FI953618A0 - Kondensoituneita heterosyklisiä glutamiinijohdannaisia antiproliferatiivisina aineina - Google Patents

Kondensoituneita heterosyklisiä glutamiinijohdannaisia antiproliferatiivisina aineina

Info

Publication number
FI953618A0
FI953618A0 FI953618A FI953618A FI953618A0 FI 953618 A0 FI953618 A0 FI 953618A0 FI 953618 A FI953618 A FI 953618A FI 953618 A FI953618 A FI 953618A FI 953618 A0 FI953618 A0 FI 953618A0
Authority
FI
Finland
Prior art keywords
substituted
compounds
antiproliferative agents
unsubstituted
sulfur
Prior art date
Application number
FI953618A
Other languages
English (en)
Swedish (sv)
Other versions
FI953618A (fi
Inventor
Michael D Varney
Cynthia L Palmer
William H Romines
Original Assignee
Agouron Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Agouron Pharma filed Critical Agouron Pharma
Publication of FI953618A0 publication Critical patent/FI953618A0/fi
Publication of FI953618A publication Critical patent/FI953618A/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyridine Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FI953618A 1993-01-29 1995-07-28 Kondensoituneita heterosyklisiä glutamiinijohdannaisia antiproliferatiivisina aineina FI953618A (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US1086193A 1993-01-29 1993-01-29
PCT/US1994/000418 WO1994017076A1 (en) 1993-01-29 1994-01-18 Condensed heterocyclic glutamic acid derivatives as antiproliferative agents

Publications (2)

Publication Number Publication Date
FI953618A0 true FI953618A0 (fi) 1995-07-28
FI953618A FI953618A (fi) 1995-07-28

Family

ID=21747775

Family Applications (1)

Application Number Title Priority Date Filing Date
FI953618A FI953618A (fi) 1993-01-29 1995-07-28 Kondensoituneita heterosyklisiä glutamiinijohdannaisia antiproliferatiivisina aineina

Country Status (19)

Country Link
EP (2) EP1094066A3 (fi)
JP (1) JPH08505877A (fi)
KR (1) KR100308526B1 (fi)
CN (1) CN1046285C (fi)
AT (1) ATE201877T1 (fi)
AU (1) AU685081B2 (fi)
CA (1) CA2154668C (fi)
DE (1) DE69427394T2 (fi)
DK (1) DK0681584T3 (fi)
ES (1) ES2159551T3 (fi)
FI (1) FI953618A (fi)
GR (1) GR3036506T3 (fi)
HK (1) HK1014715A1 (fi)
NO (1) NO305989B1 (fi)
NZ (1) NZ261497A (fi)
PT (1) PT681584E (fi)
RU (1) RU2127275C1 (fi)
SG (1) SG49234A1 (fi)
WO (1) WO1994017076A1 (fi)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW264475B (fi) * 1991-09-20 1995-12-01 Takeda Pharm Industry Co Ltd
US5831100A (en) * 1995-06-07 1998-11-03 Agouron Pharmaceuticals, Inc. Syntheses of optically pure compounds useful as GARFT inhibitors and their intermediates
US7250464B2 (en) 2000-02-18 2007-07-31 Rohm And Haas Company Distributed paint manufacturing system
WO2002014295A1 (en) * 2000-08-16 2002-02-21 Elena Alexandrovna Izakson Thiazine derivatives having antibacterial and antiviral action
US20040043959A1 (en) * 2002-03-04 2004-03-04 Bloom Laura A. Combination therapies for treating methylthioadenosine phosphorylase deficient cells

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA861235B (en) * 1985-03-08 1986-10-29 Univ Princeton Pyrido(2,3-d)pyrimidine derivatives
EP0438261A3 (en) * 1990-01-16 1992-02-26 Takeda Chemical Industries, Ltd. Condensed heterocyclic glutamic acid derivatives, their production and use

Also Published As

Publication number Publication date
DE69427394T2 (de) 2001-09-20
NO952996D0 (no) 1995-07-28
RU95117099A (ru) 1997-06-27
HK1014715A1 (en) 1999-09-30
ATE201877T1 (de) 2001-06-15
WO1994017076A1 (en) 1994-08-04
EP0681584B1 (en) 2001-06-06
PT681584E (pt) 2001-09-28
CN1046285C (zh) 1999-11-10
CN1117295A (zh) 1996-02-21
EP1094066A2 (en) 2001-04-25
EP1094066A3 (en) 2001-05-02
DE69427394D1 (de) 2001-07-12
EP0681584A1 (en) 1995-11-15
CA2154668A1 (en) 1994-08-04
AU685081B2 (en) 1998-01-15
CA2154668C (en) 2004-12-07
FI953618A (fi) 1995-07-28
ES2159551T3 (es) 2001-10-16
KR100308526B1 (ko) 2001-11-30
RU2127275C1 (ru) 1999-03-10
GR3036506T3 (en) 2001-11-30
NZ261497A (en) 1997-06-24
DK0681584T3 (da) 2001-08-27
AU6026594A (en) 1994-08-15
NO952996L (no) 1995-09-28
JPH08505877A (ja) 1996-06-25
NO305989B1 (no) 1999-08-30
SG49234A1 (en) 1998-05-18

Similar Documents

Publication Publication Date Title
CA2151588A1 (en) Antiproliferative substituted 5-thiapyrimidinone and 5-selenopyrimidinone
EA200100970A1 (ru) Аминопроизводные как ингибиторы протеазы
FI933357A0 (fi) Foerfarande foer framstaellning av benzamider
ATE203234T1 (de) Meta-guanidine, harnstoff, thioharnstoff oder azacyklische aminobenzoesäure-derivate als integrin antagonisten
GR3006247T3 (fi)
ES2164164T3 (es) Derivados de aminotetrazol utiles como inhibidores de oxido nitrico sintasa.
PL309874A1 (en) Novel derivatives of pyrrolocarbasol, method of obtaining them and pharmaceutical composition containing such derivatives
FI953618A (fi) Kondensoituneita heterosyklisiä glutamiinijohdannaisia antiproliferatiivisina aineina
PL293363A1 (en) Method of obtaining novel n-(aryloxyalkyl) heteroaryl-8-aza bicyclo-(3,2,1)-octanes
IS3828A (is) Hliðstæð aðferð til tilreiðslu á nýjum afleiðum thiazolidinone og oxazolidinone sem gagnlegar eru til æðaútvíkkunar
ATE237611T1 (de) Cyclische harnstoff- und lactamderivate von benzo(5,6)cycloheptapyridinen zur verwendung als farnesyl-protein-transferase-hemmer
DK165247C (da) 2,3,4,5-substituerede 1,6-naphthyridinderivater, deres fremstilling samt anvendelse af disse til fremstilling af laegemidler til bekaempelse af cardiale, cerebrale og perifere karlidelser, myocardial iskaemi, cerebral infarkt, lungethrombose, stenoser, arterioscleroser og hjerte-kredsloebslidelser og laegemiddel indeholdende disse derivater
NZ240404A (en) Oxysulphonyl (thio)carbamate derivatives and pharmaceutical
LV10945A (lv) N-(2-amino-2-oksoetil) butandiamida atvasinajumi ka renina inhibitori
ES2149180T3 (es) Derivado de pirazolotiazolopirimidina.

Legal Events

Date Code Title Description
FD Application lapsed