-1-yl]ethyl pyridine-3-carboxylate |
US11530184B2 (en) | 2020-06-30 | 2022-12-20 | Imbria Pharmaceuticals, Inc. | Crystal forms of 2-[4-[(2,3,4-trimethoxyphenyl)methyl]piperazin-1-yl]ethyl pyridine-3-carboxylate |
US11883396B2 (en) | 2021-05-03 | 2024-01-30 | Imbria Pharmaceuticals, Inc. | Methods of treating kidney conditions using modified forms of trimetazidine |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS57123180A (en) * | 1980-12-17 | 1982-07-31 | Schering Ag | 3-substituted beta-carboline, manufacture and psychotropic drug containing same |
DE3545776A1 (en) * | 1985-12-20 | 1987-06-25 | Schering Ag | 5-AMINOALKYL-SS-CARBOLINE DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINAL PRODUCTS |
DE3608089A1 (en) * | 1986-03-08 | 1987-09-10 | Schering Ag | HETEROARYL-OXY-SS-CARBOLINE DERIVATIVES, THEIR PRODUCTION AND THEIR USE AS MEDICINAL PRODUCTS |
AU619203B2 (en) * | 1987-08-28 | 1992-01-23 | Schering Aktiengesellschaft | Isoxazole-beta-carboline derivatives |
DE3943225A1 (en) * | 1989-12-23 | 1991-06-27 | Schering Ag | NEW SS CARBOLINE, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE IN MEDICINAL PRODUCTS |
US5350750A (en) * | 1991-04-27 | 1994-09-27 | Schering Aktiengesellschaft | β-carboline-3-hydroxyalkylcarboxylic acid ester derivatives, process for their production and their use in pharmaceutical agents |
DE4118741A1 (en) * | 1991-06-05 | 1992-12-10 | Schering Ag | NEW HETARYLOXY (BETA) CARBOLINES, THEIR PRODUCTION AND USE IN MEDICINAL PRODUCTS |
DE4120109A1 (en) * | 1991-06-15 | 1992-12-17 | Schering Ag | 3-ARYL OR 3-HETARYL (BETA) CARBOLINES, THEIR PRODUCTION AND USE IN MEDICINAL PRODUCTS |
DE4130933A1 (en) * | 1991-09-13 | 1993-03-18 | Schering Ag | NEW (BETA) CARBOLINE DERIVATIVES, THEIR PRODUCTION AND USE IN MEDICINAL PRODUCTS |
DE4212529A1 (en) * | 1992-04-10 | 1993-10-14 | Schering Ag | Use of µ-carbolines as non-competitive glutamate antagonists |
-
1993
- 1993-08-31 DE DE4330175A patent/DE4330175A1/en not_active Withdrawn
-
1994
- 1994-08-22 IL IL11074594A patent/IL110745A0/en unknown
- 1994-08-29 JP JP7507876A patent/JPH09501938A/en active Pending
- 1994-08-29 NZ NZ271615A patent/NZ271615A/en unknown
- 1994-08-29 PL PL94313230A patent/PL313230A1/en unknown
- 1994-08-29 KR KR1019960701006A patent/KR960704888A/en not_active Application Discontinuation
- 1994-08-29 WO PCT/DE1994/001009 patent/WO1995006647A1/en not_active Application Discontinuation
- 1994-08-29 EP EP94925339A patent/EP0716657A1/en not_active Withdrawn
- 1994-08-29 SK SK238-96A patent/SK23896A3/en unknown
- 1994-08-29 CN CN94193211A patent/CN1129938A/en active Pending
- 1994-08-29 CZ CZ96505A patent/CZ50596A3/en unknown
- 1994-08-29 HU HU9600505A patent/HUT73845A/en unknown
- 1994-08-29 AU AU75303/94A patent/AU7530394A/en not_active Abandoned
- 1994-08-29 CA CA002170615A patent/CA2170615A1/en not_active Abandoned
- 1994-08-31 ZA ZA946670A patent/ZA946670B/en unknown
-
1996
- 1996-02-28 FI FI960940A patent/FI960940A0/en not_active Application Discontinuation
- 1996-02-28 NO NO960812A patent/NO960812L/en unknown
Also Published As
Publication number | Publication date |
---|---|
HU9600505D0 (en) | 1996-04-29 |
AU7530394A (en) | 1995-03-22 |
WO1995006647A1 (en) | 1995-03-09 |
SK23896A3 (en) | 1996-11-06 |
CZ50596A3 (en) | 1996-06-12 |
CN1129938A (en) | 1996-08-28 |
JPH09501938A (en) | 1997-02-25 |
IL110745A0 (en) | 1994-11-11 |
EP0716657A1 (en) | 1996-06-19 |
NO960812D0 (en) | 1996-02-28 |
NZ271615A (en) | 1996-09-25 |
NO960812L (en) | 1996-02-28 |
FI960940A0 (en) | 1996-02-28 |
DE4330175A1 (en) | 1995-03-02 |
ZA946670B (en) | 1995-04-21 |
CA2170615A1 (en) | 1995-03-09 |
PL313230A1 (en) | 1996-06-10 |
KR960704888A (en) | 1996-10-09 |
HUT73845A (en) | 1996-09-30 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FD | Application lapsed |